These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.
97 related articles for article (PubMed ID: 21987304)
21. Synthesis and functional characterization of imbutamine analogs as histamine H3 and H4 receptor ligands. Geyer R; Kaske M; Baumeister P; Buschauer A Arch Pharm (Weinheim); 2014 Feb; 347(2):77-88. PubMed ID: 24493592 [TBL] [Abstract][Full Text] [Related]
22. N(alpha)-imidazolylalkyl and pyridylalkyl derivatives of histaprodifen: synthesis and in vitro evaluation of highly potent histamine H(1)-receptor agonists. Menghin S; Pertz HH; Kramer K; Seifert R; Schunack W; Elz S J Med Chem; 2003 Dec; 46(25):5458-70. PubMed ID: 14640554 [TBL] [Abstract][Full Text] [Related]
23. Cyclopropane-based stereochemical diversity-oriented conformational restriction strategy: histamine H3 and/or H4 receptor ligands with the 2,3-methanobutane backbone. Watanabe M; Kobayashi T; Hirokawa T; Yoshida A; Ito Y; Yamada S; Orimoto N; Yamasaki Y; Arisawa M; Shuto S Org Biomol Chem; 2012 Jan; 10(4):736-45. PubMed ID: 22120611 [TBL] [Abstract][Full Text] [Related]
24. Cyclopropane-based conformational restriction of histamine. (1S,2S)-2-(2-aminoethyl)-1-(1H-imidazol-4-yl)cyclopropane, a highly selective agonist for the histamine H3 receptor, having a cis-cyclopropane structure. Kazuta Y; Hirano K; Natsume K; Yamada S; Kimura R; Matsumoto S; Furuichi K; Matsuda A; Shuto S J Med Chem; 2003 May; 46(10):1980-8. PubMed ID: 12723960 [TBL] [Abstract][Full Text] [Related]
25. Histamine H4 receptor agonists. Igel P; Dove S; Buschauer A Bioorg Med Chem Lett; 2010 Dec; 20(24):7191-9. PubMed ID: 21044842 [TBL] [Abstract][Full Text] [Related]
26. Influence of the N-terminus and the E2-loop onto the binding kinetics of the antagonist mepyramine and the partial agonist phenoprodifen to H(1)R. Wittmann HJ; Seifert R; Strasser A Biochem Pharmacol; 2011 Dec; 82(12):1910-8. PubMed ID: 21933664 [TBL] [Abstract][Full Text] [Related]
27. Stereochemical diversity-oriented conformational restriction strategy. Development of potent histamine H3 and/or H4 receptor antagonists with an imidazolylcyclopropane structure. Watanabe M; Kazuta Y; Hayashi H; Yamada S; Matsuda A; Shuto S J Med Chem; 2006 Sep; 49(18):5587-96. PubMed ID: 16942032 [TBL] [Abstract][Full Text] [Related]
28. Pharmacological profile of histaprodifens at four recombinant histamine H1 receptor species isoforms. Strasser A; Striegl B; Wittmann HJ; Seifert R J Pharmacol Exp Ther; 2008 Jan; 324(1):60-71. PubMed ID: 17928567 [TBL] [Abstract][Full Text] [Related]
29. Acylguanidines as bioisosteres of guanidines: NG-acylated imidazolylpropylguanidines, a new class of histamine H2 receptor agonists. Ghorai P; Kraus A; Keller M; Götte C; Igel P; Schneider E; Schnell D; Bernhardt G; Dove S; Zabel M; Elz S; Seifert R; Buschauer A J Med Chem; 2008 Nov; 51(22):7193-204. PubMed ID: 18950149 [TBL] [Abstract][Full Text] [Related]
30. A selective human H(4)-receptor agonist: (-)-2-cyano-1-methyl-3-[(2R,5R)-5- [1H-imidazol-4(5)-yl]tetrahydrofuran-2-y] methylguanidine. Hashimoto T; Harusawa S; Araki L; Zuiderveld OP; Smit MJ; Imazu T; Takashima S; Yamamoto Y; Sakamoto Y; Kurihara T; Leurs R; Bakker RA; Yamatodani A J Med Chem; 2003 Jul; 46(14):3162-5. PubMed ID: 12825954 [TBL] [Abstract][Full Text] [Related]
31. 4-(omega-(alkyloxy)alkyl)-1H-imidazole derivatives as histamine H(3) receptor antagonists/agonists. Meier G; Krause M; Hüls A; Ligneau X; Pertz HH; Arrang JM; Ganellin CR; Schwartz JC; Schunack W; Stark H J Med Chem; 2004 May; 47(10):2678-87. PubMed ID: 15115409 [TBL] [Abstract][Full Text] [Related]
32. Optimization of 5-pyridazin-3-one phenoxypropylamines as potent, selective histamine H₃ receptor antagonists with potent cognition enhancing activity. Tao M; Aimone LD; Huang Z; Mathiasen J; Raddatz R; Lyons J; Hudkins RL J Med Chem; 2012 Jan; 55(1):414-23. PubMed ID: 22107017 [TBL] [Abstract][Full Text] [Related]
33. Discovery of quinazolines as histamine H4 receptor inverse agonists using a scaffold hopping approach. Smits RA; de Esch IJ; Zuiderveld OP; Broeker J; Sansuk K; Guaita E; Coruzzi G; Adami M; Haaksma E; Leurs R J Med Chem; 2008 Dec; 51(24):7855-65. PubMed ID: 19053770 [TBL] [Abstract][Full Text] [Related]
34. Modulation of histamine H(3) receptor function by monovalent ions. Schnell D; Seifert R Neurosci Lett; 2010 Mar; 472(2):114-8. PubMed ID: 20132865 [TBL] [Abstract][Full Text] [Related]
35. Ligand-specific contribution of the N terminus and E2-loop to pharmacological properties of the histamine H1-receptor. Strasser A; Wittmann HJ; Seifert R J Pharmacol Exp Ther; 2008 Sep; 326(3):783-91. PubMed ID: 18577700 [TBL] [Abstract][Full Text] [Related]
36. Effects of impromidine- and arpromidine-derived guanidines on recombinant human and guinea pig histamine H1 and H2 receptors. Xie SX; Schalkhausser F; Ye QZ; Seifert R; Buschauer A Arch Pharm (Weinheim); 2007 Jan; 340(1):9-16. PubMed ID: 17206612 [TBL] [Abstract][Full Text] [Related]
37. Synthesis and pharmacological identification of neutral histamine H1-receptor antagonists. Govoni M; Bakker RA; van de Wetering I; Smit MJ; Menge WM; Timmerman H; Elz S; Schunack W; Leurs R J Med Chem; 2003 Dec; 46(26):5812-24. PubMed ID: 14667234 [TBL] [Abstract][Full Text] [Related]
38. Synthesis and evaluation of novel ligands for the histamine H₄ receptor based on a pyrrolo[2,3-d]pyrimidine scaffold. Gao LJ; Schwed JS; Weizel L; De Jonghe S; Stark H; Herdewijn P Bioorg Med Chem Lett; 2013 Jan; 23(1):132-7. PubMed ID: 23218604 [TBL] [Abstract][Full Text] [Related]
39. N (α)-Methylated phenylhistamines exhibit affinity to the hH(4)R-a pharmacological and molecular modelling study. Wittmann HJ; Elz S; Seifert R; Straber A Naunyn Schmiedebergs Arch Pharmacol; 2011 Sep; 384(3):287-99. PubMed ID: 21800095 [TBL] [Abstract][Full Text] [Related]
40. New high affinity H3 receptor agonists without a basic side chain. Kitbunnadaj R; Hoffmann M; Fratantoni SA; Bongers G; Bakker RA; Wieland K; el Jilali A; De Esch IJ; Menge WM; Timmerman H; Leurs R Bioorg Med Chem; 2005 Dec; 13(23):6309-23. PubMed ID: 16213736 [TBL] [Abstract][Full Text] [Related] [Previous] [Next] [New Search]