These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.


BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

246 related articles for article (PubMed ID: 21162558)

  • 1. The antimalarial ferroquine: role of the metal and intramolecular hydrogen bond in activity and resistance.
    Dubar F; Egan TJ; Pradines B; Kuter D; Ncokazi KK; Forge D; Paul JF; Pierrot C; Kalamou H; Khalife J; Buisine E; Rogier C; Vezin H; Forfar I; Slomianny C; Trivelli X; Kapishnikov S; Leiserowitz L; Dive D; Biot C
    ACS Chem Biol; 2011 Mar; 6(3):275-87. PubMed ID: 21162558
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Opening up the advantages of the ruthenocenic bioprobes of ferroquine: distribution and localization in Plasmodium falciparum-infected erythrocytes.
    Biot C; Dubar F; Khalife J; Slomianny C
    Metallomics; 2012 Aug; 4(8):780-3. PubMed ID: 22700030
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Assessment of Plasmodium falciparum resistance to ferroquine (SSR97193) in field isolates and in W2 strain under pressure.
    Daher W; Biot C; Fandeur T; Jouin H; Pelinski L; Viscogliosi E; Fraisse L; Pradines B; Brocard J; Khalife J; Dive D
    Malar J; 2006 Feb; 5():11. PubMed ID: 16464254
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Insights into the mechanism of action of ferroquine. Relationship between physicochemical properties and antiplasmodial activity.
    Biot C; Taramelli D; Forfar-Bares I; Maciejewski LA; Boyce M; Nowogrocki G; Brocard JS; Basilico N; Olliaro P; Egan TJ
    Mol Pharm; 2005; 2(3):185-93. PubMed ID: 15934779
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Probing the role of the covalent linkage of ferrocene into a chloroquine template.
    Biot C; Daher W; Ndiaye CM; Melnyk P; Pradines B; Chavain N; Pellet A; Fraisse L; Pelinski L; Jarry C; Brocard J; Khalife J; Forfar-Bares I; Dive D
    J Med Chem; 2006 Jul; 49(15):4707-14. PubMed ID: 16854077
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Design, Synthesis, and Evaluation of Novel Ferroquine and Phenylequine Analogues as Potential Antiplasmodial Agents.
    Jacobs L; de Kock C; de Villiers KA; Smith PJ; Smith VJ; van Otterlo WA; Blackie MA
    ChemMedChem; 2015 Dec; 10(12):2099-110. PubMed ID: 26447782
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Trioxaferroquines as new hybrid antimalarial drugs.
    Bellot F; Coslédan F; Vendier L; Brocard J; Meunier B; Robert A
    J Med Chem; 2010 May; 53(10):4103-9. PubMed ID: 20443628
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Metallocene-based antimalarials: an exploration into the influence of the ferrocenyl moiety on in vitro antimalarial activity in chloroquine-sensitive and chloroquine-resistant strains of Plasmodium falciparum.
    Blackie MA; Beagley P; Croft SL; Kendrick H; Moss JR; Chibale K
    Bioorg Med Chem; 2007 Oct; 15(20):6510-6. PubMed ID: 17693090
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Investigation of the redox behavior of ferroquine, a new antimalarial.
    Chavain N; Vezin H; Dive D; Touati N; Paul JF; Buisine E; Biot C
    Mol Pharm; 2008; 5(5):710-6. PubMed ID: 18563912
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Design, synthesis, and antimalarial activity of structural chimeras of thiosemicarbazone and ferroquine analogues.
    Biot C; Pradines B; Sergeant MH; Gut J; Rosenthal PJ; Chibale K
    Bioorg Med Chem Lett; 2007 Dec; 17(23):6434-8. PubMed ID: 17949976
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Synthesis and antimalarial activities of rhenium bioorganometallics based on the 4-aminoquinoline structure.
    Arancibia R; Dubar F; Pradines B; Forfar I; Dive D; Klahn AH; Biot C
    Bioorg Med Chem; 2010 Nov; 18(22):8085-91. PubMed ID: 20934349
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Structural characteristics of chloroquine-bridged ferrocenophane analogues of ferroquine may obviate malaria drug-resistance mechanisms.
    Salas PF; Herrmann C; Cawthray JF; Nimphius C; Kenkel A; Chen J; de Kock C; Smith PJ; Patrick BO; Adam MJ; Orvig C
    J Med Chem; 2013 Feb; 56(4):1596-613. PubMed ID: 23327489
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Ferroquine, an ingenious antimalarial drug: thoughts on the mechanism of action.
    Dubar F; Khalife J; Brocard J; Dive D; Biot C
    Molecules; 2008 Nov; 13(11):2900-7. PubMed ID: 19020475
    [TBL] [Abstract][Full Text] [Related]  

  • 14. In vitro activity of ferroquine is independent of polymorphisms in transport protein genes implicated in quinoline resistance in Plasmodium falciparum.
    Henry M; Briolant S; Fontaine A; Mosnier J; Baret E; Amalvict R; Fusaï T; Fraisse L; Rogier C; Pradines B
    Antimicrob Agents Chemother; 2008 Aug; 52(8):2755-9. PubMed ID: 18505855
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Antimalarial activities of ferroquine conjugates with either glutathione reductase inhibitors or glutathione depletors via a hydrolyzable amide linker.
    Chavain N; Davioud-Charvet E; Trivelli X; Mbeki L; Rottmann M; Brun R; Biot C
    Bioorg Med Chem; 2009 Dec; 17(23):8048-59. PubMed ID: 19864147
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Synthesis, antimalarial activity, and cellular toxicity of new arylpyrrolylaminoquinolines.
    Casagrande M; Basilico N; Rusconi C; Taramelli D; Sparatore A
    Bioorg Med Chem; 2010 Sep; 18(18):6625-33. PubMed ID: 20797868
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Activity of piperaquine and other 4-aminoquinoline antiplasmodial drugs against chloroquine-sensitive and resistant blood-stages of Plasmodium falciparum. Role of beta-haematin inhibition and drug concentration in vacuolar water- and lipid-phases.
    Warhurst DC; Craig JC; Adagu IS; Guy RK; Madrid PB; Fivelman QL
    Biochem Pharmacol; 2007 Jun; 73(12):1910-26. PubMed ID: 17466277
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Synthesis and antimalarial activity of side chain modified 4-aminoquinoline derivatives.
    Solomon VR; Haq W; Srivastava K; Puri SK; Katti SB
    J Med Chem; 2007 Jan; 50(2):394-8. PubMed ID: 17228883
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Antimalarial versus cytotoxic properties of dual drugs derived from 4-aminoquinolines and Mannich bases: interaction with DNA.
    Wenzel NI; Chavain N; Wang Y; Friebolin W; Maes L; Pradines B; Lanzer M; Yardley V; Brun R; Herold-Mende C; Biot C; Tóth K; Davioud-Charvet E
    J Med Chem; 2010 Apr; 53(8):3214-26. PubMed ID: 20329733
    [TBL] [Abstract][Full Text] [Related]  

  • 20. In vitro activity of ferroquine (SAR97193) is independent of chloroquine resistance in Plasmodium falciparum.
    Kreidenweiss A; Kremsner PG; Dietz K; Mordmüller B
    Am J Trop Med Hyg; 2006 Dec; 75(6):1178-81. PubMed ID: 17172389
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 13.