146 related articles for article (PubMed ID: 22129594)
1. Characterization of COR627 and COR628, two novel positive allosteric modulators of the GABA(B) receptor.
Castelli MP; Casu A; Casti P; Lobina C; Carai MA; Colombo G; Solinas M; Giunta D; Mugnaini C; Pasquini S; Tafi A; Brogi S; Gessa GL; Corelli F
J Pharmacol Exp Ther; 2012 Mar; 340(3):529-38. PubMed ID: 22129594
[TBL] [Abstract][Full Text] [Related]
2. Synthesis and pharmacological characterization of 2-(acylamino)thiophene derivatives as metabolically stable, orally effective, positive allosteric modulators of the GABAB receptor.
Mugnaini C; Pedani V; Casu A; Lobina C; Casti A; Maccioni P; Porcu A; Giunta D; Lamponi S; Solinas M; Dragoni S; Valoti M; Colombo G; Castelli MP; Gessa GL; Corelli F
J Med Chem; 2013 May; 56(9):3620-35. PubMed ID: 23544432
[TBL] [Abstract][Full Text] [Related]
3. N,N'-Dicyclopentyl-2-methylsulfanyl-5-nitro-pyrimidine-4,6-diamine (GS39783) and structurally related compounds: novel allosteric enhancers of gamma-aminobutyric acidB receptor function.
Urwyler S; Pozza MF; Lingenhoehl K; Mosbacher J; Lampert C; Froestl W; Koller M; Kaupmann K
J Pharmacol Exp Ther; 2003 Oct; 307(1):322-30. PubMed ID: 12954816
[TBL] [Abstract][Full Text] [Related]
4. In vitro and in vivo characterization of the novel GABAB receptor positive allosteric modulator, 2-{1-[2-(4-chlorophenyl)-5-methylpyrazolo[1,5-a]pyrimidin-7-yl]-2-piperidinyl}ethanol (CMPPE).
Perdona' E; Costantini VJ; Tessari M; Martinelli P; Carignani C; Valerio E; Mok MH; Zonzini L; Visentini F; Gianotti M; Gordon L; Rocheville M; Corsi M; Capelli AM
Neuropharmacology; 2011; 61(5-6):957-66. PubMed ID: 21756923
[TBL] [Abstract][Full Text] [Related]
5. Influence of positive allosteric modulators on GABA(B) receptor coupling in rat brain: a scintillation proximity assay characterisation of G protein subtypes.
Mannoury la Cour C; Herbelles C; Pasteau V; de Nanteuil G; Millan MJ
J Neurochem; 2008 Apr; 105(2):308-23. PubMed ID: 18021295
[TBL] [Abstract][Full Text] [Related]
6. Differential regulation of GABA B receptor subunit expression and function.
Sands SA; McCarson KE; Enna SJ
J Pharmacol Exp Ther; 2003 Apr; 305(1):191-6. PubMed ID: 12649368
[TBL] [Abstract][Full Text] [Related]
7. GABA(B) receptor modulators potentiate baclofen-induced depression of dopamine neuron activity in the rat ventral tegmental area.
Chen Y; Phillips K; Minton G; Sher E
Br J Pharmacol; 2005 Apr; 144(7):926-32. PubMed ID: 15711597
[TBL] [Abstract][Full Text] [Related]
8. Positive allosteric modulation of native and recombinant gamma-aminobutyric acid(B) receptors by 2,6-Di-tert-butyl-4-(3-hydroxy-2,2-dimethyl-propyl)-phenol (CGP7930) and its aldehyde analog CGP13501.
Urwyler S; Mosbacher J; Lingenhoehl K; Heid J; Hofstetter K; Froestl W; Bettler B; Kaupmann K
Mol Pharmacol; 2001 Nov; 60(5):963-71. PubMed ID: 11641424
[TBL] [Abstract][Full Text] [Related]
9. Effects of GABA(B) receptor antagonist, agonists and allosteric positive modulator on the cocaine-induced self-administration and drug discrimination.
Filip M; Frankowska M; Przegaliński E
Eur J Pharmacol; 2007 Nov; 574(2-3):148-57. PubMed ID: 17698060
[TBL] [Abstract][Full Text] [Related]
10. Up-regulation of GABA(B) receptors by chronic administration of the GABA(B) receptor antagonist SCH 50,911.
Pibiri F; Carboni G; Carai MA; Gessa GL; Castelli MP
Eur J Pharmacol; 2005 May; 515(1-3):94-8. PubMed ID: 15893746
[TBL] [Abstract][Full Text] [Related]
11. In vitro and in vivo pharmacological characterization of SSD114, a novel GABAB positive allosteric modulator.
Porcu A; Lobina C; Giunta D; Solinas M; Mugnaini C; Castelli MP
Eur J Pharmacol; 2016 Nov; 791():115-123. PubMed ID: 27578262
[TBL] [Abstract][Full Text] [Related]
12. Effects of intraperitoneal administration of the GABAB receptor positive allosteric modulator 2,6-di tert-butyl-4-(2-hydroxy-2,2-dimethyl-propyl)-phenol (CGP7930) on food intake in non-deprived rats.
Ebenezer IS
Eur J Pharmacol; 2012 Sep; 690(1-3):115-8. PubMed ID: 22652431
[TBL] [Abstract][Full Text] [Related]
13. Role of the GABA(B) receptor in alcohol-seeking and drinking behavior.
Maccioni P; Colombo G
Alcohol; 2009 Nov; 43(7):555-8. PubMed ID: 19913200
[TBL] [Abstract][Full Text] [Related]
14. Anticonvulsant effects of structurally diverse GABA(B) positive allosteric modulators in the DBA/2J audiogenic seizure test: Comparison to baclofen and utility as a pharmacodynamic screening model.
Brown JW; Moeller A; Schmidt M; Turner SC; Nimmrich V; Ma J; Rueter LE; van der Kam E; Zhang M
Neuropharmacology; 2016 Feb; 101():358-69. PubMed ID: 26471422
[TBL] [Abstract][Full Text] [Related]
15. Allosteric modulation of GABA(B) receptor function in human frontal cortex.
Olianas MC; Ambu R; Garau L; Onali P
Neurochem Int; 2005 Jan; 46(2):149-58. PubMed ID: 15627515
[TBL] [Abstract][Full Text] [Related]
16. Positive allosteric modulators at GABAB receptors exert intrinsic actions and enhance the influence of baclofen on light-induced phase shifts of hamster circadian activity rhythms.
Gannon RL; Millan MJ
Pharmacol Biochem Behav; 2011 Oct; 99(4):712-7. PubMed ID: 21756929
[TBL] [Abstract][Full Text] [Related]
17. (R)-(3-amino-2-fluoropropyl) phosphinic acid (AZD3355), a novel GABAB receptor agonist, inhibits transient lower esophageal sphincter relaxation through a peripheral mode of action.
Lehmann A; Antonsson M; Holmberg AA; Blackshaw LA; Brändén L; Bräuner-Osborne H; Christiansen B; Dent J; Elebring T; Jacobson BM; Jensen J; Mattsson JP; Nilsson K; Oja SS; Page AJ; Saransaari P; von Unge S
J Pharmacol Exp Ther; 2009 Nov; 331(2):504-12. PubMed ID: 19648470
[TBL] [Abstract][Full Text] [Related]
18. The GABA(B) antagonist CGP56433A attenuates the effect of baclofen on cocaine but not heroin self-administration in the rat.
Brebner K; Froestl W; Roberts DC
Psychopharmacology (Berl); 2002 Feb; 160(1):49-55. PubMed ID: 11862373
[TBL] [Abstract][Full Text] [Related]
19. Characterization of the binding of [3H]CGP54626 to GABAB receptors in the male bullfrog (Rana catesbeiana).
Asay MJ; Boyd SK
Brain Res; 2006 Jun; 1094(1):76-85. PubMed ID: 16725130
[TBL] [Abstract][Full Text] [Related]
20. GABAB receptor-positive modulators: brain region-dependent effects.
Hensler JG; Advani T; Burke TF; Cheng K; Rice KC; Koek W
J Pharmacol Exp Ther; 2012 Jan; 340(1):19-26. PubMed ID: 21954301
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]
