121 related articles for article (PubMed ID: 21239511)
1. Characterization of highly efficacious allosteric agonists of the human calcium-sensing receptor.
Ma JN; Owens M; Gustafsson M; Jensen J; Tabatabaei A; Schmelzer K; Olsson R; Burstein ES
J Pharmacol Exp Ther; 2011 Apr; 337(1):275-84. PubMed ID: 21239511
[TBL] [Abstract][Full Text] [Related]
2. Discovery of a class of calcium sensing receptor positive allosteric modulators; 1-(benzothiazol-2-yl)-1-phenylethanols.
Gustafsson M; Jensen J; Bertozzi SM; Currier EA; Ma JN; Burstein ES; Olsson R
Bioorg Med Chem Lett; 2010 Oct; 20(19):5918-21. PubMed ID: 20727747
[TBL] [Abstract][Full Text] [Related]
3. Identification and characterization of novel small-molecule protease-activated receptor 2 agonists.
Gardell LR; Ma JN; Seitzberg JG; Knapp AE; Schiffer HH; Tabatabaei A; Davis CN; Owens M; Clemons B; Wong KK; Lund B; Nash NR; Gao Y; Lameh J; Schmelzer K; Olsson R; Burstein ES
J Pharmacol Exp Ther; 2008 Dec; 327(3):799-808. PubMed ID: 18768780
[TBL] [Abstract][Full Text] [Related]
4. Pharmacology of AMG 416 (Velcalcetide), a novel peptide agonist of the calcium-sensing receptor, for the treatment of secondary hyperparathyroidism in hemodialysis patients.
Walter S; Baruch A; Dong J; Tomlinson JE; Alexander ST; Janes J; Hunter T; Yin Q; Maclean D; Bell G; Mendel DB; Johnson RM; Karim F
J Pharmacol Exp Ther; 2013 Aug; 346(2):229-40. PubMed ID: 23674604
[TBL] [Abstract][Full Text] [Related]
5. Impact of clinically relevant mutations on the pharmacoregulation and signaling bias of the calcium-sensing receptor by positive and negative allosteric modulators.
Leach K; Wen A; Cook AE; Sexton PM; Conigrave AD; Christopoulos A
Endocrinology; 2013 Mar; 154(3):1105-16. PubMed ID: 23372019
[TBL] [Abstract][Full Text] [Related]
6. [Basic and clinical aspects of calcimimetics. Structure and function of calcium-sensing receptor].
Fukumoto S
Clin Calcium; 2008 Jan; 18(1):32-6. PubMed ID: 18175869
[TBL] [Abstract][Full Text] [Related]
7. Recent updates on the calcium-sensing receptor as a drug target.
Trivedi R; Mithal A; Chattopadhyay N
Curr Med Chem; 2008; 15(2):178-86. PubMed ID: 18220773
[TBL] [Abstract][Full Text] [Related]
8. The pathophysiology of primary hyperparathyroidism.
Brown EM
J Bone Miner Res; 2002 Nov; 17 Suppl 2():N24-9. PubMed ID: 12412774
[TBL] [Abstract][Full Text] [Related]
9. [Basic and clinical aspects of calcimimetics. Discovery and development of calcimimetics].
Nagano N
Clin Calcium; 2008 Jan; 18(1):37-44. PubMed ID: 18175870
[TBL] [Abstract][Full Text] [Related]
10. Design and synthesis of calindol derivatives as potent and selective calcium sensing receptor agonists.
Kiefer L; Beaumard F; Gorojankina T; Faure H; Ruat M; Dodd RH
Bioorg Med Chem; 2016 Feb; 24(4):554-69. PubMed ID: 26752095
[TBL] [Abstract][Full Text] [Related]
11. Activation of calcium-sensing receptor by allosteric agonists cinacalcet and AC-265347 abolishes the 1,25(OH)
Wongdee K; Rodrat M; Keadsai C; Jantarajit W; Teerapornpuntakit J; Thongbunchoo J; Charoenphandhu N
Arch Biochem Biophys; 2018 Nov; 657():15-22. PubMed ID: 30217510
[TBL] [Abstract][Full Text] [Related]
12. Role of the calcium-sensing receptor in parathyroid gland physiology.
Chen RA; Goodman WG
Am J Physiol Renal Physiol; 2004 Jun; 286(6):F1005-11. PubMed ID: 15130894
[TBL] [Abstract][Full Text] [Related]
13. Extracellular calcium-sensing receptors in fishes.
Loretz CA
Comp Biochem Physiol A Mol Integr Physiol; 2008 Mar; 149(3):225-45. PubMed ID: 18302989
[TBL] [Abstract][Full Text] [Related]
14. ADX47273 [S-(4-fluoro-phenyl)-{3-[3-(4-fluoro-phenyl)-[1,2,4]-oxadiazol-5-yl]-piperidin-1-yl}-methanone]: a novel metabotropic glutamate receptor 5-selective positive allosteric modulator with preclinical antipsychotic-like and procognitive activities.
Liu F; Grauer S; Kelley C; Navarra R; Graf R; Zhang G; Atkinson PJ; Popiolek M; Wantuch C; Khawaja X; Smith D; Olsen M; Kouranova E; Lai M; Pruthi F; Pulicicchio C; Day M; Gilbert A; Pausch MH; Brandon NJ; Beyer CE; Comery TA; Logue S; Rosenzweig-Lipson S; Marquis KL
J Pharmacol Exp Ther; 2008 Dec; 327(3):827-39. PubMed ID: 18753411
[TBL] [Abstract][Full Text] [Related]
15. L-type amino acids stimulate gastric acid secretion by activation of the calcium-sensing receptor in parietal cells.
Busque SM; Kerstetter JE; Geibel JP; Insogna K
Am J Physiol Gastrointest Liver Physiol; 2005 Oct; 289(4):G664-9. PubMed ID: 15961860
[TBL] [Abstract][Full Text] [Related]
16. Calcium-sensing receptor regulation of PTH-dependent calcium absorption by mouse cortical ascending limbs.
Motoyama HI; Friedman PA
Am J Physiol Renal Physiol; 2002 Sep; 283(3):F399-406. PubMed ID: 12167589
[TBL] [Abstract][Full Text] [Related]
17. The calcium-sensing receptor in taste tissue.
San Gabriel A; Uneyama H; Maekawa T; Torii K
Biochem Biophys Res Commun; 2009 Jan; 378(3):414-8. PubMed ID: 19056349
[TBL] [Abstract][Full Text] [Related]
18. The M1 muscarinic receptor allosteric agonists AC-42 and 1-[1'-(2-methylbenzyl)-1,4'-bipiperidin-4-yl]-1,3-dihydro-2H-benzimidazol-2-one bind to a unique site distinct from the acetylcholine orthosteric site.
Jacobson MA; Kreatsoulas C; Pascarella DM; O'Brien JA; Sur C
Mol Pharmacol; 2010 Oct; 78(4):648-57. PubMed ID: 20660086
[TBL] [Abstract][Full Text] [Related]
19. Biased allosteric modulation at the CaS receptor engendered by structurally diverse calcimimetics.
Cook AE; Mistry SN; Gregory KJ; Furness SG; Sexton PM; Scammells PJ; Conigrave AD; Christopoulos A; Leach K
Br J Pharmacol; 2015 Jan; 172(1):185-200. PubMed ID: 25220431
[TBL] [Abstract][Full Text] [Related]
20. Pharmacological characterization of a new, orally active and potent allosteric metabotropic glutamate receptor 1 antagonist, 4-[1-(2-fluoropyridin-3-yl)-5-methyl-1H-1,2,3-triazol-4-yl]-N-isopropyl-N-methyl-3,6-dihydropyridine-1(2H)-carboxamide (FTIDC).
Suzuki G; Kimura T; Satow A; Kaneko N; Fukuda J; Hikichi H; Sakai N; Maehara S; Kawagoe-Takaki H; Hata M; Azuma T; Ito S; Kawamoto H; Ohta H
J Pharmacol Exp Ther; 2007 Jun; 321(3):1144-53. PubMed ID: 17360958
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]
