BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

77 related articles for article (PubMed ID: 21550749)

  • 1. Expression of σ receptors of human urinary bladder tumor cells (RT-4 cells) and development of a competitive receptor binding assay for the determination of ligand affinity to human σ(2) receptors.
    Schepmann D; Lehmkuhl K; Brune S; Wünsch B
    J Pharm Biomed Anal; 2011 Jul; 55(5):1136-41. PubMed ID: 21550749
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Development of a selective competitive receptor binding assay for the determination of the affinity to NR2B containing NMDA receptors.
    Schepmann D; Frehland B; Lehmkuhl K; Tewes B; Wünsch B
    J Pharm Biomed Anal; 2010 Nov; 53(3):603-8. PubMed ID: 20462722
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Characterization of ligand binding to the σ(1) receptor in a human tumor cell line (RPMI 8226) and establishment of a competitive receptor binding assay.
    Brune S; Schepmann D; Lehmkuhl K; Frehland B; Wünsch B
    Assay Drug Dev Technol; 2012 Aug; 10(4):365-74. PubMed ID: 22192304
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Sigma-1 and sigma-2 receptors are expressed in a wide variety of human and rodent tumor cell lines.
    Vilner BJ; John CS; Bowen WD
    Cancer Res; 1995 Jan; 55(2):408-13. PubMed ID: 7812973
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Evidence for sigma-1-like receptors in isolated rat liver mitochondrial membranes.
    Klouz A; Sapena R; Liu J; Maurice T; Tillement JP; Papadopoulos V; Morin D
    Br J Pharmacol; 2002 Apr; 135(7):1607-15. PubMed ID: 11934800
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Targeting sigma receptor-binding benzamides as in vivo diagnostic and therapeutic agents for human prostate tumors.
    John CS; Vilner BJ; Geyer BC; Moody T; Bowen WD
    Cancer Res; 1999 Sep; 59(18):4578-83. PubMed ID: 10493511
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Modulation by sigma ligands of intracellular free Ca++ mobilization by N-methyl-D-aspartate in primary culture of rat frontal cortical neurons.
    Hayashi T; Kagaya A; Takebayashi M; Shimizu M; Uchitomi Y; Motohashi N; Yamawaki S
    J Pharmacol Exp Ther; 1995 Oct; 275(1):207-14. PubMed ID: 7562551
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Sigma Receptor Binding Assays.
    Chu UB; Ruoho AE
    Curr Protoc Pharmacol; 2015 Dec; 71():1.34.1-1.34.21. PubMed ID: 26646191
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Effects of (+)-pentazocine and 1,3-di-o-tolylguanidine (DTG), sigma (sigma) ligands, on micturition in anaesthetized rats.
    Shimizu I; Kawashima K; Ishii D; Oka M
    Br J Pharmacol; 2000 Oct; 131(3):610-6. PubMed ID: 11015314
    [TBL] [Abstract][Full Text] [Related]  

  • 10. 4-(tetralin-1-yl)- and 4-(naphthalen-1-yl)alkyl derivatives of 1-cyclohexylpiperazine as sigma receptor ligands with agonist sigma2 activity.
    Berardi F; Ferorelli S; Abate C; Colabufo NA; Contino M; Perrone R; Tortorella V
    J Med Chem; 2004 Apr; 47(9):2308-17. PubMed ID: 15084129
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Multiple affinity binding states of the sigma receptor: effect of GTP-binding protein-modifying agents.
    Itzhak Y
    Mol Pharmacol; 1989 Oct; 36(4):512-7. PubMed ID: 2554109
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Sigma1 and sigma2 receptor binding affinity and selectivity of SA4503 and fluoroethyl SA4503.
    Lever JR; Gustafson JL; Xu R; Allmon RL; Lever SZ
    Synapse; 2006 May; 59(6):350-8. PubMed ID: 16463398
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Naloxone-sensitive, haloperidol-sensitive, [3H](+)SKF-10047-binding protein partially purified from rat liver and rat brain membranes: an opioid/sigma receptor?
    Tsao LI; Su TP
    Synapse; 1997 Feb; 25(2):117-24. PubMed ID: 9021892
    [TBL] [Abstract][Full Text] [Related]  

  • 14. sigma Receptor ligand-induced up-regulation of the H(+)/peptide transporter PEPT1 in the human intestinal cell line Caco-2.
    Fujita T; Majikawa Y; Umehisa S; Okada N; Yamamoto A; Ganapathy V; Leibach FH
    Biochem Biophys Res Commun; 1999 Aug; 261(2):242-6. PubMed ID: 10425172
    [TBL] [Abstract][Full Text] [Related]  

  • 15. New sigma and 5-HT1A receptor ligands: omega-(tetralin-1-yl)-n-alkylamine derivatives.
    Berardi F; Colabufo NA; Giudice G; Perrone R; Tortorella V; Govoni S; Lucchi L
    J Med Chem; 1996 Jan; 39(1):176-82. PubMed ID: 8568804
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Irreversible blockade of sigma-1 receptors by haloperidol and its metabolites in guinea pig brain and SH-SY5Y human neuroblastoma cells.
    Cobos EJ; del Pozo E; Baeyens JM
    J Neurochem; 2007 Aug; 102(3):812-25. PubMed ID: 17419803
    [TBL] [Abstract][Full Text] [Related]  

  • 17. [(3)H]MRE 3008F20: a novel antagonist radioligand for the pharmacological and biochemical characterization of human A(3) adenosine receptors.
    Varani K; Merighi S; Gessi S; Klotz KN; Leung E; Baraldi PG; Cacciari B; Romagnoli R; Spalluto G; Borea PA
    Mol Pharmacol; 2000 May; 57(5):968-75. PubMed ID: 10779381
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Binding properties of [3H]MS-377, a novel sigma receptor ligand, to rat brain membranes.
    Karasawa J; Takahashi S; Horikomi K
    Eur J Pharmacol; 2000 Jul; 400(1):51-7. PubMed ID: 10913584
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Differential solubilization of rat liver sigma 1 and sigma 2 receptors: retention of sigma 2 sites in particulate fractions.
    Torrence-Campbell C; Bowen WD
    Eur J Pharmacol; 1996 May; 304(1-3):201-10. PubMed ID: 8813603
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Radioiodination and preclinical evaluation of 4-benzyl-1-(3-[
    Sadeghzadeh M; Alirezapour B; Charkhlooie GA; Baghery MK; Khorouti A
    Ann Nucl Med; 2017 May; 31(4):335-346. PubMed ID: 28315150
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 4.