BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

427 related articles for article (PubMed ID: 21723734)

  • 1. Synthesis and antimalarial activity of new heterocyclic hybrids based on chloroquine and thiazolidinone scaffolds.
    Rojas Ruiz FA; García-Sánchez RN; Estupiñan SV; Gómez-Barrio A; Torres Amado DF; Pérez-Solórzano BM; Nogal-Ruiz JJ; Martínez-Fernández AR; Kouznetsov VV
    Bioorg Med Chem; 2011 Aug; 19(15):4562-73. PubMed ID: 21723734
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Synthesis and in vitro evaluation of new chloroquine-chalcone hybrids against chloroquine-resistant strain of Plasmodium falciparum.
    Sashidhara KV; Avula SR; Palnati GR; Singh SV; Srivastava K; Puri SK; Saxena JK
    Bioorg Med Chem Lett; 2012 Sep; 22(17):5455-9. PubMed ID: 22850213
    [TBL] [Abstract][Full Text] [Related]  

  • 3. 4-aminoquinoline-triazine-based hybrids with improved in vitro antimalarial activity against CQ-sensitive and CQ-resistant strains of Plasmodium falciparum.
    Manohar S; Khan SI; Rawat DS
    Chem Biol Drug Des; 2013 May; 81(5):625-30. PubMed ID: 23331618
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Chloroquine-astemizole hybrids with potent in vitro and in vivo antiplasmodial activity.
    Musonda CC; Whitlock GA; Witty MJ; Brun R; Kaiser M
    Bioorg Med Chem Lett; 2009 Jan; 19(2):481-4. PubMed ID: 19054674
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Toward a novel metal-based chemotherapy against tropical diseases. 7. Synthesis and in vitro antimalarial activity of new gold-chloroquine complexes.
    Navarro M; Vásquez F; Sánchez-Delgado RA; Pérez H; Sinou V; Schrével J
    J Med Chem; 2004 Oct; 47(21):5204-9. PubMed ID: 15456263
    [TBL] [Abstract][Full Text] [Related]  

  • 6. 4-Aminoquinoline quinolizidinyl- and quinolizidinylalkyl-derivatives with antimalarial activity.
    Sparatore A; Basilico N; Parapini S; Romeo S; Novelli F; Sparatore F; Taramelli D
    Bioorg Med Chem; 2005 Sep; 13(18):5338-45. PubMed ID: 16054368
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Synthesis and antimalarial activity in vitro and in vivo of a new ferrocene-chloroquine analogue.
    Biot C; Glorian G; Maciejewski LA; Brocard JS
    J Med Chem; 1997 Nov; 40(23):3715-8. PubMed ID: 9371235
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Synthesis, characterization and antimalarial activity of quinoline-pyrimidine hybrids.
    Pretorius SI; Breytenbach WJ; de Kock C; Smith PJ; N'Da DD
    Bioorg Med Chem; 2013 Jan; 21(1):269-77. PubMed ID: 23168082
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Antimalarial acridines: synthesis, in vitro activity against P. falciparum and interaction with hematin.
    Guetzoyan L; Yu XM; Ramiandrasoa F; Pethe S; Rogier C; Pradines B; Cresteil T; Perrée-Fauvet M; Mahy JP
    Bioorg Med Chem; 2009 Dec; 17(23):8032-9. PubMed ID: 19879150
    [TBL] [Abstract][Full Text] [Related]  

  • 10. In vitro and in vivo chloroquine-potentiating action of Strychnos myrtoides alkaloids against chloroquine-resistant strains of Plasmodium malaria.
    Rasoanaivo P; Ratsimamanga-Urverg S; Milijaona R; Rafatro H; Rakoto-Ratsimamanga A; Galeffi C; Nicoletti M
    Planta Med; 1994 Feb; 60(1):13-6. PubMed ID: 8134408
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Malagashanine potentiates chloroquine antimalarial activity in drug resistant Plasmodium malaria by modifying both its efflux and influx.
    Ramanitrahasimbola D; Rasoanaivo P; Ratsimamanga S; Vial H
    Mol Biochem Parasitol; 2006 Mar; 146(1):58-67. PubMed ID: 16313982
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Toward a novel metal-based chemotherapy against tropical diseases. 2. Synthesis and antimalarial activity in vitro and in vivo of new ruthenium- and rhodium-chloroquine complexes.
    Sánchez-Delgado RA; Navarro M; Pérez H; Urbina JA
    J Med Chem; 1996 Mar; 39(5):1095-99. PubMed ID: 8676344
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Toward a novel metal-based chemotherapy against tropical diseases. 3. Synthesis and antimalarial activity in vitro and in vivo of the new gold-chloroquine complex [Au(PPh3)(CQ)]PF6.
    Navarro M; Pérez H; Sánchez-Delgado RA
    J Med Chem; 1997 Jun; 40(12):1937-9. PubMed ID: 9191972
    [No Abstract]   [Full Text] [Related]  

  • 14. Antiplasmodial activity of novel keto-enamine chalcone-chloroquine based hybrid pharmacophores.
    Sashidhara KV; Kumar M; Modukuri RK; Srivastava RK; Soni A; Srivastava K; Singh SV; Saxena JK; Gauniyal HM; Puri SK
    Bioorg Med Chem; 2012 May; 20(9):2971-81. PubMed ID: 22464685
    [TBL] [Abstract][Full Text] [Related]  

  • 15. In vitro efficacy of 7-benzylamino-1-isoquinolinamines against Plasmodium falciparum related to the efficacy of chalcones.
    Gutteridge CE; Hoffman MM; Bhattacharjee AK; Milhous WK; Gerena L
    Bioorg Med Chem Lett; 2011 Jan; 21(2):786-9. PubMed ID: 21168330
    [TBL] [Abstract][Full Text] [Related]  

  • 16. A new class of phenazines with activity against a chloroquine resistant Plasmodium falciparum strain and antimicrobial activity.
    Hussain H; Specht S; Sarite SR; Saeftel M; Hoerauf A; Schulz B; Krohn K
    J Med Chem; 2011 Jul; 54(13):4913-7. PubMed ID: 21591758
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Quinoline antimalarials containing a dibemethin group are active against chloroquinone-resistant Plasmodium falciparum and inhibit chloroquine transport via the P. falciparum chloroquine-resistance transporter (PfCRT).
    Zishiri VK; Joshi MC; Hunter R; Chibale K; Smith PJ; Summers RL; Martin RE; Egan TJ
    J Med Chem; 2011 Oct; 54(19):6956-68. PubMed ID: 21875063
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Synthesis and antimalarial evaluation of novel isocryptolepine derivatives.
    Whittell LR; Batty KT; Wong RP; Bolitho EM; Fox SA; Davis TM; Murray PE
    Bioorg Med Chem; 2011 Dec; 19(24):7519-25. PubMed ID: 22055713
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Synthesis and antimalarial properties of new chloro-9H-xanthones with an aminoalkyl side chain.
    Portela C; Afonso CM; Pinto MM; Lopes D; Nogueira F; do Rosário V
    Chem Biodivers; 2007 Jul; 4(7):1508-19. PubMed ID: 17638332
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Fluoxetine potentiates chloroquine and mefloquine effect on multidrug-resistant Plasmodium falciparum in vitro.
    Khairul MF; Min TH; Low JH; Nasriyyah CH; A'shikin AN; Norazmi MN; Ravichandran M; Raju SS
    Jpn J Infect Dis; 2006 Oct; 59(5):329-31. PubMed ID: 17060702
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 22.