BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

109 related articles for article (PubMed ID: 21355526)

  • 1. Synthesis and LAR inhibition of 7-alkoxy analogues of illudalic acid.
    Ling Q; Zhou YY; Cai ZL; Zhang YH; Xiong B; Ma LP; Wang X; Li X; Li J; Shen JK
    Yao Xue Xue Bao; 2010 Nov; 45(11):1385-97. PubMed ID: 21355526
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Synthesis and PTP Inhibitory Activity of Illudalic Acid and Its Methyl Ether, with Insights into Selectivity for LAR PTP over Other Tyrosine Phosphatases under Physiologically Relevant Conditions.
    McCullough BS; Batsomboon P; Hutchinson KB; Dudley GB; Barrios AM
    J Nat Prod; 2019 Dec; 82(12):3386-3393. PubMed ID: 31809044
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Illudalic acid as a potential LAR inhibitor: synthesis, SAR, and preliminary studies on the mechanism of action.
    Ling Q; Huang Y; Zhou Y; Cai Z; Xiong B; Zhang Y; Ma L; Wang X; Li X; Li J; Shen J
    Bioorg Med Chem; 2008 Aug; 16(15):7399-409. PubMed ID: 18579388
    [TBL] [Abstract][Full Text] [Related]  

  • 4. The mechanism of covalent inhibition of LAR phosphatase by illudalic acid.
    Hansen DT; Rueb NJ; Levinzon ND; Cheatham TE; Gaston R; Tanvir Ahmed K; Osburn-Staker S; Cox JE; Dudley GB; Barrios AM
    Bioorg Med Chem Lett; 2024 May; 104():129740. PubMed ID: 38599294
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Structure-activity studies of PTPRD phosphatase inhibitors identify a 7-cyclopentymethoxy illudalic acid analog candidate for development.
    Henderson IM; Zeng F; Bhuiyan NH; Luo D; Martinez M; Smoake J; Bi F; Perera C; Johnson D; Prisinzano TE; Wang W; Uhl GR
    Biochem Pharmacol; 2022 Jan; 195():114868. PubMed ID: 34863978
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Design, synthesis, biological evaluation and molecular dynamics of LAR inhibitors.
    Sun YZ; Wu JW; Du S; Ma YC; Zhou L; Ma Y; Wang RL
    Comput Biol Chem; 2021 Jun; 92():107481. PubMed ID: 33838390
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Discovery of potent inhibitors of receptor protein tyrosine phosphatase sigma through the structure-based virtual screening.
    Park H; Chien PN; Ryu SE
    Bioorg Med Chem Lett; 2012 Oct; 22(20):6333-7. PubMed ID: 22989533
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Coumarin sulfonates: New alkaline phosphatase inhibitors; in vitro and in silico studies.
    Salar U; Khan KM; Iqbal J; Ejaz SA; Hameed A; Al-Rashida M; Perveen S; Tahir MN
    Eur J Med Chem; 2017 May; 131():29-47. PubMed ID: 28288318
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Identification of novel protein tyrosine phosphatase sigma inhibitors promoting neurite extension.
    Lee HS; Ku B; Park TH; Park H; Choi JK; Chang KT; Kim CH; Ryu SE; Kim SJ
    Bioorg Med Chem Lett; 2016 Jan; 26(1):87-93. PubMed ID: 26602279
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Divalent and trivalent alpha-ketocarboxylic acids as inhibitors of protein tyrosine phosphatases.
    Chen YT; Seto CT
    J Med Chem; 2002 Aug; 45(18):3946-52. PubMed ID: 12190316
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Discovery of new 7-substituted-4-imidazolylmethyl coumarins and 4'-substituted-2-imidazolyl acetophenones open analogues as potent and selective inhibitors of steroid-11β-hydroxylase.
    Stefanachi A; Hanke N; Pisani L; Leonetti F; Nicolotti O; Catto M; Cellamare S; Hartmann RW; Carotti A
    Eur J Med Chem; 2015 Jan; 89():106-14. PubMed ID: 25462231
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Synthesis and biological evaluation of 2,4,6-trihydroxychalcone derivatives as novel protein tyrosine phosphatase 1B inhibitors.
    Sun LP; Gao LX; Ma WP; Nan FJ; Li J; Piao HR
    Chem Biol Drug Des; 2012 Oct; 80(4):584-90. PubMed ID: 22805439
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Substituted coumarins as potent 5-lipoxygenase inhibitors.
    Grimm EL; Brideau C; Chauret N; Chan CC; Delorme D; Ducharme Y; Ethier D; Falgueyret JP; Friesen RW; Guay J; Hamel P; Riendeau D; Soucy-Breau C; Tagari P; Girard Y
    Bioorg Med Chem Lett; 2006 May; 16(9):2528-31. PubMed ID: 16464579
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Synthesis and characterization of a potent and selective protein tyrosine phosphatase inhibitor, 2.
    Hamaguchi T; Takahashi A; Kagamizono T; Manaka A; Sato M; Osada H
    Bioorg Med Chem Lett; 2000 Dec; 10(23):2657-60. PubMed ID: 11128645
    [TBL] [Abstract][Full Text] [Related]  

  • 15. [Design, synthesis and evaluation of malonic acid-based PTP1B inhibitors].
    Du X; Zhang SE; Liu JZ; Nie FL; Ye F; Tian JY; Xiao ZY
    Yao Xue Xue Bao; 2012 Mar; 47(3):367-73. PubMed ID: 22645761
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Novel Imbricatolic acid derivatives as protein tyrosine phosphatase-1B inhibitors: Design, synthesis, biological evaluation and molecular docking.
    Khan MF; Azad CS; Kumar A; Saini M; Narula AK; Jain S
    Bioorg Med Chem Lett; 2016 Apr; 26(8):1988-92. PubMed ID: 26965864
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Synthesis of illudalic acid and analogous phosphatase inhibitors.
    Fulo HF; Rueb NJ; Gaston R; Batsomboon P; Ahmed KT; Barrios AM; Dudley GB
    Org Biomol Chem; 2021 Dec; 19(48):10596-10600. PubMed ID: 34847212
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Novel thiophene derivatives as PTP1B inhibitors with selectivity and cellular activity.
    Ye D; Zhang Y; Wang F; Zheng M; Zhang X; Luo X; Shen X; Jiang H; Liu H
    Bioorg Med Chem; 2010 Mar; 18(5):1773-82. PubMed ID: 20153651
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Identification of small molecule inhibitors of PTPσ through an integrative virtual and biochemical approach.
    Martin KR; Narang P; Xu Y; Kauffman AL; Petit J; Xu HE; Meurice N; MacKeigan JP
    PLoS One; 2012; 7(11):e50217. PubMed ID: 23185579
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Investigations of linker structure on the potency of a series of bidentate protein tyrosine phosphatase inhibitors.
    Xie J; Seto CT
    Bioorg Med Chem; 2005 Apr; 13(8):2981-91. PubMed ID: 15781408
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 6.