189 related articles for article (PubMed ID: 21084189)
1. Click chemistry inspired one-pot synthesis of 1,4-disubstituted 1,2,3-triazoles and their Src kinase inhibitory activity.
Kumar D; Reddy VB; Kumar A; Mandal D; Tiwari R; Parang K
Bioorg Med Chem Lett; 2011 Jan; 21(1):449-52. PubMed ID: 21084189
[TBL] [Abstract][Full Text] [Related]
2. Synthesis of 1,4-disubstituted 1,2,3-triazole Derivatives Using Click Chemistry and their Src Kinase Activities.
Lebeau A; Abrioux C; Bénimèlis D; Benfodda Z; Meffre P
Med Chem; 2016; 13(1):40-48. PubMed ID: 27041552
[TBL] [Abstract][Full Text] [Related]
3. Discovery of novel purine derivatives with potent and selective inhibitory activity against c-Src tyrosine kinase.
Huang H; Ma J; Shi J; Meng L; Jiang H; Ding J; Liu H
Bioorg Med Chem; 2010 Jul; 18(13):4615-24. PubMed ID: 20570525
[TBL] [Abstract][Full Text] [Related]
4. A facile and one pot synthesis of 1,4-disubstituted-1H-1,2,3-triazoles from terminal alkynes and phenacyl azides prepared from styrenes by CAN oxidant and sodium azide.
Keshavarz M; Badri R
Mol Divers; 2011 Nov; 15(4):957-62. PubMed ID: 21800069
[TBL] [Abstract][Full Text] [Related]
5. Facile one-pot synthesis of 4,5-disubstituted 1,2,3-(NH)-triazoles through Sonogashira coupling/1,3-dipolar cycloaddition of acid chlorides, terminal acetylenes, and sodium azide.
Li J; Wang D; Zhang Y; Li J; Chen B
Org Lett; 2009 Jul; 11(14):3024-7. PubMed ID: 19537825
[TBL] [Abstract][Full Text] [Related]
6. Synthesis and biological evaluation of 1-(6-methylpyridin-2-yl)-5-(quinoxalin-6-yl)-1,2,3-triazoles as transforming growth factor-β type 1 receptor kinase inhibitors.
Li F; Park Y; Hah JM; Ryu JS
Bioorg Med Chem Lett; 2013 Feb; 23(4):1083-6. PubMed ID: 23294702
[TBL] [Abstract][Full Text] [Related]
7. Click chemistry inspired synthesis of morpholine-fused triazoles.
Mishra KB; Tiwari VK
J Org Chem; 2014 Jun; 79(12):5752-62. PubMed ID: 24845771
[TBL] [Abstract][Full Text] [Related]
8. Click approach to the discovery of 1,2,3-triazolylsalicylamides as potent Aurora kinase inhibitors.
Song D; Park Y; Yoon J; Aman W; Hah JM; Ryu JS
Bioorg Med Chem; 2014 Sep; 22(17):4855-66. PubMed ID: 25042560
[TBL] [Abstract][Full Text] [Related]
9. Diamino-1,2,4-triazole derivatives are selective inhibitors of TYK2 and JAK1 over JAK2 and JAK3.
Malerich JP; Lam JS; Hart B; Fine RM; Klebansky B; Tanga MJ; D'Andrea A
Bioorg Med Chem Lett; 2010 Dec; 20(24):7454-7. PubMed ID: 21106455
[TBL] [Abstract][Full Text] [Related]
10. Synthesis of 3-phenylpyrazolopyrimidine-1,2,3-triazole conjugates and evaluation of their Src kinase inhibitory and anticancer activities.
Kumar A; Ahmad I; Chhikara BS; Tiwari R; Mandal D; Parang K
Bioorg Med Chem Lett; 2011 Mar; 21(5):1342-6. PubMed ID: 21300544
[TBL] [Abstract][Full Text] [Related]
11. ZINClick: a database of 16 million novel, patentable, and readily synthesizable 1,4-disubstituted triazoles.
Massarotti A; Brunco A; Sorba G; Tron GC
J Chem Inf Model; 2014 Feb; 54(2):396-406. PubMed ID: 24451008
[TBL] [Abstract][Full Text] [Related]
12. Rapid preparation of triazolyl substituted NH-heterocyclic kinase inhibitors via one-pot Sonogashira coupling-TMS-deprotection-CuAAC sequence.
Merkul E; Klukas F; Dorsch D; Grädler U; Greiner HE; Müller TJ
Org Biomol Chem; 2011 Jul; 9(14):5129-36. PubMed ID: 21625704
[TBL] [Abstract][Full Text] [Related]
13. Ynamide Click chemistry in development of triazole VEGFR2 TK modulators.
Vojtičková M; Dobiaš J; Hanquet G; Addová G; Cetin-Atalay R; Yildirim DC; Boháč A
Eur J Med Chem; 2015 Oct; 103():105-22. PubMed ID: 26344911
[TBL] [Abstract][Full Text] [Related]
14. Exploration of acridine scaffold as a potentially interesting scaffold for discovering novel multi-target VEGFR-2 and Src kinase inhibitors.
Luan X; Gao C; Zhang N; Chen Y; Sun Q; Tan C; Liu H; Jin Y; Jiang Y
Bioorg Med Chem; 2011 Jun; 19(11):3312-9. PubMed ID: 21576023
[TBL] [Abstract][Full Text] [Related]
15. 'Click' synthesis of a triazole-based inhibitor of Met functions in cancer cells.
Colombo F; Tintori C; Furlan A; Borrelli S; Christodoulou MS; Dono R; Maina F; Botta M; Amat M; Bosch J; Passarella D
Bioorg Med Chem Lett; 2012 Jul; 22(14):4693-6. PubMed ID: 22738633
[TBL] [Abstract][Full Text] [Related]
16. Synthesis and structure-activity relationships of 4-fluorophenyl-imidazole p38α MAPK, CK1δ and JAK2 kinase inhibitors.
Seerden JP; Leusink-Ionescu G; Woudenberg-Vrenken T; Dros B; Molema G; Kamps JA; Kellogg RM
Bioorg Med Chem Lett; 2014 Aug; 24(15):3412-8. PubMed ID: 24930833
[TBL] [Abstract][Full Text] [Related]
17. Alkyne-azide click chemistry mediated carbanucleosides synthesis.
Broggi J; Joubert N; Aucagne V; Berteina-Raboin S; Diez-Gonzalez S; Nolan S; Topalis D; Deville-Bonne D; Balzarini J; Neyts J; Andrei G; Snoeck R; Agrofoglio LA
Nucleosides Nucleotides Nucleic Acids; 2007; 26(10-12):1391-4. PubMed ID: 18066789
[TBL] [Abstract][Full Text] [Related]
18. One-pot synthesis of 1,4-disubstituted 1,2,3-triazoles from in situ generated azides.
Feldman AK; Colasson B; Fokin VV
Org Lett; 2004 Oct; 6(22):3897-9. PubMed ID: 15496058
[TBL] [Abstract][Full Text] [Related]
19. Synthesis and evaluation of 3-phenylpyrazolo[3,4-d]pyrimidine-peptide conjugates as Src kinase inhibitors.
Kumar A; Wang Y; Lin X; Sun G; Parang K
ChemMedChem; 2007 Sep; 2(9):1346-60. PubMed ID: 17530729
[TBL] [Abstract][Full Text] [Related]
20. Design, synthesis and characterization of "clickable" 4-anilinoquinazoline kinase inhibitors.
Perera BG; Maly DJ
Mol Biosyst; 2008 Jun; 4(6):542-50. PubMed ID: 18493651
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]
