These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.


BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

197 related articles for article (PubMed ID: 22248858)

  • 1. Synthesis and antikinetoplastid activity of a series of N,N'-substituted diamines.
    Caminos AP; Panozzo-Zenere EA; Wilkinson SR; Tekwani BL; Labadie GR
    Bioorg Med Chem Lett; 2012 Feb; 22(4):1712-5. PubMed ID: 22248858
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Design, synthesis and evaluation of 2,4-diaminoquinazolines as inhibitors of trypanosomal and leishmanial dihydrofolate reductase.
    Khabnadideh S; Pez D; Musso A; Brun R; Pérez LM; González-Pacanowska D; Gilbert IH
    Bioorg Med Chem; 2005 Apr; 13(7):2637-49. PubMed ID: 15755663
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Preparation and antileishmanial activity of lipophilic N-alkyl diamines.
    da Costa CF; Coimbra ES; Braga FG; dos Reis RC; da Silva AD; de Almeida MV
    Biomed Pharmacother; 2009 Jan; 63(1):40-2. PubMed ID: 18262385
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Screening strategies to identify new chemical diversity for drug development to treat kinetoplastid infections.
    Don R; Ioset JR
    Parasitology; 2014 Jan; 141(1):140-6. PubMed ID: 23985066
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Antikinetoplastid antimitotic activity and metabolic stability of dinitroaniline sulfonamides and benzamides.
    George TG; Johnsamuel J; Delfín DA; Yakovich A; Mukherjee M; Phelps MA; Dalton JT; Sackett DL; Kaiser M; Brun R; Werbovetz KA
    Bioorg Med Chem; 2006 Aug; 14(16):5699-710. PubMed ID: 16675220
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Biological evaluation and structure-activity relationships of imidazole-based compounds as antiprotozoal agents.
    Saccoliti F; Madia VN; Tudino V; De Leo A; Pescatori L; Messore A; De Vita D; Scipione L; Brun R; Kaiser M; Mäser P; Calvet CM; Jennings GK; Podust LM; Costi R; Di Santo R
    Eur J Med Chem; 2018 Aug; 156():53-60. PubMed ID: 30006174
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Synthesis and in vitro antikinetoplastid activity of polyamine-hydroxybenzotriazole conjugates.
    Jagu E; Pomel S; Diez-Martinez A; Ramiandrasoa F; Krauth-Siegel RL; Pethe S; Blonski C; Labruère R; Loiseau PM
    Bioorg Med Chem; 2017 Jan; 25(1):84-90. PubMed ID: 27793448
    [TBL] [Abstract][Full Text] [Related]  

  • 8. SAR refinement of antileishmanial N(2),N(4)-disubstituted quinazoline-2,4-diamines.
    Zhu X; Van Horn KS; Barber MM; Yang S; Wang MZ; Manetsch R; Werbovetz KA
    Bioorg Med Chem; 2015 Aug; 23(16):5182-9. PubMed ID: 25749014
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Synthesis and characterization of a pyridine-2-thiol N-oxide gold(I) complex with potent antiproliferative effect against Trypanosoma cruzi and Leishmania sp. insight into its mechanism of action.
    Vieites M; Smircich P; Guggeri L; Marchán E; Gómez-Barrio A; Navarro M; Garat B; Gambino D
    J Inorg Biochem; 2009 Oct; 103(10):1300-6. PubMed ID: 19361864
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Synthesis, cytotoxicity, and in vitro antileishmanial activity of mono-t-butyloxycarbonyl-protected diamines.
    Pinheiro AC; Rocha MN; Nogueira PM; Nogueira TC; Jasmim LF; de Souza MV; Soares RP
    Diagn Microbiol Infect Dis; 2011 Nov; 71(3):273-8. PubMed ID: 21907525
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Design, synthesis and in vitro antikinetoplastid evaluation of N-acylated putrescine, spermidine and spermine derivatives.
    Jagu E; Djilali R; Pomel S; Ramiandrasoa F; Pethe S; Labruère R; Loiseau PM; Blonski C
    Bioorg Med Chem Lett; 2015 Jan; 25(2):207-9. PubMed ID: 25499437
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Screening a Natural Product-Based Library against Kinetoplastid Parasites.
    Zulfiqar B; Jones AJ; Sykes ML; Shelper TB; Davis RA; Avery VM
    Molecules; 2017 Oct; 22(10):. PubMed ID: 29023425
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Synthesis and tripanocidal activity of ferrocenyl and benzyl diamines against Trypanosoma brucei and Trypanosoma cruzi.
    Velásquez AM; Francisco AI; Kohatsu AA; Silva FA; Rodrigues DF; Teixeira RG; Chiari BG; de Almeida MG; Isaac VL; Vargas MD; Cicarelli RM
    Bioorg Med Chem Lett; 2014 Apr; 24(7):1707-10. PubMed ID: 24630563
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Potent antiprotozoal activity of a novel semi-synthetic berberine derivative.
    Bahar M; Deng Y; Zhu X; He S; Pandharkar T; Drew ME; Navarro-Vázquez A; Anklin C; Gil RR; Doskotch RW; Werbovetz KA; Kinghorn AD
    Bioorg Med Chem Lett; 2011 May; 21(9):2606-10. PubMed ID: 21474310
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Antitrypanosomal and cysteine protease inhibitory activities of alkyldiamine cryptolepine derivatives.
    Lavrado J; Mackey Z; Hansell E; McKerrow JH; Paulo A; Moreira R
    Bioorg Med Chem Lett; 2012 Oct; 22(19):6256-60. PubMed ID: 22926067
    [TBL] [Abstract][Full Text] [Related]  

  • 16. High-throughput screening platform for natural product-based drug discovery against 3 neglected tropical diseases: human African trypanosomiasis, leishmaniasis, and Chagas disease.
    Annang F; Pérez-Moreno G; García-Hernández R; Cordon-Obras C; Martín J; Tormo JR; Rodríguez L; de Pedro N; Gómez-Pérez V; Valente M; Reyes F; Genilloud O; Vicente F; Castanys S; Ruiz-Pérez LM; Navarro M; Gamarro F; González-Pacanowska D
    J Biomol Screen; 2015 Jan; 20(1):82-91. PubMed ID: 25332350
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Synthesis of a small library of 2-phenoxy-1,4-naphthoquinone and 2-phenoxy-1,4-anthraquinone derivatives bearing anti-trypanosomal and anti-leishmanial activity.
    Bolognesi ML; Lizzi F; Perozzo R; Brun R; Cavalli A
    Bioorg Med Chem Lett; 2008 Apr; 18(7):2272-6. PubMed ID: 18353643
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Infectious diseases. Overcoming neglect of kinetoplastid diseases.
    Bilbe G
    Science; 2015 May; 348(6238):974-6. PubMed ID: 26023124
    [No Abstract]   [Full Text] [Related]  

  • 19. Synthesis, biological evaluation, and molecular modeling of 3,5-substituted-N1-phenyl-N4,N4-di-n-butylsulfanilamides as antikinetoplastid antimicrotubule agents.
    George TG; Endeshaw MM; Morgan RE; Mahasenan KV; Delfín DA; Mukherjee MS; Yakovich AJ; Fotie J; Li C; Werbovetz KA
    Bioorg Med Chem; 2007 Sep; 15(18):6071-9. PubMed ID: 17618122
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Squalamine analogues as potential anti-trypanosomal and anti-leishmanial compounds.
    Khabnadideh S; Tan CL; Croft SL; Kendrick H; Yardley V; Gilbert IH
    Bioorg Med Chem Lett; 2000 Jun; 10(11):1237-9. PubMed ID: 10866389
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 10.