214 related articles for article (PubMed ID: 22424978)
1. Discovery of novel and potent heterocyclic carboxylic acid derivatives as protein tyrosine phosphatase 1B inhibitors.
Basu S; Prasad UV; Barawkar DA; De S; Palle VP; Menon S; Patel M; Thorat S; Singh UP; Das Sarma K; Waman Y; Niranjan S; Pathade V; Gaur A; Reddy S; Ansari S
Bioorg Med Chem Lett; 2012 Apr; 22(8):2843-9. PubMed ID: 22424978
[TBL] [Abstract][Full Text] [Related]
2. Isoxazole carboxylic acids as protein tyrosine phosphatase 1B (PTP1B) inhibitors.
Zhao H; Liu G; Xin Z; Serby MD; Pei Z; Szczepankiewicz BG; Hajduk PJ; Abad-Zapatero C; Hutchins CW; Lubben TH; Ballaron SJ; Haasch DL; Kaszubska W; Rondinone CM; Trevillyan JM; Jirousek MR
Bioorg Med Chem Lett; 2004 Nov; 14(22):5543-6. PubMed ID: 15482920
[TBL] [Abstract][Full Text] [Related]
3. Discovery of potent, selective and orally bioavailable triaryl-sulfonamide based PTP1B inhibitors.
Patel D; Jain M; Shah SR; Bahekar R; Jadav P; Joharapurkar A; Dhanesha N; Shaikh M; Sairam KV; Kapadnis P
Bioorg Med Chem Lett; 2012 Jan; 22(2):1111-7. PubMed ID: 22189136
[TBL] [Abstract][Full Text] [Related]
4. Rational design, synthesis, and structure-activity relationships of 5-amino-1H-pyrazole-4-carboxylic acid derivatives as protein tyrosine phosphatase 1B inhibitors.
Basu S; Prathipati P; Thorat S; Ansari S; Patel M; Jain V; Jinugu RR; Niranjan S; De S; Reddy S
Bioorg Med Chem; 2017 Jan; 25(1):67-74. PubMed ID: 28340988
[TBL] [Abstract][Full Text] [Related]
5. 4-Quinolone-3-carboxylic acids as cell-permeable inhibitors of protein tyrosine phosphatase 1B.
Zhi Y; Gao LX; Jin Y; Tang CL; Li JY; Li J; Long YQ
Bioorg Med Chem; 2014 Jul; 22(14):3670-83. PubMed ID: 24906513
[TBL] [Abstract][Full Text] [Related]
6. Preparation of triazole-linked glycosylated α-ketocarboxylic acid derivatives as new PTP1B inhibitors.
Song Z; He XP; Li C; Gao LX; Wang ZX; Tang Y; Xie J; Li J; Chen GR
Carbohydr Res; 2011 Jan; 346(1):140-5. PubMed ID: 21111404
[TBL] [Abstract][Full Text] [Related]
7. Synthesis and biological evaluation of heterocyclic ring-substituted maslinic acid derivatives as novel inhibitors of protein tyrosine phosphatase 1B.
Qiu WW; Shen Q; Yang F; Wang B; Zou H; Li JY; Li J; Tang J
Bioorg Med Chem Lett; 2009 Dec; 19(23):6618-22. PubMed ID: 19846303
[TBL] [Abstract][Full Text] [Related]
8. 7-Phenyl-pyrido[2,3-d]pyrimidine-2,4-diamines: novel and highly selective protein tyrosine phosphatase 1B inhibitors.
Cheung AW; Banner B; Bose J; Kim K; Li S; Marcopulos N; Orzechowski L; Sergi JA; Thakkar KC; Wang BB; Yun W; Zwingelstein C; Berthel S; Olivier AR
Bioorg Med Chem Lett; 2012 Dec; 22(24):7518-22. PubMed ID: 23122867
[TBL] [Abstract][Full Text] [Related]
9. Bromophenols as inhibitors of protein tyrosine phosphatase 1B with antidiabetic properties.
Shi D; Li J; Jiang B; Guo S; Su H; Wang T
Bioorg Med Chem Lett; 2012 Apr; 22(8):2827-32. PubMed ID: 22444684
[TBL] [Abstract][Full Text] [Related]
10. Identification of 2-substituted ethenesulfonic acid ester derivatives as novel, potent and selective inhibitors of protein tyrosine phosphatase 1B.
Deng X; Liu J; Jin Y; Zhang Y; He W; Bao J; Liu W; Jiang F; Fu L
Pharmazie; 2015 Dec; 70(12):777-83. PubMed ID: 26817274
[TBL] [Abstract][Full Text] [Related]
11. Discovery of orally active, potent, and selective benzotriazole-based PTP1B inhibitors.
Patel D; Jain M; Shah SR; Bahekar R; Jadav P; Darji B; Siriki Y; Bandyopadhyay D; Joharapurkar A; Kshirsagar S; Patel H; Shaikh M; Sairam KV; Patel P
ChemMedChem; 2011 Jun; 6(6):1011-6. PubMed ID: 21506278
[No Abstract] [Full Text] [Related]
12. Investigations of linker structure on the potency of a series of bidentate protein tyrosine phosphatase inhibitors.
Xie J; Seto CT
Bioorg Med Chem; 2005 Apr; 13(8):2981-91. PubMed ID: 15781408
[TBL] [Abstract][Full Text] [Related]
13. Novel thiophene derivatives as PTP1B inhibitors with selectivity and cellular activity.
Ye D; Zhang Y; Wang F; Zheng M; Zhang X; Luo X; Shen X; Jiang H; Liu H
Bioorg Med Chem; 2010 Mar; 18(5):1773-82. PubMed ID: 20153651
[TBL] [Abstract][Full Text] [Related]
14. Selective protein tyrosine phosphatase 1B inhibitors: targeting the second phosphotyrosine binding site with non-carboxylic acid-containing ligands.
Liu G; Xin Z; Liang H; Abad-Zapatero C; Hajduk PJ; Janowick DA; Szczepankiewicz BG; Pei Z; Hutchins CW; Ballaron SJ; Stashko MA; Lubben TH; Berg CE; Rondinone CM; Trevillyan JM; Jirousek MR
J Med Chem; 2003 Jul; 46(16):3437-40. PubMed ID: 12877578
[TBL] [Abstract][Full Text] [Related]
15. Discovery of di-indolinone as a novel scaffold for protein tyrosine phosphatase 1B inhibitors.
Dai HL; Gao LX; Yang Y; Li JY; Cheng JG; Li J; Wen R; Peng YQ; Zheng JB
Bioorg Med Chem Lett; 2012 Dec; 22(24):7440-3. PubMed ID: 23122522
[TBL] [Abstract][Full Text] [Related]
16. Synthesis and evaluation of some novel dibenzo[b,d]furan carboxylic acids as potential anti-diabetic agents.
Lakshminarayana N; Prasad YR; Gharat L; Thomas A; Narayanan S; Raghuram A; Srinivasan CV; Gopalan B
Eur J Med Chem; 2010 Sep; 45(9):3709-18. PubMed ID: 20627471
[TBL] [Abstract][Full Text] [Related]
17. Pyrrolo[2,3-c]azepine derivatives: a new class of potent protein tyrosine phosphatase 1B inhibitors.
Xie J; Tian J; Su L; Huang M; Zhu X; Ye F; Wan Y
Bioorg Med Chem Lett; 2011 Jul; 21(14):4306-9. PubMed ID: 21696953
[TBL] [Abstract][Full Text] [Related]
18. Structure-based optimization of benzoic acids as inhibitors of protein tyrosine phosphatase 1B and low molecular weight protein tyrosine phosphatase.
Maccari R; Ottanà R; Ciurleo R; Paoli P; Manao G; Camici G; Laggner C; Langer T
ChemMedChem; 2009 Jun; 4(6):957-62. PubMed ID: 19288492
[TBL] [Abstract][Full Text] [Related]
19. Synthesis and biological evaluation of 2,4,6-trihydroxychalcone derivatives as novel protein tyrosine phosphatase 1B inhibitors.
Sun LP; Gao LX; Ma WP; Nan FJ; Li J; Piao HR
Chem Biol Drug Des; 2012 Oct; 80(4):584-90. PubMed ID: 22805439
[TBL] [Abstract][Full Text] [Related]
20. Potent inhibition of protein tyrosine phosphatases by copper complexes with multi-benzimidazole derivatives.
Li Y; Lu L; Zhu M; Wang Q; Yuan C; Xing S; Fu X; Mei Y
Biometals; 2011 Dec; 24(6):993-1004. PubMed ID: 21618062
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]
