BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

252 related articles for article (PubMed ID: 21684751)

  • 1. Design, synthesis and antileishmanial in vitro activity of new series of chalcones-like compounds: a molecular hybridization approach.
    Barbosa TP; Sousa SC; Amorim FM; Rodrigues YK; de Assis PA; Caldas JP; Oliveira MR; Vasconcellos ML
    Bioorg Med Chem; 2011 Jul; 19(14):4250-6. PubMed ID: 21684751
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Synthesis, evaluation against Leishmania amazonensis and cytotoxicity assays in macrophages of sixteen new congeners Morita-Baylis-Hillman adducts.
    Silva FP; de Assis PA; Junior CG; de Andrade NG; da Cunha SM; Oliveira MR; Vasconcellos ML
    Eur J Med Chem; 2011 Sep; 46(9):4295-301. PubMed ID: 21775030
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Improved synthesis of seven aromatic Baylis-Hillman adducts (BHA): evaluation against Artemia salina Leach. and Leishmania chagasi.
    Barbosa TP; Junior CG; Silva FP; Lopes HM; Figueiredo LR; Sousa SC; Batista GN; da Silva TG; Silva TM; de Oliveira MR; Vasconcellos ML
    Eur J Med Chem; 2009 Apr; 44(4):1726-30. PubMed ID: 18448204
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Efficient synthesis of 16 aromatic Morita-Baylis-Hillman adducts: Biological evaluation on Leishmania amazonensis and Leishmania chagasi.
    Junior CG; de Assis PA; Silva FP; Sousa SC; de Andrade NG; Barbosa TP; Nerís PL; Segundo LV; Anjos IC; Carvalho GA; Rocha GB; Oliveira MR; Vasconcellos ML
    Bioorg Chem; 2010 Dec; 38(6):279-84. PubMed ID: 20855101
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Synthesis and evaluation of new furanyl and thiophenyl azoles as antileishmanial agents.
    Marrapu VK; Mittal M; Shivahare R; Gupta S; Bhandari K
    Eur J Med Chem; 2011 May; 46(5):1694-700. PubMed ID: 21385661
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Synthesis, analytical behaviour and biological evaluation of new 4-substituted pyrrolo[1,2-a]quinoxalines as antileishmanial agents.
    Guillon J; Forfar I; Mamani-Matsuda M; Desplat V; Saliège M; Thiolat D; Massip S; Tabourier A; Léger JM; Dufaure B; Haumont G; Jarry C; Mossalayi D
    Bioorg Med Chem; 2007 Jan; 15(1):194-210. PubMed ID: 17049253
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Synthesis and antileishmanial evaluation of 1-aryl-4-(4,5-dihydro-1H-imidazol-2-yl)-1H-pyrazole derivatives.
    dos Santos MS; Oliveira ML; Bernardino AM; de Léo RM; Amaral VF; de Carvalho FT; Leon LL; Canto-Cavalheiro MM
    Bioorg Med Chem Lett; 2011 Dec; 21(24):7451-4. PubMed ID: 22055204
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Synthesis and in vitro evaluation of leishmanicidal and trypanocidal activities of N-quinolin-8-yl-arylsulfonamides.
    da Silva LE; Joussef AC; Pacheco LK; da Silva DG; Steindel M; Rebelo RA; Schmidt B
    Bioorg Med Chem; 2007 Dec; 15(24):7553-60. PubMed ID: 17889546
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Preparation and antileishmanial activity of lipophilic N-alkyl diamines.
    da Costa CF; Coimbra ES; Braga FG; dos Reis RC; da Silva AD; de Almeida MV
    Biomed Pharmacother; 2009 Jan; 63(1):40-2. PubMed ID: 18262385
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Synthesis and In Vitro Anti Leishmania amazonensis Biological Screening of Morita-Baylis-Hillman Adducts Prepared from Eugenol, Thymol and Carvacrol.
    Xavier FJ; Rodrigues KA; de Oliveira RG; Lima Junior CG; Rocha JD; Keesen TS; de Oliveira MR; Silva FP; Vasconcellos ML
    Molecules; 2016 Nov; 21(11):. PubMed ID: 27834831
    [TBL] [Abstract][Full Text] [Related]  

  • 11. A comprehensive review of chalcone derivatives as antileishmanial agents.
    de Mello MVP; Abrahim-Vieira BA; Domingos TFS; de Jesus JB; de Sousa ACC; Rodrigues CR; Souza AMT
    Eur J Med Chem; 2018 Apr; 150():920-929. PubMed ID: 29602038
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Novel 3,4-methylenedioxyde-6-X-benzaldehyde-thiosemicarbazones: Synthesis and antileishmanial effects against Leishmania amazonensis.
    de Melos JL; Torres-Santos EC; Faiões Vdos S; Del Cistia Cde N; Sant'Anna CM; Rodrigues-Santos CE; Echevarria A
    Eur J Med Chem; 2015 Oct; 103():409-17. PubMed ID: 26375353
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Trimethoxy-chalcone derivatives inhibit growth of Leishmania braziliensis: synthesis, biological evaluation, molecular modeling and structure-activity relationship (SAR).
    Bello ML; Chiaradia LD; Dias LR; Pacheco LK; Stumpf TR; Mascarello A; Steindel M; Yunes RA; Castro HC; Nunes RJ; Rodrigues CR
    Bioorg Med Chem; 2011 Aug; 19(16):5046-52. PubMed ID: 21757358
    [TBL] [Abstract][Full Text] [Related]  

  • 14. A comparative study of mesoionic compounds in Leishmania sp. and toxicity evaluation.
    Rodrigues RF; da Silva EF; Echevarria A; Fajardo-Bonin R; Amaral VF; Leon LL; Canto-Cavalheiro MM
    Eur J Med Chem; 2007 Jul; 42(7):1039-43. PubMed ID: 17367894
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Antiprotozoal activity of chloroquinoline based chalcones.
    Hayat F; Moseley E; Salahuddin A; Van Zyl RL; Azam A
    Eur J Med Chem; 2011 May; 46(5):1897-905. PubMed ID: 21377771
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Biological activity of Morita-Baylis-Hillman adduct homodimers in L. infantum and L. amazonensis: anti-Leishmania activity and cytotoxicity.
    da Câmara Rocha J; da Franca Rodrigues KA; do Nascimento Néris PL; da Silva LV; Almeida FS; Lima VS; Peixoto RF; da Câmara Rocha J; de Azevedo FLAA; Veras RC; de Medeiros IA; da Silva WAV; Lima-Junior CG; de Almeida Vasconcellos MLA; do Amaral IPG; de Oliveira MR; de Souza Lima Keesen T
    Parasitol Res; 2019 Oct; 118(10):3067-3076. PubMed ID: 31392413
    [TBL] [Abstract][Full Text] [Related]  

  • 17. In vitro and in vivo anti-Leishmania activity of polysubstituted synthetic chalcones.
    Aponte JC; Castillo D; Estevez Y; Gonzalez G; Arevalo J; Hammond GB; Sauvain M
    Bioorg Med Chem Lett; 2010 Jan; 20(1):100-3. PubMed ID: 19962891
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Design, synthesis and biological evaluation of aryl pyrimidine derivatives as potential leishmanicidal agents.
    Suryawanshi SN; Kumar S; Shivahare R; Pandey S; Tiwari A; Gupta S
    Bioorg Med Chem Lett; 2013 Sep; 23(18):5235-8. PubMed ID: 23910597
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Dihydropyrido[2,3-d]pyrimidines as a new class of antileishmanial agents.
    Agarwal A; Ramesh ; Ashutosh ; Goyal N; Chauhan PM; Gupta S
    Bioorg Med Chem; 2005 Dec; 13(24):6678-84. PubMed ID: 16126395
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Triazolopyridopyrimidines: an emerging family of effective DNA photocleavers. DNA binding. Antileishmanial activity.
    Adam R; Bilbao-Ramos P; Abarca B; Ballesteros R; González-Rosende ME; Dea-Ayuela MA; Estevan F; Alzuet-Piña G
    Org Biomol Chem; 2015 May; 13(17):4903-17. PubMed ID: 25812028
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 13.