249 related articles for article (PubMed ID: 21185180)
1. Design, synthesis and antibacterial activity of 3-methylenepyrrolidine formyl hydroxyamino derivatives as novel peptide deformylase inhibitors.
Shi W; Ma H; Duan Y; Aubart K; Fang Y; Zonis R; Yang L; Hu W
Bioorg Med Chem Lett; 2011 Feb; 21(3):1060-3. PubMed ID: 21185180
[TBL] [Abstract][Full Text] [Related]
2. Synthesis, antibacterial activity, and biological evaluation of formyl hydroxyamino derivatives as novel potent peptide deformylase inhibitors against drug-resistant bacteria.
Yang S; Shi W; Xing D; Zhao Z; Lv F; Yang L; Yang Y; Hu W
Eur J Med Chem; 2014 Oct; 86():133-52. PubMed ID: 25151577
[TBL] [Abstract][Full Text] [Related]
3. Design, synthesis, and antibacterial activity of 2,5-dihydropyrrole formyl hydroxyamino derivatives as novel peptide deformylase inhibitors.
Shi W; Duan Y; Qian Y; Li M; Yang L; Hu W
Bioorg Med Chem Lett; 2010 Jun; 20(12):3592-5. PubMed ID: 20510610
[TBL] [Abstract][Full Text] [Related]
4. Peptide deformylase inhibitors with retro-amide scaffold: synthesis and structure-activity relationships.
Lee SK; Choi KH; Lee SJ; Suh SW; Kim BM; Lee BJ
Bioorg Med Chem Lett; 2010 Aug; 20(15):4317-9. PubMed ID: 20615695
[TBL] [Abstract][Full Text] [Related]
5. In vitro antibacterial activity of the peptide deformylase inhibitor BB-83698.
Lofland D; Difuntorum S; Waller A; Clements JM; Weaver MK; Karlowsky JA; Johnson K
J Antimicrob Chemother; 2004 Apr; 53(4):664-8. PubMed ID: 14973152
[TBL] [Abstract][Full Text] [Related]
6. Peptide deformylase inhibitors with non-peptide scaffold: synthesis and structure-activity relationships.
Lee SK; Choi KH; Lee SJ; Lee JS; Park JY; Kim BM; Lee BJ
Bioorg Med Chem Lett; 2011 Jan; 21(1):133-6. PubMed ID: 21146987
[TBL] [Abstract][Full Text] [Related]
7. Synthesis and antibacterial activity of novel 4''-carbamates of 6,11-di-O-methylerythromycin A.
Wu Z; Lu Y; Luo M; He X; Xiao Y; Yang J; Pan Y; Qiu G; Xu Y; Huang W; Long P; Li R; Hu X
J Antibiot (Tokyo); 2010 Jul; 63(7):343-50. PubMed ID: 20448668
[TBL] [Abstract][Full Text] [Related]
8. Peptidomimetic inhibitors of bacterial peptide deformylase.
East SP; Ayscough A; Toogood-Johnson I; Taylor S; Thomas W
Bioorg Med Chem Lett; 2011 Jul; 21(13):4032-5. PubMed ID: 21621999
[TBL] [Abstract][Full Text] [Related]
9. Design, synthesis, and antibacterial activities of novel 3,6-bicyclolide oximes: length optimization and zero carbon linker oximes.
Tang D; Gai Y; Polemeropoulos A; Chen Z; Wang Z; Or YS
Bioorg Med Chem Lett; 2008 Sep; 18(18):5078-82. PubMed ID: 18762418
[TBL] [Abstract][Full Text] [Related]
10. Synthesis and preliminary antibacterial evaluation of 2-butyl succinate-based hydroxamate derivatives containing isoxazole rings.
Zhang D; Jia J; Meng L; Xu W; Tang L; Wang J
Arch Pharm Res; 2010 Jun; 33(6):831-42. PubMed ID: 20607487
[TBL] [Abstract][Full Text] [Related]
11. Exploration of the activity of 7-pyrrolidino-8-methoxyisothiazoloquinolones against methicillin-resistant Staphylococcus aureus (MRSA).
Kim HY; Wiles JA; Wang Q; Pais GC; Lucien E; Hashimoto A; Nelson DM; Thanassi JA; Podos SD; Deshpande M; Pucci MJ; Bradbury BJ
J Med Chem; 2011 May; 54(9):3268-82. PubMed ID: 21425851
[TBL] [Abstract][Full Text] [Related]
12. N-heterocyclic dicarboxylic acids: broad-spectrum inhibitors of metallo-β-lactamases with co-antibacterial effect against antibiotic-resistant bacteria.
Feng L; Yang KW; Zhou LS; Xiao JM; Yang X; Zhai L; Zhang YL; Crowder MW
Bioorg Med Chem Lett; 2012 Aug; 22(16):5185-9. PubMed ID: 22796180
[TBL] [Abstract][Full Text] [Related]
13. Design, synthesis and structure-activity relationship studies of novel indazole analogues as DNA gyrase inhibitors with Gram-positive antibacterial activity.
Tanitame A; Oyamada Y; Ofuji K; Kyoya Y; Suzuki K; Ito H; Kawasaki M; Nagai K; Wachi M; Yamagishi J
Bioorg Med Chem Lett; 2004 Jun; 14(11):2857-62. PubMed ID: 15125947
[TBL] [Abstract][Full Text] [Related]
14. Discovery of 4-Pyridone derivatives as specific inhibitors of enoyl-acyl carrier protein reductase (FabI) with antibacterial activity against Staphylococcus aureus.
Takahata S; Iida M; Yoshida T; Kumura K; Kitagawa H; Hoshiko S
J Antibiot (Tokyo); 2007 Feb; 60(2):123-8. PubMed ID: 17420562
[TBL] [Abstract][Full Text] [Related]
15. Synthesis and SAR study of novel 7-(pyridinium-3-yl)-carbonyl imidazo[5,1-b]thiazol-2-yl carbapenems.
Maruyama T; Kano Y; Yamamoto Y; Kurazono M; Iwamatsu K; Atsumi K; Shitara E
Bioorg Med Chem; 2007 Jan; 15(1):392-402. PubMed ID: 17055731
[TBL] [Abstract][Full Text] [Related]
16. Synthesis and in vitro antibacterial activity of (2S)-N-(substitutedphenyl)-1-[(2R)-2-[(formylhydroxyamino)methyl]-1-oxohexyl]-2-pyrrolidinecarboxamides as potential peptide deformylase inhibitors.
Wang Z; Zhou W
Chem Biol Drug Des; 2009 Jan; 73(1):142-6. PubMed ID: 19152643
[TBL] [Abstract][Full Text] [Related]
17. Structure-activity relationship analysis and therapeutic potential of peptide deformylase inhibitors.
Boularot A; Giglione C; Artaud I; Meinnel T
Curr Opin Investig Drugs; 2004 Aug; 5(8):809-22. PubMed ID: 15600237
[TBL] [Abstract][Full Text] [Related]
18. Structures of Staphylococcus aureus peptide deformylase in complex with two classes of new inhibitors.
Lee SJ; Lee SJ; Lee SK; Yoon HJ; Lee HH; Kim KK; Lee BJ; Lee BI; Suh SW
Acta Crystallogr D Biol Crystallogr; 2012 Jul; 68(Pt 7):784-93. PubMed ID: 22751663
[TBL] [Abstract][Full Text] [Related]
19. Synthesis and antibacterial activity of C-12 pyrazolinyl spiro ketolides.
Hu L; Lan P; Song QL; Huang ZJ; Sun PH; Zhuo C; Wang Y; Xiao S; Chen WM
Eur J Med Chem; 2010 Dec; 45(12):5943-9. PubMed ID: 20970894
[TBL] [Abstract][Full Text] [Related]
20. Design, synthesis, and antibacterial activity of demethylvancomycin analogues against drug-resistant bacteria.
Chang J; Zhang SJ; Jiang YW; Xu L; Yu JM; Zhou WJ; Sun X
ChemMedChem; 2013 Jun; 8(6):976-84. PubMed ID: 23576378
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]
