369 related articles for article (PubMed ID: 21141892)
1. Antimalarial activity of novel 5-aryl-8-aminoquinoline derivatives.
Shiraki H; Kozar MP; Melendez V; Hudson TH; Ohrt C; Magill AJ; Lin AJ
J Med Chem; 2011 Jan; 54(1):131-42. PubMed ID: 21141892
[TBL] [Abstract][Full Text] [Related]
2. 4-Aminoquinoline quinolizidinyl- and quinolizidinylalkyl-derivatives with antimalarial activity.
Sparatore A; Basilico N; Parapini S; Romeo S; Novelli F; Sparatore F; Taramelli D
Bioorg Med Chem; 2005 Sep; 13(18):5338-45. PubMed ID: 16054368
[TBL] [Abstract][Full Text] [Related]
3. Antimalarial activity of novel pyrrolizidinyl derivatives of 4-aminoquinoline.
Sparatore A; Basilico N; Casagrande M; Parapini S; Taramelli D; Brun R; Wittlin S; Sparatore F
Bioorg Med Chem Lett; 2008 Jul; 18(13):3737-40. PubMed ID: 18538567
[TBL] [Abstract][Full Text] [Related]
4. Synthesis, antimalarial activity, and cellular toxicity of new arylpyrrolylaminoquinolines.
Casagrande M; Basilico N; Rusconi C; Taramelli D; Sparatore A
Bioorg Med Chem; 2010 Sep; 18(18):6625-33. PubMed ID: 20797868
[TBL] [Abstract][Full Text] [Related]
5. Antiplasmodial activity of new 4-aminoquinoline derivatives against chloroquine resistant strain.
Sinha M; Dola VR; Agarwal P; Srivastava K; Haq W; Puri SK; Katti SB
Bioorg Med Chem; 2014 Jul; 22(14):3573-86. PubMed ID: 24906512
[TBL] [Abstract][Full Text] [Related]
6. 4-Aminoquinoline derivatives: Synthesis, in vitro and in vivo antiplasmodial activity against chloroquine-resistant parasites.
Singh S; Agarwal D; Sharma K; Sharma M; Nielsen MA; Alifrangis M; Singh AK; Gupta RD; Awasthi SK
Eur J Med Chem; 2016 Oct; 122():394-407. PubMed ID: 27394399
[TBL] [Abstract][Full Text] [Related]
7. Synthesis and bioevaluation of novel 4-aminoquinoline-tetrazole derivatives as potent antimalarial agents.
Pandey S; Agarwal P; Srivastava K; Rajakumar S; Puri SK; Verma P; Saxena JK; Sharma A; Lal J; Chauhan PM
Eur J Med Chem; 2013 Aug; 66():69-81. PubMed ID: 23792317
[TBL] [Abstract][Full Text] [Related]
8. Incorporation of a 3-(2,2,2-trifluoroethyl)-γ-hydroxy-γ-lactam motif in the side chain of 4-aminoquinolines. Syntheses and antimalarial activities.
Cornut D; Lemoine H; Kanishchev O; Okada E; Albrieux F; Beavogui AH; Bienvenu AL; Picot S; Bouillon JP; Médebielle M
J Med Chem; 2013 Jan; 56(1):73-83. PubMed ID: 23102258
[TBL] [Abstract][Full Text] [Related]
9. Synthesis of oxalamide and triazine derivatives as a novel class of hybrid 4-aminoquinoline with potent antiplasmodial activity.
Sunduru N; Sharma M; Srivastava K; Rajakumar S; Puri SK; Saxena JK; Chauhan PM
Bioorg Med Chem; 2009 Sep; 17(17):6451-62. PubMed ID: 19665899
[TBL] [Abstract][Full Text] [Related]
10. Synthesis of ring-substituted 4-aminoquinolines and evaluation of their antimalarial activities.
Madrid PB; Sherrill J; Liou AP; Weisman JL; Derisi JL; Guy RK
Bioorg Med Chem Lett; 2005 Feb; 15(4):1015-8. PubMed ID: 15686903
[TBL] [Abstract][Full Text] [Related]
11. Synthesis and antiplasmodial activity of new heteroaryl derivatives of 7-chloro-4-aminoquinoline.
Casagrande M; Barteselli A; Basilico N; Parapini S; Taramelli D; Sparatore A
Bioorg Med Chem; 2012 Oct; 20(19):5965-79. PubMed ID: 22917857
[TBL] [Abstract][Full Text] [Related]
12. Synthesis and antimalarial activity of side chain modified 4-aminoquinoline derivatives.
Solomon VR; Haq W; Srivastava K; Puri SK; Katti SB
J Med Chem; 2007 Jan; 50(2):394-8. PubMed ID: 17228883
[TBL] [Abstract][Full Text] [Related]
13. 4-aminoquinoline-triazine-based hybrids with improved in vitro antimalarial activity against CQ-sensitive and CQ-resistant strains of Plasmodium falciparum.
Manohar S; Khan SI; Rawat DS
Chem Biol Drug Des; 2013 May; 81(5):625-30. PubMed ID: 23331618
[TBL] [Abstract][Full Text] [Related]
14. Optimization of 4-aminoquinoline/clotrimazole-based hybrid antimalarials: further structure-activity relationships, in vivo studies, and preliminary toxicity profiling.
Gemma S; Camodeca C; Sanna Coccone S; Joshi BP; Bernetti M; Moretti V; Brogi S; Bonache de Marcos MC; Savini L; Taramelli D; Basilico N; Parapini S; Rottmann M; Brun R; Lamponi S; Caccia S; Guiso G; Summers RL; Martin RE; Saponara S; Gorelli B; Novellino E; Campiani G; Butini S
J Med Chem; 2012 Aug; 55(15):6948-67. PubMed ID: 22783984
[TBL] [Abstract][Full Text] [Related]
15. Antimalarial dual drugs based on potent inhibitors of glutathione reductase from Plasmodium falciparum.
Friebolin W; Jannack B; Wenzel N; Furrer J; Oeser T; Sanchez CP; Lanzer M; Yardley V; Becker K; Davioud-Charvet E
J Med Chem; 2008 Mar; 51(5):1260-77. PubMed ID: 18260613
[TBL] [Abstract][Full Text] [Related]
16. Antimalarial activities of new guanidylimidazole and guanidylimidazoline derivatives.
Zhang L; Sathunuru R; Caridha D; Pybus B; O'Neil MT; Kozar MP; Lin AJ
J Med Chem; 2011 Oct; 54(19):6634-46. PubMed ID: 21848332
[TBL] [Abstract][Full Text] [Related]
17. Synthesis and evaluation of sulfonylurea derivatives as novel antimalarials.
León C; Rodrigues J; Gamboa de Domínguez N; Charris J; Gut J; Rosenthal PJ; Domínguez JN
Eur J Med Chem; 2007 Jun; 42(6):735-42. PubMed ID: 17321641
[TBL] [Abstract][Full Text] [Related]
18. Plasmodium berghei: dehydroepiandrosterone sulfate reverses chloroquino-resistance in experimental malaria infection; correlation with glucose 6-phosphate dehydrogenase and glutathione synthesis pathway.
Safeukui I; Mangou F; Malvy D; Vincendeau P; Mossalayi D; Haumont G; Vatan R; Olliaro P; Millet P
Biochem Pharmacol; 2004 Nov; 68(10):1903-10. PubMed ID: 15476661
[TBL] [Abstract][Full Text] [Related]
19. Synthesis and antimalarial activity in vitro and in vivo of a new ferrocene-chloroquine analogue.
Biot C; Glorian G; Maciejewski LA; Brocard JS
J Med Chem; 1997 Nov; 40(23):3715-8. PubMed ID: 9371235
[TBL] [Abstract][Full Text] [Related]
20. Synthesis, antimalarial activity and cytotoxicity of 4-aminoquinoline-triazine conjugates.
Manohar S; Khan SI; Rawat DS
Bioorg Med Chem Lett; 2010 Jan; 20(1):322-5. PubMed ID: 19910192
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]