135 related articles for article (PubMed ID: 21958118)
21. First crystal structures of human carbonic anhydrase II in complex with dual aromatase-steroid sulfatase inhibitors.
Lloyd MD; Thiyagarajan N; Ho YT; Woo LW; Sutcliffe OB; Purohit A; Reed MJ; Acharya KR; Potter BV
Biochemistry; 2005 May; 44(18):6858-66. PubMed ID: 15865431
[TBL] [Abstract][Full Text] [Related]
22. Carbonic anhydrase inhibitors: binding of an antiglaucoma glycosyl-sulfanilamide derivative to human isoform II and its consequences for the drug design of enzyme inhibitors incorporating sugar moieties.
Di Fiore A; Scozzafava A; Winum JY; Montero JL; Pedone C; Supuran CT; De Simone G
Bioorg Med Chem Lett; 2007 Mar; 17(6):1726-31. PubMed ID: 17251017
[TBL] [Abstract][Full Text] [Related]
23. 4-[N-(substituted 4-pyrimidinyl)amino]benzenesulfonamides as inhibitors of carbonic anhydrase isozymes I, II, VII, and XIII.
Sūdžius J; Baranauskienė L; Golovenko D; Matulienė J; Michailovienė V; Torresan J; Jachno J; Sukackaitė R; Manakova E; Gražulis S; Tumkevičius S; Matulis D
Bioorg Med Chem; 2010 Nov; 18(21):7413-21. PubMed ID: 20889345
[TBL] [Abstract][Full Text] [Related]
24. Virtual screening-driven identification of human carbonic anhydrase inhibitors incorporating an original, new pharmacophore.
Pala N; Dallocchio R; Dessì A; Brancale A; Carta F; Ihm S; Maresca A; Sechi M; Supuran CT
Bioorg Med Chem Lett; 2011 Apr; 21(8):2515-20. PubMed ID: 21420862
[TBL] [Abstract][Full Text] [Related]
25. Carbonic anhydrase inhibitors. Zonisamide is an effective inhibitor of the cytosolic isozyme II and mitochondrial isozyme V: solution and X-ray crystallographic studies.
De Simone G; Di Fiore A; Menchise V; Pedone C; Antel J; Casini A; Scozzafava A; Wurl M; Supuran CT
Bioorg Med Chem Lett; 2005 May; 15(9):2315-20. PubMed ID: 15837316
[TBL] [Abstract][Full Text] [Related]
26. NO-releasing esters show carbonic anhydrase inhibitory action against human isoforms I and II.
Ekinci D; Cavdar H; Talaz O; Sentürk M; Supuran CT
Bioorg Med Chem; 2010 May; 18(10):3559-63. PubMed ID: 20430631
[TBL] [Abstract][Full Text] [Related]
27. Carbonic anhydrase inhibitory activity and ocular pharmacology of organic sulfamates.
Brechue WF; Maren TH
J Pharmacol Exp Ther; 1993 Feb; 264(2):670-5. PubMed ID: 8437114
[TBL] [Abstract][Full Text] [Related]
28. Carbonic anhydrase inhibitors. Sulfonamide diuretics revisited--old leads for new applications?
Temperini C; Cecchi A; Scozzafava A; Supuran CT
Org Biomol Chem; 2008 Jul; 6(14):2499-506. PubMed ID: 18600270
[TBL] [Abstract][Full Text] [Related]
29. Carbonic anhydrase inhibitors: Valdecoxib binds to a different active site region of the human isoform II as compared to the structurally related cyclooxygenase II "selective" inhibitor celecoxib.
Di Fiore A; Pedone C; D'Ambrosio K; Scozzafava A; De Simone G; Supuran CT
Bioorg Med Chem Lett; 2006 Jan; 16(2):437-42. PubMed ID: 16290146
[TBL] [Abstract][Full Text] [Related]
30. Mechanistic Explanation of the Weak Carbonic Anhydrase's Esterase Activity.
Piazzetta P; Marino T; Russo N
Molecules; 2017 Jun; 22(6):. PubMed ID: 28629166
[TBL] [Abstract][Full Text] [Related]
31. Selective hydrophobic pocket binding observed within the carbonic anhydrase II active site accommodate different 4-substituted-ureido-benzenesulfonamides and correlate to inhibitor potency.
Pacchiano F; Aggarwal M; Avvaru BS; Robbins AH; Scozzafava A; McKenna R; Supuran CT
Chem Commun (Camb); 2010 Nov; 46(44):8371-3. PubMed ID: 20922253
[TBL] [Abstract][Full Text] [Related]
32. Carbonic anhydrase inhibitors: the X-ray crystal structure of ethoxzolamide complexed to human isoform II reveals the importance of thr200 and gln92 for obtaining tight-binding inhibitors.
Di Fiore A; Pedone C; Antel J; Waldeck H; Witte A; Wurl M; Scozzafava A; Supuran CT; De Simone G
Bioorg Med Chem Lett; 2008 Apr; 18(8):2669-74. PubMed ID: 18359629
[TBL] [Abstract][Full Text] [Related]
33. Ureido-substituted sulfamates show potent carbonic anhydrase IX inhibitory and antiproliferative activities against breast cancer cell lines.
Winum JY; Carta F; Ward C; Mullen P; Harrison D; Langdon SP; Cecchi A; Scozzafava A; Kunkler I; Supuran CT
Bioorg Med Chem Lett; 2012 Jul; 22(14):4681-5. PubMed ID: 22721713
[TBL] [Abstract][Full Text] [Related]
34. Carbonic anhydrase inhibitors. The X-ray crystal structure of human isoform II in adduct with an adamantyl analogue of acetazolamide resides in a less utilized binding pocket than most hydrophobic inhibitors.
Avvaru BS; Wagner JM; Maresca A; Scozzafava A; Robbins AH; Supuran CT; McKenna R
Bioorg Med Chem Lett; 2010 Aug; 20(15):4376-81. PubMed ID: 20605094
[TBL] [Abstract][Full Text] [Related]
35. Effects of new 5-amino-1,3,4-thiadiazole-2-sulfonamide derivatives on human carbonic anhydrase isozymes.
Kasimoğullari R; Bülbül M; Günhan H; Güleryüz H
Bioorg Med Chem; 2009 May; 17(9):3295-301. PubMed ID: 19362844
[TBL] [Abstract][Full Text] [Related]
36. Inhibition profiling of human carbonic anhydrase II by high-throughput screening of structurally diverse, biologically active compounds.
Iyer R; Barrese AA; Parakh S; Parker CN; Tripp BC
J Biomol Screen; 2006 Oct; 11(7):782-91. PubMed ID: 16858005
[TBL] [Abstract][Full Text] [Related]
37. Design, synthesis, and docking studies of new 1,3,4-thiadiazole-2-thione derivatives with carbonic anhydrase inhibitory activity.
Abdel-Hamid MK; Abdel-Hafez AA; El-Koussi NA; Mahfouz NM; Innocenti A; Supuran CT
Bioorg Med Chem; 2007 Nov; 15(22):6975-84. PubMed ID: 17822907
[TBL] [Abstract][Full Text] [Related]
38. Screening derivatized peptide libraries for tight binding inhibitors to carbonic anhydrase II by electrospray ionization-mass spectrometry.
Gao J; Cheng X; Chen R; Sigal GB; Bruce JE; Schwartz BL; Hofstadler SA; Anderson GA; Smith RD; Whitesides GM
J Med Chem; 1996 May; 39(10):1949-55. PubMed ID: 8642553
[TBL] [Abstract][Full Text] [Related]
39. An overview of carbohydrate-based carbonic anhydrase inhibitors.
Cuffaro D; Nuti E; Rossello A
J Enzyme Inhib Med Chem; 2020 Dec; 35(1):1906-1922. PubMed ID: 33078634
[TBL] [Abstract][Full Text] [Related]
40. Synthesis and characterisation of two novel proton transfer compounds and their inhibition studies on carbonic anhydrase isoenzymes.
Yenikaya C; Sari M; Bülbül M; Ilkimen H; Cinar B; Büyükgüngör O
J Enzyme Inhib Med Chem; 2011 Feb; 26(1):104-14. PubMed ID: 20860527
[TBL] [Abstract][Full Text] [Related]
[Previous] [Next] [New Search]