BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

156 related articles for article (PubMed ID: 22377519)

  • 21. Design, synthesis, structure-activity relationships, and docking studies of 1-(γ-1,2,3-triazol substituted prolyl)-(S)-3,3-difluoropyrrolidines as a novel series of potent and selective dipeptidyl peptidase-4 inhibitors.
    Zhang L; Su M; Li J; Ji X; Wang J; Li Z; Li J; Liu H
    Chem Biol Drug Des; 2013 Feb; 81(2):198-207. PubMed ID: 22994702
    [TBL] [Abstract][Full Text] [Related]  

  • 22. Dipeptidyl peptidase 9 (DPP9) in human skin cells.
    Gabrilovac J; Čupić B; Zapletal E; Kraus O; Jakić-Razumović J
    Immunobiology; 2017 Feb; 222(2):327-342. PubMed ID: 27682012
    [TBL] [Abstract][Full Text] [Related]  

  • 23. Dipeptidyl peptidases in atherosclerosis: expression and role in macrophage differentiation, activation and apoptosis.
    Matheeussen V; Waumans Y; Martinet W; Van Goethem S; Van der Veken P; Scharpé S; Augustyns K; De Meyer GR; De Meester I
    Basic Res Cardiol; 2013 May; 108(3):350. PubMed ID: 23608773
    [TBL] [Abstract][Full Text] [Related]  

  • 24. Expression of dipeptidyl peptidase-IV activity and/or structure homologs in human meningiomas.
    Stremenová J; Mares V; Lisá V; Hilser M; Krepela E; Vanicková Z; Syrucek M; Soula O; Sedo A
    Int J Oncol; 2010 Feb; 36(2):351-8. PubMed ID: 20043068
    [TBL] [Abstract][Full Text] [Related]  

  • 25. Discovery, structure-activity relationship, and pharmacological evaluation of (5-substituted-pyrrolidinyl-2-carbonyl)-2-cyanopyrrolidines as potent dipeptidyl peptidase IV inhibitors.
    Pei Z; Li X; Longenecker K; von Geldern TW; Wiedeman PE; Lubben TH; Zinker BA; Stewart K; Ballaron SJ; Stashko MA; Mika AK; Beno DW; Long M; Wells H; Kempf-Grote AJ; Madar DJ; McDermott TS; Bhagavatula L; Fickes MG; Pireh D; Solomon LR; Lake MR; Edalji R; Fry EH; Sham HL; Trevillyan JM
    J Med Chem; 2006 Jun; 49(12):3520-35. PubMed ID: 16759095
    [TBL] [Abstract][Full Text] [Related]  

  • 26. A virtual screening approach to finding novel and potent antagonists at the melanin-concentrating hormone 1 receptor.
    Clark DE; Higgs C; Wren SP; Dyke HJ; Wong M; Norman D; Lockey PM; Roach AG
    J Med Chem; 2004 Jul; 47(16):3962-71. PubMed ID: 15267235
    [TBL] [Abstract][Full Text] [Related]  

  • 27. Glutamic acid analogues as potent dipeptidyl peptidase IV and 8 inhibitors.
    Lu IL; Lee SJ; Tsu H; Wu SY; Kao KH; Chien CH; Chang YY; Chen YS; Cheng JH; Chang CN; Chen TW; Chang SP; Chen X; Jiaang WT
    Bioorg Med Chem Lett; 2005 Jul; 15(13):3271-5. PubMed ID: 15927466
    [TBL] [Abstract][Full Text] [Related]  

  • 28. New amide derivatives as melanin-concentrating hormone receptor 1 antagonists for the treatment of obesity.
    Cirauqui N; Ceras J; Galiano S; Pérez-Silanes S; Juanenea L; Rivera G; Aldana I; Monge A
    Arzneimittelforschung; 2008; 58(11):585-91. PubMed ID: 19137910
    [TBL] [Abstract][Full Text] [Related]  

  • 29. Vildagliptin-Derived Dipeptidyl Peptidase 9 (DPP9) Inhibitors: Identification of a DPP8/9-Specific Lead.
    Benramdane S; De Loose J; Beyens O; Van Rymenant Y; Vliegen G; Augustyns K; De Winter H; De Meester I; Van der Veken P
    ChemMedChem; 2022 Aug; 17(15):e202200097. PubMed ID: 35760756
    [TBL] [Abstract][Full Text] [Related]  

  • 30. Dipeptidyl peptidases 8 and 9: specificity and molecular characterization compared with dipeptidyl peptidase IV.
    Bjelke JR; Christensen J; Nielsen PF; Branner S; Kanstrup AB; Wagtmann N; Rasmussen HB
    Biochem J; 2006 Jun; 396(2):391-9. PubMed ID: 16475979
    [TBL] [Abstract][Full Text] [Related]  

  • 31. Novel N-substituted 4-hydrazino piperidine derivative as a dipeptidyl peptidase IV inhibitor.
    Gupta RC; Chhipa L; Mandhare AB; Zambad SP; Chauthaiwale V; Nadkarni SS; Dutt C
    Bioorg Med Chem Lett; 2009 Sep; 19(17):5021-5. PubMed ID: 19643608
    [TBL] [Abstract][Full Text] [Related]  

  • 32. Establishment of a dipeptidyl peptidases (DPP) 8/9 expressing cell model for evaluating the selectivity of DPP4 inhibitors.
    Huan Y; Jiang Q; Liu JL; Shen ZF
    J Pharmacol Toxicol Methods; 2015; 71():8-12. PubMed ID: 25464020
    [TBL] [Abstract][Full Text] [Related]  

  • 33. Extraenzymatic functions of the dipeptidyl peptidase IV-related proteins DP8 and DP9 in cell adhesion, migration and apoptosis.
    Yu DM; Wang XM; McCaughan GW; Gorrell MD
    FEBS J; 2006 Jun; 273(11):2447-60. PubMed ID: 16704418
    [TBL] [Abstract][Full Text] [Related]  

  • 34. Expression, subcellular localisation, and possible roles of dipeptidyl peptidase 9 (DPP9) in murine macrophages.
    Zapletal E; Cupic B; Gabrilovac J
    Cell Biochem Funct; 2017 Mar; 35(2):124-137. PubMed ID: 28256001
    [TBL] [Abstract][Full Text] [Related]  

  • 35. 2-[3-[2-[(2S)-2-Cyano-1-pyrrolidinyl]-2-oxoethylamino]-3-methyl-1-oxobutyl]- 1,2,3,4-tetrahydroisoquinoline: a potent, selective, and orally bioavailable dipeptide-derived inhibitor of dipeptidyl peptidase IV.
    Tsu H; Chen X; Chen CT; Lee SJ; Chang CN; Kao KH; Coumar MS; Yeh YT; Chien CH; Wang HS; Lin KT; Chang YY; Wu SH; Chen YS; Lu IL; Wu SY; Tsai TY; Chen WC; Hsieh HP; Chao YS; Jiaang WT
    J Med Chem; 2006 Jan; 49(1):373-80. PubMed ID: 16392822
    [TBL] [Abstract][Full Text] [Related]  

  • 36. Discovery of orally efficacious melanin-concentrating hormone receptor-1 antagonists as antiobesity agents. Synthesis, SAR, and biological evaluation of bicyclo[3.1.0]hexyl ureas.
    McBriar MD; Guzik H; Shapiro S; Paruchova J; Xu R; Palani A; Clader JW; Cox K; Greenlee WJ; Hawes BE; Kowalski TJ; O'neill K; Spar BD; Weig B; Weston DJ; Farley C; Cook J
    J Med Chem; 2006 Apr; 49(7):2294-310. PubMed ID: 16570926
    [TBL] [Abstract][Full Text] [Related]  

  • 37. Outside or inside: role of the subcellular localization of DP4-like enzymes for substrate conversion and inhibitor effects.
    Bank U; Heimburg A; Wohlfarth A; Koch G; Nordhoff K; Julius H; Helmuth M; Breyer D; Reinhold D; Täger M; Ansorge S
    Biol Chem; 2011 Mar; 392(3):169-87. PubMed ID: 21194378
    [TBL] [Abstract][Full Text] [Related]  

  • 38. Discovery of imidazo[1,2-a]pyridines as potent MCH1R antagonists.
    Kishino H; Moriya M; Sakuraba S; Sakamoto T; Takahashi H; Suzuki T; Moriya R; Ito M; Iwaasa H; Takenaga N; Ishihara A; Kanatani A; Sato N; Fukami T
    Bioorg Med Chem Lett; 2009 Aug; 19(16):4589-93. PubMed ID: 19615899
    [TBL] [Abstract][Full Text] [Related]  

  • 39. A novel role of dipeptidyl peptidase 9 in epidermal growth factor signaling.
    Yao TW; Kim WS; Yu DM; Sharbeen G; McCaughan GW; Choi KY; Xia P; Gorrell MD
    Mol Cancer Res; 2011 Jul; 9(7):948-59. PubMed ID: 21622624
    [TBL] [Abstract][Full Text] [Related]  

  • 40. Method comparison of dipeptidyl peptidase IV activity assays and their application in biological samples containing reversible inhibitors.
    Matheeussen V; Lambeir AM; Jungraithmayr W; Gomez N; Mc Entee K; Van der Veken P; Scharpé S; De Meester I
    Clin Chim Acta; 2012 Feb; 413(3-4):456-62. PubMed ID: 22093941
    [TBL] [Abstract][Full Text] [Related]  

    [Previous]   [Next]    [New Search]
    of 8.