142 related articles for article (PubMed ID: 21916484)
1. 6-arylcoumarins as novel nonsteroidal type progesterone antagonists: an example with receptor-binding-dependent fluorescence.
Sakai H; Hirano T; Mori S; Fujii S; Masuno H; Kinoshita M; Kagechika H; Tanatani A
J Med Chem; 2011 Oct; 54(20):7055-65. PubMed ID: 21916484
[TBL] [Abstract][Full Text] [Related]
2. Development of 6-arylcoumarins as nonsteroidal progesterone antagonists. Structure-activity relationships and fluorescence properties.
Kinoshita M; Negishi M; Sakai H; Hirano T; Mori S; Fujii S; Kagechika H; Tanatani A
Bioorg Med Chem; 2016 Nov; 24(21):5602-5610. PubMed ID: 27665178
[TBL] [Abstract][Full Text] [Related]
3. Characterization of a new class of selective nonsteroidal progesterone receptor agonists.
Dong Y; Roberge JY; Wang Z; Wang X; Tamasi J; Dell V; Golla R; Corte JR; Liu Y; Fang T; Anthony MN; Schnur DM; Agler ML; Dickson JK; Lawrence RM; Prack MM; Seethala R; Feyen JH
Steroids; 2004 Mar; 69(3):201-17. PubMed ID: 15072922
[TBL] [Abstract][Full Text] [Related]
4. 1,5-Dihydro-benzo[e][1,4]oxazepin-2(1H)-ones containing a 7-(5'-cyanopyrrol-2-yl) group as nonsteroidal progesterone receptor modulators.
Kern JC; Terefenko EA; Fensome A; Unwalla R; Wrobel J; Cohen J; Zhu Y; Berrodin TJ; Yudt MR; Winneker RC; Zhang Z; Zhang P
Bioorg Med Chem Lett; 2008 Sep; 18(18):5015-7. PubMed ID: 18722119
[TBL] [Abstract][Full Text] [Related]
5. Progesterone receptor antagonists with a 3-phenylquinazoline-2,4-dione/2-phenylisoquinoline-1,3-dione skeleton.
Nakagawa A; Uno S; Makishima M; Miyachi H; Hashimoto Y
Bioorg Med Chem; 2008 Jul; 16(14):7046-54. PubMed ID: 18586498
[TBL] [Abstract][Full Text] [Related]
6. 1-Methyl-1H-pyrrole-2-carbonitrile containing tetrahydronaphthalene derivatives as non-steroidal progesterone receptor antagonists.
Kern JC; Terefenko E; Trybulski E; Berrodin TJ; Cohen J; Winneker RC; Yudt MR; Zhang Z; Zhu Y; Zhang P
Bioorg Med Chem Lett; 2010 Aug; 20(16):4816-8. PubMed ID: 20638844
[TBL] [Abstract][Full Text] [Related]
7. Synthesis and biological evaluation of (6- and 7-phenyl) coumarin derivatives as selective nonsteroidal inhibitors of 17β-hydroxysteroid dehydrogenase type 1.
Starcević S; Brozic P; Turk S; Cesar J; Rizner TL; Gobec S
J Med Chem; 2011 Jan; 54(1):248-61. PubMed ID: 21138273
[TBL] [Abstract][Full Text] [Related]
8. 5-Aryl indanones and derivatives as non-steroidal progesterone receptor modulators.
Kern JC; Terefenko E; Trybulski E; Berrodin TJ; Cohen J; Winneker RC; Yudt MR; Zhang Z; Zhu Y; Zhang P
Bioorg Med Chem Lett; 2009 Dec; 19(23):6666-9. PubMed ID: 19864132
[TBL] [Abstract][Full Text] [Related]
9. Synthesis and structure-activity relationship of novel 6-aryl-1,4-dihydrobenzo[d][1,3]oxazine-2-thiones as progesterone receptor modulators leading to the potent and selective nonsteroidal progesterone receptor agonist tanaproget.
Fensome A; Bender R; Chopra R; Cohen J; Collins MA; Hudak V; Malakian K; Lockhead S; Olland A; Svenson K; Terefenko EA; Unwalla RJ; Wilhelm JM; Wolfrom S; Zhu Y; Zhang Z; Zhang P; Winneker RC; Wrobel J
J Med Chem; 2005 Aug; 48(16):5092-5. PubMed ID: 16078826
[TBL] [Abstract][Full Text] [Related]
10. Synthesis and adenosine receptors binding affinities of a series of 3-arylcoumarins.
Matos MJ; Hogger V; Gaspar A; Kachler S; Borges F; Uriarte E; Santana L; Klotz KN
J Pharm Pharmacol; 2013 Nov; 65(11):1590-7. PubMed ID: 24118065
[TBL] [Abstract][Full Text] [Related]
11. Nonsteroidal progesterone receptor ligands (I): synthesis and SAR of new tetrahydronaphthofuranone derivatives.
Shinei R; Kurihara K; Tanabe K; Tabata Y; Kurata Y; Hoshiko S; Okonogi T
Bioorg Med Chem; 2006 Jul; 14(14):4850-61. PubMed ID: 16580213
[TBL] [Abstract][Full Text] [Related]
12. A fluorescence-based assay for fatty acid amide hydrolase compatible with high-throughput screening.
Ramarao MK; Murphy EA; Shen MW; Wang Y; Bushell KN; Huang N; Pan N; Williams C; Clark JD
Anal Biochem; 2005 Aug; 343(1):143-51. PubMed ID: 16018870
[TBL] [Abstract][Full Text] [Related]
13. 5-Aryl-1,2,3,4-tetrahydrochromeno[3,4-f]quinolin-3-ones as a novel class of nonsteroidal progesterone receptor agonists: effect of A-ring modification.
Zhi L; Tegley CM; Marschke KB; Mais DE; Jones TK
J Med Chem; 1999 Apr; 42(8):1466-72. PubMed ID: 10212133
[TBL] [Abstract][Full Text] [Related]
14. Development of a library of 6-arylcoumarins as candidate fluorescent sensors.
Hirano T; Hiromoto K; Kagechika H
Org Lett; 2007 Mar; 9(7):1315-8. PubMed ID: 17326649
[TBL] [Abstract][Full Text] [Related]
15. Nonsteroidal progesterone receptor ligands (II); synthesis and SAR of new tetrahydrobenzindolone derivatives.
Kurihara K; Shinei R; Tanabe K; Tabata Y; Kurata Y; Hoshiko S; Okonogi T
Bioorg Med Chem; 2006 Jul; 14(14):4862-78. PubMed ID: 16580209
[TBL] [Abstract][Full Text] [Related]
16. Designing better coumarin-based fluorogenic substrates for PTP1B.
Holmes CP; Macher N; Grove JR; Jang L; Irvine JD
Bioorg Med Chem Lett; 2008 Jun; 18(11):3382-5. PubMed ID: 18442911
[TBL] [Abstract][Full Text] [Related]
17. 7-aryl 1,5-dihydro-benzo[e][1,4]oxazepin-2-ones and analogs as non-steroidal progesterone receptor antagonists.
Zhang P; Kern JC; Terefenko EA; Fensome A; Unwalla R; Zhang Z; Cohen J; Berrodin TJ; Yudt MR; Winneker RC; Wrobel J
Bioorg Med Chem; 2008 Jul; 16(13):6589-600. PubMed ID: 18504132
[TBL] [Abstract][Full Text] [Related]
18. Polarity-sensitive coumarins tailored to live cell imaging.
Signore G; Nifosì R; Albertazzi L; Storti B; Bizzarri R
J Am Chem Soc; 2010 Feb; 132(4):1276-88. PubMed ID: 20050646
[TBL] [Abstract][Full Text] [Related]
19. Two-photon fluorescent probes for biological Mg(2+) detection based on 7-substituted coumarin.
Yin H; Zhang B; Yu H; Zhu L; Feng Y; Zhu M; Guo Q; Meng X
J Org Chem; 2015 May; 80(9):4306-12. PubMed ID: 25844880
[TBL] [Abstract][Full Text] [Related]
20. Novel irreversible fluorescent probes targeting the 18 kDa translocator protein: synthesis and biological characterization.
Taliani S; Da Pozzo E; Bellandi M; Bendinelli S; Pugliesi I; Simorini F; La Motta C; Salerno S; Marini AM; Da Settimo F; Cosimelli B; Greco G; Novellino E; Martini C
J Med Chem; 2010 May; 53(10):4085-93. PubMed ID: 20438080
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]
