134 related articles for article (PubMed ID: 21958118)
1. Promiscuity of carbonic anhydrase II. Unexpected ester hydrolysis of carbohydrate-based sulfamate inhibitors.
Lopez M; Vu H; Wang CK; Wolf MG; Groenhof G; Innocenti A; Supuran CT; Poulsen SA
J Am Chem Soc; 2011 Nov; 133(45):18452-62. PubMed ID: 21958118
[TBL] [Abstract][Full Text] [Related]
2. Examination of two independent kinetic assays for determining the inhibition of carbonic anhydrases I and II: structure-activity comparison of sulfamates and sulfamides.
Shank RP; McComsey DF; Smith-Swintosky VL; Maryanoff BE
Chem Biol Drug Des; 2006 Aug; 68(2):113-9. PubMed ID: 16999776
[TBL] [Abstract][Full Text] [Related]
3. Inhibition of carbonic anhydrase II by thioxolone: a mechanistic and structural study.
Barrese AA; Genis C; Fisher SZ; Orwenyo JN; Kumara MT; Dutta SK; Phillips E; Kiddle JJ; Tu C; Silverman DN; Govindasamy L; Agbandje-McKenna M; McKenna R; Tripp BC
Biochemistry; 2008 Mar; 47(10):3174-84. PubMed ID: 18266323
[TBL] [Abstract][Full Text] [Related]
4. Design, synthesis, and biological evaluation of novel carbohydrate-based sulfamates as carbonic anhydrase inhibitors.
Lopez M; Trajkovic J; Bornaghi LF; Innocenti A; Vullo D; Supuran CT; Poulsen SA
J Med Chem; 2011 Mar; 54(5):1481-9. PubMed ID: 21314129
[TBL] [Abstract][Full Text] [Related]
5. Carbonic anhydrase inhibitors. Comparison of aliphatic sulfamate/bis-sulfamate adducts with isozymes II and IX as a platform for designing tight-binding, more isoform-selective inhibitors.
Vitale RM; Alterio V; Innocenti A; Winum JY; Monti SM; De Simone G; Supuran CT
J Med Chem; 2009 Oct; 52(19):5990-8. PubMed ID: 19731956
[TBL] [Abstract][Full Text] [Related]
6. Inhibition of carbonic anhydrase-II by sulfamate and sulfamide groups: an investigation involving direct thermodynamic binding measurements.
Klinger AL; McComsey DF; Smith-Swintosky V; Shank RP; Maryanoff BE
J Med Chem; 2006 Jun; 49(12):3496-500. PubMed ID: 16759092
[TBL] [Abstract][Full Text] [Related]
7. Comparison of sulfamate and sulfamide groups for the inhibition of carbonic anhydrase-II by using topiramate as a structural platform.
Maryanoff BE; McComsey DF; Costanzo MJ; Hochman C; Smith-Swintosky V; Shank RP
J Med Chem; 2005 Mar; 48(6):1941-7. PubMed ID: 15771438
[TBL] [Abstract][Full Text] [Related]
8. In vitro inhibition of α-carbonic anhydrase isozymes by some phenolic compounds.
Oztürk Sarikaya SB; Topal F; Sentürk M; Gülçin I; Supuran CT
Bioorg Med Chem Lett; 2011 Jul; 21(14):4259-62. PubMed ID: 21669522
[TBL] [Abstract][Full Text] [Related]
9. Sulfamates of methyl triterpenoates are effective and competitive inhibitors of carbonic anhydrase II.
Schwarz S; Sommerwerk S; Lucas SD; Heller L; Csuk R
Eur J Med Chem; 2014 Oct; 86():95-102. PubMed ID: 25147151
[TBL] [Abstract][Full Text] [Related]
10. Structures of human carbonic anhydrase II/inhibitor complexes reveal a second binding site for steroidal and nonsteroidal inhibitors.
Cozier GE; Leese MP; Lloyd MD; Baker MD; Thiyagarajan N; Acharya KR; Potter BV
Biochemistry; 2010 Apr; 49(16):3464-76. PubMed ID: 20297840
[TBL] [Abstract][Full Text] [Related]
11. S-glycosyl primary sulfonamides--a new structural class for selective inhibition of cancer-associated carbonic anhydrases.
Lopez M; Paul B; Hofmann A; Morizzi J; Wu QK; Charman SA; Innocenti A; Vullo D; Supuran CT; Poulsen SA
J Med Chem; 2009 Oct; 52(20):6421-32. PubMed ID: 19827837
[TBL] [Abstract][Full Text] [Related]
12. Sulfonamides incorporating 1,3,5-triazine moieties selectively and potently inhibit carbonic anhydrase transmembrane isoforms IX, XII and XIV over cytosolic isoforms I and II: Solution and X-ray crystallographic studies.
Carta F; Garaj V; Maresca A; Wagner J; Avvaru BS; Robbins AH; Scozzafava A; McKenna R; Supuran CT
Bioorg Med Chem; 2011 May; 19(10):3105-19. PubMed ID: 21515057
[TBL] [Abstract][Full Text] [Related]
13. Structure-activity studies on anticonvulsant sugar sulfamates related to topiramate. Enhanced potency with cyclic sulfate derivatives.
Maryanoff BE; Costanzo MJ; Nortey SO; Greco MN; Shank RP; Schupsky JJ; Ortegon MP; Vaught JL
J Med Chem; 1998 Apr; 41(8):1315-43. PubMed ID: 9548821
[TBL] [Abstract][Full Text] [Related]
14. Carbonic anhydrase inhibitors. DNA cloning, characterization, and inhibition studies of the human secretory isoform VI, a new target for sulfonamide and sulfamate inhibitors.
Nishimori I; Minakuchi T; Onishi S; Vullo D; Scozzafava A; Supuran CT
J Med Chem; 2007 Jan; 50(2):381-8. PubMed ID: 17228881
[TBL] [Abstract][Full Text] [Related]
15. Sulfamates and their therapeutic potential.
Winum JY; Scozzafava A; Montero JL; Supuran CT
Med Res Rev; 2005 Mar; 25(2):186-228. PubMed ID: 15478125
[TBL] [Abstract][Full Text] [Related]
16. Synthesis, structure and bioactivity of primary sulfamate-containing natural products.
Mujumdar P; Bua S; Supuran CT; Peat TS; Poulsen SA
Bioorg Med Chem Lett; 2018 Sep; 28(17):3009-3013. PubMed ID: 29685656
[TBL] [Abstract][Full Text] [Related]
17. Synthesis, characterization and antiglaucoma activity of a novel proton transfer compound and a mixed-ligand Zn(II) complex.
Yenikaya C; Sari M; Bülbül M; Ilkimen H; Celik H; Büyükgüngör O
Bioorg Med Chem; 2010 Jan; 18(2):930-8. PubMed ID: 20006931
[TBL] [Abstract][Full Text] [Related]
18. Structural basis for the interaction between carbonic anhydrase and 1,2,3,4-tetrahydroisoquinolin-2-ylsulfonamides.
Mader P; Brynda J; Gitto R; Agnello S; Pachl P; Supuran CT; Chimirri A; Řezáčová P
J Med Chem; 2011 Apr; 54(7):2522-6. PubMed ID: 21395315
[TBL] [Abstract][Full Text] [Related]
19. Carbonic anhydrase inhibitors: binding of indanesulfonamides to the human isoform II.
D'Ambrosio K; Masereel B; Thiry A; Scozzafava A; Supuran CT; De Simone G
ChemMedChem; 2008 Mar; 3(3):473-7. PubMed ID: 18161740
[TBL] [Abstract][Full Text] [Related]
20. Carbonic anhydrase inhibitors. X-ray crystal studies of the carbonic anhydrase II-trithiocarbonate adduct--an inhibitor mimicking the sulfonamide and urea binding to the enzyme.
Temperini C; Scozzafava A; Supuran CT
Bioorg Med Chem Lett; 2010 Jan; 20(2):474-8. PubMed ID: 20005709
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]
