These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.
4. Structure-activity relationships of gamma-MSH analogues at the human melanocortin MC3, MC4, and MC5 receptors. Discovery of highly selective hMC3R, hMC4R, and hMC5R analogues. Balse-Srinivasan P; Grieco P; Cai M; Trivedi D; Hruby VJ J Med Chem; 2003 Nov; 46(23):4965-73. PubMed ID: 14584947 [TBL] [Abstract][Full Text] [Related]
5. Identification of putative agouti-related protein(87-132)-melanocortin-4 receptor interactions by homology molecular modeling and validation using chimeric peptide ligands. Wilczynski A; Wang XS; Joseph CG; Xiang Z; Bauzo RM; Scott JW; Sorensen NB; Shaw AM; Millard WJ; Richards NG; Haskell-Luevano C J Med Chem; 2004 Apr; 47(9):2194-207. PubMed ID: 15084118 [TBL] [Abstract][Full Text] [Related]
9. End-capping of the modified melanocortin tetrapeptide (p-Cl)Phe-D-Phe-Arg-Trp-NH2 as a route to hMC4R agonists. Koikov LN; Ebetino FH; Hayes JC; Cross-Doersen D; Knittel JJ Bioorg Med Chem Lett; 2004 Oct; 14(19):4839-42. PubMed ID: 15341935 [TBL] [Abstract][Full Text] [Related]
10. Novel alpha-melanocyte stimulating hormone peptide analogues with high candidacidal activity. Grieco P; Rossi C; Colombo G; Gatti S; Novellino E; Lipton JM; Catania A J Med Chem; 2003 Feb; 46(5):850-5. PubMed ID: 12593664 [TBL] [Abstract][Full Text] [Related]
11. N-terminal fatty acylated His-dPhe-Arg-Trp-NH(2) tetrapeptides: influence of fatty acid chain length on potency and selectivity at the mouse melanocortin receptors and human melanocytes. Todorovic A; Holder JR; Bauzo RM; Scott JW; Kavanagh R; Abdel-Malek Z; Haskell-Luevano C J Med Chem; 2005 May; 48(9):3328-36. PubMed ID: 15857138 [TBL] [Abstract][Full Text] [Related]
12. Potent and selective agonists of human melanocortin receptor 5: cyclic analogues of alpha-melanocyte-stimulating hormone. Bednarek MA; MacNeil T; Tang R; Fong TM; Cabello MA; Maroto M; Teran A J Med Chem; 2007 May; 50(10):2520-6. PubMed ID: 17455928 [TBL] [Abstract][Full Text] [Related]
13. Multimeric alpha-MSH has increased efficacy to activate the melanocortin MC4 receptor. Tiesjema B; Merkestein M; Garner KM; de Krom M; Adan RA Eur J Pharmacol; 2008 May; 585(1):24-30. PubMed ID: 18378226 [TBL] [Abstract][Full Text] [Related]
14. Analogs of alpha-melanocyte stimulating hormone with high agonist potency and selectivity at human melanocortin receptor 1b: the role of Trp(9) in molecular recognition. Bednarek MA; Macneil T; Tang R; Fong TM; Angeles Cabello M; Maroto M; Teran A Biopolymers; 2008 May; 89(5):401-8. PubMed ID: 17926329 [TBL] [Abstract][Full Text] [Related]
15. alpha-MSH and gamma-MSH inhibit IL-1beta induced activation of the hypothalamic-pituitary-adrenal axis through central melanocortin receptors. Cragnolini AB; Perelló M; Schiöth HB; Scimonelli TN Regul Pept; 2004 Nov; 122(3):185-90. PubMed ID: 15491790 [TBL] [Abstract][Full Text] [Related]
16. Discovery and structure-activity relationships of novel alpha-melanocyte-stimulating hormone inhibitors. Sawyer TK; Staples DJ; Castrucci AM; Hadley ME Pept Res; 1989; 2(1):140-6. PubMed ID: 2562482 [TBL] [Abstract][Full Text] [Related]
17. Functional selectivity of melanocortin 4 receptor peptide and nonpeptide agonists: evidence for ligand-specific conformational states. Nickolls SA; Fleck B; Hoare SR; Maki RA J Pharmacol Exp Ther; 2005 Jun; 313(3):1281-8. PubMed ID: 15743921 [TBL] [Abstract][Full Text] [Related]
18. Structure and function of the potent cyclic and linear melanocortin analogues. Cho MK; Lee CJ; Lee CH; Li SZ; Lim SK; Baik JH; Lee W J Struct Biol; 2005 Jun; 150(3):300-8. PubMed ID: 15890278 [TBL] [Abstract][Full Text] [Related]
19. Role of melanocortinergic neurons in feeding and the agouti obesity syndrome. Fan W; Boston BA; Kesterson RA; Hruby VJ; Cone RD Nature; 1997 Jan; 385(6612):165-8. PubMed ID: 8990120 [TBL] [Abstract][Full Text] [Related]
20. Potent and selective agonists of alpha-melanotropin (alphaMSH) action at human melanocortin receptor 5; linear analogs of alpha-melanotropin. Bednarek MA; MacNeil T; Tang R; Fong TM; Cabello MA; Maroto M; Teran A Peptides; 2007 May; 28(5):1020-8. PubMed ID: 17376561 [TBL] [Abstract][Full Text] [Related] [Next] [New Search]