These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.


BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

131 related articles for article (PubMed ID: 22330635)

  • 1. Discovery of vinylcycloalkyl-substituted benzimidazole TRPM8 antagonists effective in the treatment of cold allodynia.
    Calvo RR; Meegalla SK; Parks DJ; Parsons WH; Ballentine SK; Lubin ML; Schneider C; Colburn RW; Flores CM; Player MR
    Bioorg Med Chem Lett; 2012 Mar; 22(5):1903-7. PubMed ID: 22330635
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Design and optimization of benzimidazole-containing transient receptor potential melastatin 8 (TRPM8) antagonists.
    Parks DJ; Parsons WH; Colburn RW; Meegalla SK; Ballentine SK; Illig CR; Qin N; Liu Y; Hutchinson TL; Lubin ML; Stone DJ; Baker JF; Schneider CR; Ma J; Damiano BP; Flores CM; Player MR
    J Med Chem; 2011 Jan; 54(1):233-47. PubMed ID: 21128593
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Evaluation of milnacipran, in comparison with amitriptyline, on cold and mechanical allodynia in a rat model of neuropathic pain.
    Berrocoso E; Mico JA; Vitton O; Ladure P; Newman-Tancredi A; Depoortère R; Bardin L
    Eur J Pharmacol; 2011 Mar; 655(1-3):46-51. PubMed ID: 21277295
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Antinociceptive activity of transient receptor potential channel TRPV1, TRPA1, and TRPM8 antagonists in neurogenic and neuropathic pain models in mice.
    Sałat K; Filipek B
    J Zhejiang Univ Sci B; 2015 Mar; 16(3):167-78. PubMed ID: 25743118
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Fused piperidines as a novel class of potent and orally available transient receptor potential melastatin type 8 (TRPM8) antagonists.
    Tamayo NA; Bo Y; Gore V; Ma V; Nishimura N; Tang P; Deng H; Klionsky L; Lehto SG; Wang W; Youngblood B; Chen J; Correll TL; Bartberger MD; Gavva NR; Norman MH
    J Med Chem; 2012 Feb; 55(4):1593-611. PubMed ID: 22329507
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Antinociceptive effect of two novel transient receptor potential melastatin 8 antagonists in acute and chronic pain models in rat.
    De Caro C; Russo R; Avagliano C; Cristiano C; Calignano A; Aramini A; Bianchini G; Allegretti M; Brandolini L
    Br J Pharmacol; 2018 May; 175(10):1691-1706. PubMed ID: 29485712
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Ethosuximide reduces allodynia and hyperalgesia and potentiates morphine effects in the chronic constriction injury model of neuropathic pain.
    Hamidi GA; Ramezani MH; Arani MN; Talaei SA; Mesdaghinia A; Banafshe HR
    Eur J Pharmacol; 2012 Jan; 674(2-3):260-4. PubMed ID: 22134003
    [TBL] [Abstract][Full Text] [Related]  

  • 8. TRPM8 mechanism of cold allodynia after chronic nerve injury.
    Xing H; Chen M; Ling J; Tan W; Gu JG
    J Neurosci; 2007 Dec; 27(50):13680-90. PubMed ID: 18077679
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Role of TRPM8 in dorsal root ganglion in nerve injury-induced chronic pain.
    Su L; Wang C; Yu YH; Ren YY; Xie KL; Wang GL
    BMC Neurosci; 2011 Nov; 12():120. PubMed ID: 22111979
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Identification of a Potent Tryptophan-Based TRPM8 Antagonist With in Vivo Analgesic Activity.
    Bertamino A; Iraci N; Ostacolo C; Ambrosino P; Musella S; Di Sarno V; Ciaglia T; Pepe G; Sala M; Soldovieri MV; Mosca I; Gonzalez-Rodriguez S; Fernandez-Carvajal A; Ferrer-Montiel A; Novellino E; Taglialatela M; Campiglia P; Gomez-Monterrey I
    J Med Chem; 2018 Jul; 61(14):6140-6152. PubMed ID: 29939028
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Amelioration of neuropathic pain by novel transient receptor potential vanilloid 1 antagonist AS1928370 in rats without hyperthermic effect.
    Watabiki T; Kiso T; Kuramochi T; Yonezawa K; Tsuji N; Kohara A; Kakimoto S; Aoki T; Matsuoka N
    J Pharmacol Exp Ther; 2011 Mar; 336(3):743-50. PubMed ID: 21098091
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Exploration of TRPM8 Binding Sites by β-Carboline-Based Antagonists and Their In Vitro Characterization and In Vivo Analgesic Activities.
    Bertamino A; Ostacolo C; Medina A; Di Sarno V; Lauro G; Ciaglia T; Vestuto V; Pepe G; Basilicata MG; Musella S; Smaldone G; Cristiano C; Gonzalez-Rodriguez S; Fernandez-Carvajal A; Bifulco G; Campiglia P; Gomez-Monterrey I; Russo R
    J Med Chem; 2020 Sep; 63(17):9672-9694. PubMed ID: 32787109
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Anti-hyperalgesic effects of a novel TRPM8 agonist in neuropathic rats: a comparison with topical menthol.
    Patel R; Gonçalves L; Leveridge M; Mack SR; Hendrick A; Brice NL; Dickenson AH
    Pain; 2014 Oct; 155(10):2097-107. PubMed ID: 25083927
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Involvement of increased expression of transient receptor potential melastatin 8 in oxaliplatin-induced cold allodynia in mice.
    Gauchan P; Andoh T; Kato A; Kuraishi Y
    Neurosci Lett; 2009 Jul; 458(2):93-5. PubMed ID: 19375484
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Arylglycine derivatives as potent transient receptor potential melastatin 8 (TRPM8) antagonists.
    Zhu B; Xia M; Xu X; Ludovici DW; Tennakoon M; Youngman MA; Matthews JM; Dax SL; Colburn RW; Qin N; Hutchinson TL; Lubin ML; Brandt MR; Stone DJ; Flores CM; Macielag MJ
    Bioorg Med Chem Lett; 2013 Apr; 23(7):2234-7. PubMed ID: 23411075
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Antinociceptive Effects of Isosakuranetin in a Rat Model of Peripheral Neuropathy.
    Jia S; Zhang Y; Yu J
    Pharmacology; 2017; 100(3-4):201-207. PubMed ID: 28715803
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Synthesis and pharmacological evaluation of novel N-aryl-3,4-dihydro-1'H-spiro[chromene-2,4'-piperidine]-1'-carboxamides as TRPM8 antagonists.
    Chaudhari SS; Kadam AB; Khairatkar-Joshi N; Mukhopadhyay I; Karnik PV; Raghuram A; Rao SS; Vaiyapuri TS; Wale DP; Bhosale VM; Gudi GS; Sangana RR; Thomas A
    Bioorg Med Chem; 2013 Nov; 21(21):6542-53. PubMed ID: 24055075
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Optimization of potency and pharmacokinetic properties of tetrahydroisoquinoline transient receptor potential melastatin 8 (TRPM8) antagonists.
    Horne DB; Tamayo NA; Bartberger MD; Bo Y; Clarine J; Davis CD; Gore VK; Kaller MR; Lehto SG; Ma VV; Nishimura N; Nguyen TT; Tang P; Wang W; Youngblood BD; Zhang M; Gavva NR; Monenschein H; Norman MH
    J Med Chem; 2014 Apr; 57(7):2989-3004. PubMed ID: 24597733
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Menthol derivative WS-12 selectively activates transient receptor potential melastatin-8 (TRPM8) ion channels.
    Ma S; G G; Ak VE; Jf D; H H
    Pak J Pharm Sci; 2008 Oct; 21(4):370-8. PubMed ID: 18930858
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Gosha-jinki-gan reduced oxaliplatin-induced hypersensitivity to cold sensation and its effect would be related to suppression of the expression of TRPM8 and TRPA1 in rats.
    Kato Y; Tateai Y; Ohkubo M; Saito Y; Amagai SY; Kimura YS; Iimura N; Okada M; Matsumoto A; Mano Y; Hirosawa I; Ohuchi K; Tajima M; Asahi M; Kotaki H; Yamada H
    Anticancer Drugs; 2014 Jan; 25(1):39-43. PubMed ID: 24052105
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 7.