190 related articles for article (PubMed ID: 2202831)
1. Antimalarial activity of new water-soluble dihydroartemisinin derivatives. 3. Aromatic amine analogues.
Lin AJ; Li LQ; Klayman DL; George CF; Flippen-Anderson JL
J Med Chem; 1990 Sep; 33(9):2610-4. PubMed ID: 2202831
[TBL] [Abstract][Full Text] [Related]
2. Antimalarial activity of new dihydroartemisinin derivatives. 5. Sugar analogues.
Lin AJ; Li LQ; Andersen SL; Klayman DL
J Med Chem; 1992 May; 35(9):1639-42. PubMed ID: 1578492
[TBL] [Abstract][Full Text] [Related]
3. Antimalarial activity of new water-soluble dihydroartemisinin derivatives.
Lin AJ; Klayman DL; Milhous WK
J Med Chem; 1987 Nov; 30(11):2147-50. PubMed ID: 3669021
[TBL] [Abstract][Full Text] [Related]
4. Antimalarial activity of new dihydroartemisinin derivatives. 7. 4-(p-substituted phenyl)-4(R or S)-[10(alpha or beta)-dihydroartemisininoxy]butyric acids.
Lin AJ; Zikry AB; Kyle DE
J Med Chem; 1997 Apr; 40(9):1396-400. PubMed ID: 9135037
[TBL] [Abstract][Full Text] [Related]
5. Synthesis and antimalarial activities of fluoroalkyl derivatives of dihydroartemisinin.
Thanh Nga TT; Ménage C; Bégué JP; Bonnet-Delpon D; Gantier JC; Pradines B; Doury JC; Thac TD
J Med Chem; 1998 Oct; 41(21):4101-8. PubMed ID: 9767645
[TBL] [Abstract][Full Text] [Related]
6. Structure-activity relationships of the antimalarial agent artemisinin. 7. Direct modification of (+)-artemisinin and in vivo antimalarial screening of new, potential preclinical antimalarial candidates.
Avery MA; Alvim-Gaston M; Vroman JA; Wu B; Ager A; Peters W; Robinson BL; Charman W
J Med Chem; 2002 Sep; 45(19):4321-35. PubMed ID: 12213073
[TBL] [Abstract][Full Text] [Related]
7. Mechanism-based design of parasite-targeted artemisinin derivatives: synthesis and antimalarial activity of new diamine containing analogues.
Hindley S; Ward SA; Storr RC; Searle NL; Bray PG; Park BK; Davies J; O'Neill PM
J Med Chem; 2002 Feb; 45(5):1052-63. PubMed ID: 11855985
[TBL] [Abstract][Full Text] [Related]
8. Antimalarial activity of new water-soluble dihydroartemisinin derivatives. 2. Stereospecificity of the ether side chain.
Lin AJ; Lee M; Klayman DL
J Med Chem; 1989 Jun; 32(6):1249-52. PubMed ID: 2657065
[TBL] [Abstract][Full Text] [Related]
9. Antimalarial activity of novel ring-contracted artemisinin derivatives.
Venugopalan B; Bapat CP; Karnik PJ; Chatterjee DK; Iyer N; Lepcha D
J Med Chem; 1995 May; 38(11):1922-7. PubMed ID: 7783124
[TBL] [Abstract][Full Text] [Related]
10. Synthesis, antimalarial activity, biomimetic iron(II) chemistry, and in vivo metabolism of novel, potent C-10-phenoxy derivatives of dihydroartemisinin.
O'Neill PM; Miller A; Bishop LP; Hindley S; Maggs JL; Ward SA; Roberts SM; Scheinmann F; Stachulski AV; Posner GH; Park BK
J Med Chem; 2001 Jan; 44(1):58-68. PubMed ID: 11141088
[TBL] [Abstract][Full Text] [Related]
11. Syntheses and antimalarial activities of N-substituted 11-azaartemisinins.
Torok DS; Ziffer H; Meshnick SR; Pan XQ; Ager A
J Med Chem; 1995 Dec; 38(26):5045-50. PubMed ID: 8544181
[TBL] [Abstract][Full Text] [Related]
12. Synthesis and in vitro and in vivo antimalarial activity of new 4-anilinoquinolines.
Delarue S; Girault S; Maes L; Debreu-Fontaine MA; Labaeïd M; Grellier P; Sergheraert C
J Med Chem; 2001 Aug; 44(17):2827-33. PubMed ID: 11495593
[TBL] [Abstract][Full Text] [Related]
13. Antimalarial activity of dihydroartemisinin derivatives by transdermal application.
Lin AJ; Ager AL; Klayman DL
Am J Trop Med Hyg; 1994 Jun; 50(6):777-83. PubMed ID: 8024074
[TBL] [Abstract][Full Text] [Related]
14. Docking, synthesis and antimalarial activity of novel 4-anilinoquinoline derivatives.
Vijayaraghavan S; Mahajan S
Bioorg Med Chem Lett; 2017 Apr; 27(8):1693-1697. PubMed ID: 28318947
[TBL] [Abstract][Full Text] [Related]
15. Artemisinin derivatives bearing Mannich base group: synthesis and antimalarial activity.
Li Y; Yang ZS; Zhang H; Cao BJ; Wang FD; Zhang Y; Shi YL; Yang JD; Wu BA
Bioorg Med Chem; 2003 Oct; 11(20):4363-8. PubMed ID: 13129573
[TBL] [Abstract][Full Text] [Related]
16. Endoperoxides as potential antimalarial agents.
Kepler JA; Philip A; Lee YW; Musallam HA; Carroll FI
J Med Chem; 1987 Aug; 30(8):1505-9. PubMed ID: 3302259
[TBL] [Abstract][Full Text] [Related]
17. 2-Acetylpyridine thiosemicarbazones. 9. Derivatives of 2-acetylpyridine 1-oxide as potential antimalarial agents.
Scovill JP; Klayman DL; Lambros C; Childs GE; Notsch JD
J Med Chem; 1984 Jan; 27(1):87-91. PubMed ID: 6361258
[TBL] [Abstract][Full Text] [Related]
18. New quinoline derivatives demonstrate a promising antimalarial activity against Plasmodium falciparum in vitro and Plasmodium berghei in vivo.
Soares RR; da Silva JM; Carlos BC; da Fonseca CC; de Souza LS; Lopes FV; de Paula Dias RM; Moreira PO; Abramo C; Viana GH; de Pila Varotti F; da Silva AD; Scopel KK
Bioorg Med Chem Lett; 2015 Jun; 25(11):2308-13. PubMed ID: 25920564
[TBL] [Abstract][Full Text] [Related]
19. Antimalarial activity of new dihydroartemisinin derivatives. 6. alpha-Alkylbenzylic ethers.
Lin AJ; Miller RE
J Med Chem; 1995 Mar; 38(5):764-70. PubMed ID: 7877142
[TBL] [Abstract][Full Text] [Related]
20. Syntheses and antimalarial activities of 10-substituted deoxoartemisinins.
Ma J; Katz E; Kyle DE; Ziffer H
J Med Chem; 2000 Nov; 43(22):4228-32. PubMed ID: 11063619
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]