BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

155 related articles for article (PubMed ID: 22124202)

  • 1. Synthesis and screening of aromatase inhibitory activity of substituted C19 steroidal 17-oxime analogs.
    Pokhrel M; Ma E
    Molecules; 2011 Nov; 16(12):9868-85. PubMed ID: 22124202
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Synthesis of some epoxy and/or N-oxy 17-picolyl and 17-picolinylidene-androst-5-ene derivatives and evaluation of their biological activity.
    Djurendić E; Daljev J; Sakac M; Canadi J; Santa SJ; Andrić S; Klisurić O; Kojić V; Bogdanović G; Djurendić-Brenesel M; Novaković S; Gasi KP
    Steroids; 2008 Jan; 73(1):129-38. PubMed ID: 17963806
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Exploring new chemical functionalities to improve aromatase inhibition of steroids.
    Varela CL; Amaral C; Correia-da-Silva G; Costa SC; Carvalho RA; Costa G; Alcaro S; Teixeira NA; Tavares-da-Silva EJ; Roleira FM
    Bioorg Med Chem; 2016 Jun; 24(12):2823-31. PubMed ID: 27160054
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Synthesis of 19-oxygenated 4beta,5beta-epoxy derivatives of 16alpha-hydroxyandrostenedione as mechanistic and catalytic probes for aromatase reaction.
    Numazawa M; Yoshimura A
    Chem Pharm Bull (Tokyo); 2000 Sep; 48(9):1359-62. PubMed ID: 10993239
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Synthesis and aromatase inhibitory activity of some new 16E-arylidenosteroids.
    Bansal R; Thota S; Karkra N; Minu M; Zimmer C; Hartmann RW
    Bioorg Chem; 2012 Dec; 45():36-40. PubMed ID: 23064126
    [TBL] [Abstract][Full Text] [Related]  

  • 6. 6beta,19-Bridged androstenedione analogs as aromatase inhibitors.
    Komatsu S; Yaguchi A; Yamashita K; Nagaoka M; Numazawa M
    Steroids; 2009 Nov; 74(12):884-9. PubMed ID: 19524602
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Steroidal pyrazolines evaluated as aromatase and quinone reductase-2 inhibitors for chemoprevention of cancer.
    Abdalla MM; Al-Omar MA; Bhat MA; Amr AG; Al-Mohizea AM
    Int J Biol Macromol; 2012 May; 50(4):1127-32. PubMed ID: 22361454
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Synthesis and biochemical studies of 17-substituted androst-3-enes and 3,4-epoxyandrostanes as aromatase inhibitors.
    Cepa MM; Tavares da Silva EJ; Correia-da-Silva G; Roleira FM; Teixeira NA
    Steroids; 2008 Dec; 73(14):1409-15. PubMed ID: 18691607
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Synthesis and biological evaluation of 16E-arylidenosteroids as cytotoxic and anti-aromatase agents.
    Bansal R; Guleria S; Thota S; Hartmann RW; Zimmer C
    Chem Pharm Bull (Tokyo); 2011; 59(3):327-31. PubMed ID: 21372413
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Molecular mechanisms of aromatase inhibition by new A, D-ring modified steroids.
    Cepa M; Correia-da-Silva G; Tavares da Silva EJ; Roleira FM; Hong Y; Chen S; Teixeira NA
    Biol Chem; 2008 Sep; 389(9):1183-91. PubMed ID: 18713005
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Synthesis and 5α-reductase inhibitory activity of C₂₁ steroids having 1,4-diene or 4,6-diene 20-ones and 4-azasteroid 20-oximes.
    Kim S; Kim YU; Ma E
    Molecules; 2011 Dec; 17(1):355-68. PubMed ID: 22210173
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Synthesis and bioconversions of formestane.
    Martin GD; Narvaez J; Marti A
    J Nat Prod; 2013 Oct; 76(10):1966-9. PubMed ID: 24074257
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Molecular docking and QSAR study on steroidal compounds as aromatase inhibitors.
    Dai Y; Wang Q; Zhang X; Jia S; Zheng H; Feng D; Yu P
    Eur J Med Chem; 2010 Dec; 45(12):5612-20. PubMed ID: 20926163
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Design, synthesis, and antitumor activity evaluation of steroidal oximes.
    Gomes AR; Pires AS; Abrantes AM; Gonçalves AC; Costa SC; Varela CL; Silva ET; Botelho MF; Roleira FMF
    Bioorg Med Chem; 2021 Sep; 46():116360. PubMed ID: 34425478
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Steroidal Oximes: Useful Compounds with Antitumor Activities.
    Canario C; Silvestre S; Falcao A; Alves G
    Curr Med Chem; 2018 Feb; 25(6):660-686. PubMed ID: 28971759
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Synthesis of androst-5-en-7-ones and androsta-3,5-dien-7-ones and their related 7-deoxy analogs as conformational and catalytic probes for the active site of aromatase.
    Numazawa M; Mutsumi A; Tachibana M; Hoshi K
    J Med Chem; 1994 Jul; 37(14):2198-205. PubMed ID: 8035427
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Synthesis, structure elucidation, and biochemical evaluation of 7 alpha- and 7 beta-arylaliphatic-substituted androst-4-ene-3,17-diones as inhibitors of aromatase.
    O'Reilly JM; Li N; Duax WL; Brueggemeier RW
    J Med Chem; 1995 Jul; 38(15):2842-50. PubMed ID: 7636845
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Synthesis and anti-aromatase activity of some new steroidal D-lactones.
    Gasi KM; Stojanović SZ; Sakac MN; Popsavin M; Santa SJ; Stanković SM; Klisurić OR; Andrić N; Kovacević R
    Steroids; 2005 Jan; 70(1):47-53. PubMed ID: 15610896
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Studies of the time-dependent inactivation of aromatase by 4beta,5beta-epoxy-6-one and 5beta,6beta-epoxy-4-one steroids under various conditions.
    Numazawa M; Yamada K
    Biol Pharm Bull; 1999 Nov; 22(11):1207-11. PubMed ID: 10598029
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Synthesis and aromatase inhibitory evaluation of 4-N-nitrophenyl substituted amino-4H-1,2,4-triazole derivatives.
    Song Z; Liu Y; Dai Z; Liu W; Zhao K; Zhang T; Hu Y; Zhang X; Dai Y
    Bioorg Med Chem; 2016 Oct; 24(19):4723-4730. PubMed ID: 27567077
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 8.