BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

154 related articles for article (PubMed ID: 2190554)

  • 1. Substitution of proline with pipecolic acid at the scissile bond converts a peptide substrate of HIV proteinase into a selective inhibitor.
    Copeland TD; Wondrak EM; Tozser J; Roberts MM; Oroszlan S
    Biochem Biophys Res Commun; 1990 May; 169(1):310-4. PubMed ID: 2190554
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Hydrolysis of synthetic chromogenic substrates by HIV-1 and HIV-2 proteinases.
    Phylip LH; Richards AD; Kay J; Kovalinka J; Strop P; Blaha I; Velek J; Kostka V; Ritchie AJ; Broadhurst AV
    Biochem Biophys Res Commun; 1990 Aug; 171(1):439-44. PubMed ID: 2203349
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Specificity and inhibition of proteases from human immunodeficiency viruses 1 and 2.
    Tomasselli AG; Hui JO; Sawyer TK; Staples DJ; Bannow C; Reardon IM; Howe WJ; DeCamp DL; Craik CS; Heinrikson RL
    J Biol Chem; 1990 Aug; 265(24):14675-83. PubMed ID: 2201691
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Rational design of peptide-based HIV proteinase inhibitors.
    Roberts NA; Martin JA; Kinchington D; Broadhurst AV; Craig JC; Duncan IB; Galpin SA; Handa BK; Kay J; Kröhn A
    Science; 1990 Apr; 248(4953):358-61. PubMed ID: 2183354
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Novel fluorogenic substrates for assaying retroviral proteases by resonance energy transfer.
    Matayoshi ED; Wang GT; Krafft GA; Erickson J
    Science; 1990 Feb; 247(4945):954-8. PubMed ID: 2106161
    [TBL] [Abstract][Full Text] [Related]  

  • 6. In vitro inhibition of HIV-1 proteinase by cerulenin.
    Moelling K; Schulze T; Knoop MT; Kay J; Jupp R; Nicolaou G; Pearl LH
    FEBS Lett; 1990 Feb; 261(2):373-7. PubMed ID: 1690152
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Modified oligopeptides designed to interact with the HIV-1 proteinase inhibit viral replication.
    Grinde B; Hungnes O; Tjøtta E
    Arch Virol; 1990; 114(3-4):167-73. PubMed ID: 2241573
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Sensitive, soluble chromogenic substrates for HIV-1 proteinase.
    Richards AD; Phylip LH; Farmerie WG; Scarborough PE; Alvarez A; Dunn BM; Hirel PH; Konvalinka J; Strop P; Pavlickova L
    J Biol Chem; 1990 May; 265(14):7733-6. PubMed ID: 2186027
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Studies on the role of the S4 substrate binding site of HIV proteinases.
    Tözsér J; Gustchina A; Weber IT; Blaha I; Wondrak EM; Oroszlan S
    FEBS Lett; 1991 Feb; 279(2):356-60. PubMed ID: 2001747
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Synthesis of homologous peptides using fragment condensation: analogs of an HIV proteinase substrate.
    Bláha I; Nemec J; Tözsér J; Oroszlan S
    Int J Pept Protein Res; 1991 Nov; 38(5):453-8. PubMed ID: 1802863
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Selective phosphinate transition-state analogue inhibitors of the protease of human immunodeficiency virus.
    Grobelny D; Wondrak EM; Galardy RE; Oroszlan S
    Biochem Biophys Res Commun; 1990 Jun; 169(3):1111-6. PubMed ID: 2114105
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Mutational analysis of a native substrate of the human immunodeficiency virus type 1 proteinase.
    Partin K; Kräusslich HG; Ehrlich L; Wimmer E; Carter C
    J Virol; 1990 Aug; 64(8):3938-47. PubMed ID: 2196384
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Substrate analogue inhibition and active site titration of purified recombinant HIV-1 protease.
    Tomasselli AG; Olsen MK; Hui JO; Staples DJ; Sawyer TK; Heinrikson RL; Tomich CS
    Biochemistry; 1990 Jan; 29(1):264-9. PubMed ID: 2182116
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Sub-site preferences of the aspartic proteinase from the human immunodeficiency virus, HIV-1.
    Konvalinka J; Strop P; Velek J; Cerna V; Kostka V; Phylip LH; Richards AD; Dunn BM; Kay J
    FEBS Lett; 1990 Jul; 268(1):35-8. PubMed ID: 2200711
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Hydroxyethylamine analogues of the p17/p24 substrate cleavage site are tight-binding inhibitors of HIV protease.
    Rich DH; Green J; Toth MV; Marshall GR; Kent SB
    J Med Chem; 1990 May; 33(5):1285-8. PubMed ID: 2184237
    [No Abstract]   [Full Text] [Related]  

  • 16. Substitutions at the P2' site of gag p17-p24 affect cleavage efficiency by HIV-1 protease.
    Margolin N; Heath W; Osborne E; Lai M; Vlahos C
    Biochem Biophys Res Commun; 1990 Mar; 167(2):554-60. PubMed ID: 2182016
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Subsite preferences of retroviral proteinases.
    Dunn BM; Gustchina A; Wlodawer A; Kay J
    Methods Enzymol; 1994; 241():254-78. PubMed ID: 7854181
    [No Abstract]   [Full Text] [Related]  

  • 18. Affinity purification of the HIV-1 protease.
    Heimbach JC; Garsky VM; Michelson SR; Dixon RA; Sigal IS; Darke PL
    Biochem Biophys Res Commun; 1989 Nov; 164(3):955-60. PubMed ID: 2686642
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Structure at 2.5-A resolution of chemically synthesized human immunodeficiency virus type 1 protease complexed with a hydroxyethylene-based inhibitor.
    Jaskólski M; Tomasselli AG; Sawyer TK; Staples DG; Heinrikson RL; Schneider J; Kent SB; Wlodawer A
    Biochemistry; 1991 Feb; 30(6):1600-9. PubMed ID: 1993177
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Design, activity, and 2.8 A crystal structure of a C2 symmetric inhibitor complexed to HIV-1 protease.
    Erickson J; Neidhart DJ; VanDrie J; Kempf DJ; Wang XC; Norbeck DW; Plattner JJ; Rittenhouse JW; Turon M; Wideburg N
    Science; 1990 Aug; 249(4968):527-33. PubMed ID: 2200122
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 8.