These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.
195 related articles for article (PubMed ID: 21351438)
1. [Design, synthesis of quinolinone acid-containing compounds with anti-HIV integrase activity]. Chen XF; Wu YB; Jin J; Wang RZ; Wang C; Liu J Yao Xue Xue Bao; 2010 Feb; 45(2):263-7. PubMed ID: 21351438 [TBL] [Abstract][Full Text] [Related]
2. Synthesis, biological evaluation and molecular modeling studies of quinolonyl diketo acid derivatives: new structural insight into the HIV-1 integrase inhibition. Vandurm P; Guiguen A; Cauvin C; Georges B; Le Van K; Michaux C; Cardona C; Mbemba G; Mouscadet JF; Hevesi L; Van Lint C; Wouters J Eur J Med Chem; 2011 May; 46(5):1749-56. PubMed ID: 21385662 [TBL] [Abstract][Full Text] [Related]
3. Design and synthesis of novel nitrogen-containing polyhydroxylated aromatics as HIV-1 integrase inhibitors from caffeic acid phenethyl ester. Wang P; Liu C; Sanches T; Zhong Y; Liu B; Xiong J; Neamati N; Zhao G Bioorg Med Chem Lett; 2009 Aug; 19(16):4574-8. PubMed ID: 19625188 [TBL] [Abstract][Full Text] [Related]
4. Synthesis and biological evaluation of HQCAs with aryl or benzyl substituents on N-1 position as potential HIV-1 integrase inhibitors. He QQ; Zhang X; Wu HQ; Gu SX; Ma XD; Yang LM; Zheng YT; Chen FE Bioorg Med Chem; 2011 Sep; 19(18):5553-8. PubMed ID: 21862337 [TBL] [Abstract][Full Text] [Related]
5. CoMFA and CoMSIA 3D-QSAR studies on quionolone caroxylic acid derivatives inhibitors of HIV-1 integrase. Lu P; Wei X; Zhang R Eur J Med Chem; 2010 Aug; 45(8):3413-9. PubMed ID: 20488589 [TBL] [Abstract][Full Text] [Related]
6. Amide-containing diketoacids as HIV-1 integrase inhibitors: synthesis, structure-activity relationship analysis, and biological activity. Li H; Wang C; Sanchez T; Tan Y; Jiang C; Neamati N; Zhao G Bioorg Med Chem; 2009 Apr; 17(7):2913-9. PubMed ID: 19269185 [TBL] [Abstract][Full Text] [Related]
7. Synthesis of pyrimidine and quinolone conjugates as a scaffold for dual inhibitors of HIV reverse transcriptase and integrase. Wang Z; Vince R Bioorg Med Chem Lett; 2008 Feb; 18(4):1293-6. PubMed ID: 18226894 [TBL] [Abstract][Full Text] [Related]
8. Design and synthesis of novel β-diketo derivatives as HIV-1 integrase inhibitors. Hu L; Zhang S; He X; Luo Z; Wang X; Liu W; Qin X Bioorg Med Chem; 2012 Jan; 20(1):177-82. PubMed ID: 22154762 [TBL] [Abstract][Full Text] [Related]
9. Synthesis, antiviral, and anti-HIV-1 integrase activities of 3-aroyl-1,1-dioxo-1,4,2-benzodithiazines. Brzozowski Z; Saczewski F; Sanchez T; Kuo CL; Gdaniec M; Neamati N Bioorg Med Chem; 2004 Jul; 12(13):3663-72. PubMed ID: 15186851 [TBL] [Abstract][Full Text] [Related]
10. Design, synthesis, and anti-integrase activity of catechol-DKA hybrids. Maurin C; Bailly F; Mbemba G; Mouscadet JF; Cotelle P Bioorg Med Chem; 2006 May; 14(9):2978-84. PubMed ID: 16412645 [TBL] [Abstract][Full Text] [Related]
11. Novel HIV-1 integrase inhibitors derived from quinolone antibiotics. Sato M; Motomura T; Aramaki H; Matsuda T; Yamashita M; Ito Y; Kawakami H; Matsuzaki Y; Watanabe W; Yamataka K; Ikeda S; Kodama E; Matsuoka M; Shinkai H J Med Chem; 2006 Mar; 49(5):1506-8. PubMed ID: 16509568 [TBL] [Abstract][Full Text] [Related]
12. Rational design of 2-pyrrolinones as inhibitors of HIV-1 integrase. Ma K; Wang P; Fu W; Wan X; Zhou L; Chu Y; Ye D Bioorg Med Chem Lett; 2011 Nov; 21(22):6724-7. PubMed ID: 21996518 [TBL] [Abstract][Full Text] [Related]
13. Synthesis and HIV-1 integrase inhibitory activities of caffeic acid dimers derived from Salvia officinalis. Bailly F; Queffelec C; Mbemba G; Mouscadet JF; Cotelle P Bioorg Med Chem Lett; 2005 Nov; 15(22):5053-6. PubMed ID: 16183277 [TBL] [Abstract][Full Text] [Related]
14. Quinolone carboxylic acids as a novel monoketo acid class of human immunodeficiency virus type 1 integrase inhibitors. Sato M; Kawakami H; Motomura T; Aramaki H; Matsuda T; Yamashita M; Ito Y; Matsuzaki Y; Yamataka K; Ikeda S; Shinkai H J Med Chem; 2009 Aug; 52(15):4869-82. PubMed ID: 19719237 [TBL] [Abstract][Full Text] [Related]
15. Investigations on the 4-quinolone-3-carboxylic acid motif. 1. Synthesis and structure-activity relationship of a class of human immunodeficiency virus type 1 integrase inhibitors. Pasquini S; Mugnaini C; Tintori C; Botta M; Trejos A; Arvela RK; Larhed M; Witvrouw M; Michiels M; Christ F; Debyser Z; Corelli F J Med Chem; 2008 Aug; 51(16):5125-9. PubMed ID: 18665580 [TBL] [Abstract][Full Text] [Related]
16. Design and synthesis of novel indole beta-diketo acid derivatives as HIV-1 integrase inhibitors. Sechi M; Derudas M; Dallocchio R; Dessì A; Bacchi A; Sannia L; Carta F; Palomba M; Ragab O; Chan C; Shoemaker R; Sei S; Dayam R; Neamati N J Med Chem; 2004 Oct; 47(21):5298-310. PubMed ID: 15456274 [TBL] [Abstract][Full Text] [Related]
17. Novel bifunctional quinolonyl diketo acid derivatives as HIV-1 integrase inhibitors: design, synthesis, biological activities, and mechanism of action. Di Santo R; Costi R; Roux A; Artico M; Lavecchia A; Marinelli L; Novellino E; Palmisano L; Andreotti M; Amici R; Galluzzo CM; Nencioni L; Palamara AT; Pommier Y; Marchand C J Med Chem; 2006 Mar; 49(6):1939-45. PubMed ID: 16539381 [TBL] [Abstract][Full Text] [Related]
18. Conformationally restrained carbazolone-containing alpha,gamma-diketo acids as inhibitors of HIV integrase. Li X; Vince R Bioorg Med Chem; 2006 May; 14(9):2942-55. PubMed ID: 16386908 [TBL] [Abstract][Full Text] [Related]
19. Synthesis of polyhydroxylated aromatics having amidation of piperazine nitrogen as HIV-1 integrase inhibitor. Yang L; Xu X; Huang Y; Zhang B; Zeng C; He H; Wang C; Hu L Bioorg Med Chem Lett; 2010 Sep; 20(18):5469-71. PubMed ID: 20709544 [TBL] [Abstract][Full Text] [Related]
20. Design and optimization of tricyclic phtalimide analogues as novel inhibitors of HIV-1 integrase. Verschueren WG; Dierynck I; Amssoms KI; Hu L; Boonants PM; Pille GM; Daeyaert FF; Hertogs K; Surleraux DL; Wigerinck PB J Med Chem; 2005 Mar; 48(6):1930-40. PubMed ID: 15771437 [TBL] [Abstract][Full Text] [Related] [Next] [New Search]