BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

112 related articles for article (PubMed ID: 21729714)

  • 1. New ester derivatives of dehydroepiandrosterone as 5α-reductase inhibitors.
    Arellano Y; Bratoeff E; Garrido M; Soriano J; Heuze Y; Cabeza M
    Steroids; 2011 Nov; 76(12):1241-6. PubMed ID: 21729714
    [TBL] [Abstract][Full Text] [Related]  

  • 2. New steroidal lactones as 5α-reductase inhibitors and antagonists for the androgen receptor.
    Garrido M; Bratoeff E; Bonilla D; Soriano J; Heuze Y; Cabeza M
    J Steroid Biochem Mol Biol; 2011 Nov; 127(3-5):367-73. PubMed ID: 21782943
    [TBL] [Abstract][Full Text] [Related]  

  • 3. In vivo and in vitro effect of androstene derivatives as 5α-reductase type 1 enzyme inhibitors.
    Bratoeff E; Sánchez A; Arellano Y; Heuze Y; Soriano J; Cabeza M
    J Enzyme Inhib Med Chem; 2013 Dec; 28(6):1247-54. PubMed ID: 23051174
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Novel C-6 substituted and unsubstituted pregnane derivatives as 5alpha-reductase inhibitors and their effect on hamster flank organs diameter size.
    Cabeza M; Zambrano A; Heuze I; Carrizales E; Palacios A; Segura T; Valencia N; Bratoeff E
    Steroids; 2009 Oct; 74(10-11):793-802. PubMed ID: 19406144
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Synthesis and biological activity of progesterone derivatives as 5alpha-reductase inhibitors, and their effect on hamster prostate weight.
    Bratoeff E; Zambrano A; Heuze I; Palacios A; Ramírez D; Cabeza M
    J Enzyme Inhib Med Chem; 2010 Jun; 25(3):306-11. PubMed ID: 19874206
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Aromatic esters of progesterone as 5alpha-reductase and prostate growth inhibitors.
    Bratoeff E; Segura T; Recillas S; Carrizales E; Palacios A; Heuze I; Cabeza M
    J Enzyme Inhib Med Chem; 2009 Jun; 24(3):655-62. PubMed ID: 18825535
    [TBL] [Abstract][Full Text] [Related]  

  • 7. In vivo and in vitro effect of novel 4,16-pregnadiene-6,20-dione derivatives, as 5alpha-reductase inhibitors.
    Bratoeff E; Cabeza M; Pérez-Ornelas V; Recillas S; Heuze I
    J Steroid Biochem Mol Biol; 2008 Sep; 111(3-5):275-81. PubMed ID: 18644453
    [TBL] [Abstract][Full Text] [Related]  

  • 8. New 5alpha-reductase inhibitors: in vitro and in vivo effects.
    Pérez-Ornelas V; Cabeza M; Bratoeff E; Heuze I; Sánchez M; Ramírez E; Naranjo-Rodríguez E
    Steroids; 2005 Mar; 70(3):217-24. PubMed ID: 15763601
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Effect of dehydroepiandrosterone derivatives on the activity of 5α-reductase isoenzymes and on cancer cell line PC-3.
    Bratoeff E; Garrido M; Ramírez-Apan T; Heuze Y; Sánchez A; Soriano J; Cabeza M
    Bioorg Med Chem; 2014 Nov; 22(21):6233-41. PubMed ID: 25261928
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Synthesis and activity of novel 16-dehydropregnenolone acetate derivatives as inhibitors of type 1 5α-reductase and on cancer cell line SK-LU-1.
    Silva-Ortiz AV; Bratoeff E; Ramírez-Apan T; Heuze Y; Sánchez A; Soriano J; Cabeza M
    Bioorg Med Chem; 2015 Dec; 23(24):7535-42. PubMed ID: 26631442
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Novel dehydroepiandrosterone benzimidazolyl derivatives as 5α-reductase isozymes inhibitors.
    Arellano Y; Bratoeff E; Segura T; Mendoza ME; Sánchez-Márquez A; Medina Y; Heuze Y; Soriano J; Cabeza M
    J Enzyme Inhib Med Chem; 2016 Dec; 31(6):908-14. PubMed ID: 26394987
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Synthesis and biological evaluation of novel unsaturated carboxysteroids as human 5α-reductase inhibitors: a legitimate approach.
    Aggarwal S; Thareja S; Bhardwaj TR; Haupenthal J; Hartmann RW; Kumar M
    Eur J Med Chem; 2012 Aug; 54():728-39. PubMed ID: 22776417
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Activity of steroid 4 and derivatives 4a-4f as inhibitors of the enzyme 5α-reductase 1.
    Arellano Y; Bratoeff E; Heuze Y; Bravo M; Soriano J; Cabeza M
    Bioorg Med Chem; 2018 Aug; 26(14):4058-4064. PubMed ID: 30007568
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Molecular interactions of progesterone derivatives with 5 alpha-reductase types 1 and 2 and androgen receptors.
    Bratoeff E; García P; Heuze Y; Soriano J; Mejía A; Labastida AM; Valencia N; Cabeza M
    Steroids; 2010 Jul; 75(7):499-505. PubMed ID: 20359488
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Steroids with a carbamate function at C-17, a novel class of inhibitors for human and hamster steroid 5alpha-reductase.
    Bratoeff E; Sainz T; Cabeza M; Heuze I; Recillas S; Pérez V; Rodríguez C; Segura T; Gonzáles J; Ramírez E
    J Steroid Biochem Mol Biol; 2007 Oct; 107(1-2):48-56. PubMed ID: 17629476
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Activity of 17beta-(N-alkyl/arylformamido) and 17beta-[(N-alkyl/aryl) alkyl/arylamido]-4-methyl-4-aza-5alpha-androstan-3-ones as 5alpha-reductase inhibitors in the hamster flank organ and ear.
    Chen C; Li X; Singh SM; Labrie F
    J Invest Dermatol; 1998 Aug; 111(2):273-8. PubMed ID: 9699729
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Synthesis and biological evaluation of 3-tetrazolo steroidal analogs: Novel class of 5α-reductase inhibitors.
    Aggarwal S; Mahapatra MK; Kumar R; Bhardwaj TR; Hartmann RW; Haupenthal J; Kumar M
    Bioorg Med Chem; 2016 Feb; 24(4):779-88. PubMed ID: 26780831
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Antiandrogenic effect of 16-substituted, non-substituted and D-homopregnane derivatives.
    Bratoeff EA; Herrera H; Ramírez E; Solorzano K; Murillo E; Quiróz A; Cabeza M
    Chem Pharm Bull (Tokyo); 2000 Sep; 48(9):1249-55. PubMed ID: 10993221
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Synthesis and biological evaluation of esters of 16-formyl-17-methoxy-dehydroepiandrosterone derivatives as inhibitors of 5α-reductase type 2.
    Sánchez-Márquez A; Arellano Y; Bratoeff E; Heuze Y; Córdova K; Nieves G; Soriano J; Cabeza M
    J Enzyme Inhib Med Chem; 2016 Dec; 31(6):1170-6. PubMed ID: 26526826
    [TBL] [Abstract][Full Text] [Related]  

  • 20. 5α-Reductase, an enzyme regulating glucocorticoid action in the testis of Rhinella arenarum (Amphibia: Anura).
    Tesone AJ; Regueira E; Canosa LF; Ceballos NR
    Gen Comp Endocrinol; 2012 May; 176(3):500-6. PubMed ID: 22285601
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 6.