152 related articles for article (PubMed ID: 22530893)
1. Biological and anti-inflammatory evaluation of two thiazole compounds in RAW cell line: potential cyclooxygenase-2 specific inhibitors.
Hamade E; Habib A; Hachem A; Hussein AH; Abbas M; Hirz T; Al Masri M; Faour WH
Med Chem; 2012 May; 8(3):401-8. PubMed ID: 22530893
[TBL] [Abstract][Full Text] [Related]
2. Design, synthesis and molecular docking of novel D-ring substituted steroidal 4,5-dihydropyrazole thiazole derivatives that act as iNOS/COX-2 inhibitors with potent anti-inflammatory activity against LPS-induced RAW264.7 macrophage cells.
Fang S; Huang X; Cai F; Qiu G; Lin F; Cai X
J Steroid Biochem Mol Biol; 2024 Jun; 240():106478. PubMed ID: 38430971
[TBL] [Abstract][Full Text] [Related]
3. Synthesis of New Tricyclic and Tetracyclic Fused Coumarin Sulfonate Derivatives and Their Inhibitory Effects on LPS-Induced Nitric Oxide and PGE
El-Gamal MI; Lee WS; Shin JS; Oh CH; Lee KT; Choi J; Myoung N; Baek D
Arch Pharm (Weinheim); 2016 Nov; 349(11):853-863. PubMed ID: 27779319
[TBL] [Abstract][Full Text] [Related]
4. Synthesis, pharmacological evaluation and docking studies of N-(benzo[d]thiazol-2-yl)-2-(piperazin-1-yl)acetamide analogs as COX-2 inhibitors.
Raghavendra NM; Jyothsna A; Venkateswara Rao A; Subrahmanyam CV
Bioorg Med Chem Lett; 2012 Jan; 22(2):820-3. PubMed ID: 22222039
[TBL] [Abstract][Full Text] [Related]
5. New methyl 5-(halomethyl)-1-aryl-1H-1,2,4-triazole-3-carboxylates as selective COX-2 inhibitors and anti-inflammatory agents: Design, synthesis, biological evaluation, and docking study.
Li SM; Tsai SE; Chiang CY; Chung CY; Chuang TJ; Tseng CC; Jiang WP; Huang GJ; Lin CY; Yang YC; Fuh MT; Wong FF
Bioorg Chem; 2020 Nov; 104():104333. PubMed ID: 33142408
[TBL] [Abstract][Full Text] [Related]
6. Identification and development of thiazole leads as COX-2/5-LOX inhibitors through in-vitro and in-vivo biological evaluation for anti-inflammatory activity.
Jacob P J; Manju SL
Bioorg Chem; 2020 Jul; 100():103882. PubMed ID: 32361295
[TBL] [Abstract][Full Text] [Related]
7. Design, synthesis, anti-inflammatory activity, and molecular docking studies of perimidine derivatives containing triazole.
Zhang HJ; Wang XZ; Cao Q; Gong GH; Quan ZS
Bioorg Med Chem Lett; 2017 Sep; 27(18):4409-4414. PubMed ID: 28823493
[TBL] [Abstract][Full Text] [Related]
8. Design, synthesis and biological assessment of new selective COX-2 inhibitors including methyl sulfonyl moiety.
Sağlık BN; Osmaniye D; Levent S; Çevik UA; Çavuşoğlu BK; Özkay Y; Kaplancıklı ZA
Eur J Med Chem; 2021 Jan; 209():112918. PubMed ID: 33071054
[TBL] [Abstract][Full Text] [Related]
9. Selective cyclooxygenase inhibition and ulcerogenic liability of some newly prepared anti-inflammatory agents having thiazolo[4,5-d]pyrimidine scaffold.
Bakr RB; Ghoneim AA; Azouz AA
Bioorg Chem; 2019 Jul; 88():102964. PubMed ID: 31075742
[TBL] [Abstract][Full Text] [Related]
10. Stomopneulactone D from long-spined sea urchin Stomopneustes variolaris: Anti-inflammatory macrocylic lactone attenuates cyclooxygenase-2 expression in lipopolysaccharide-activated macrophages.
Chakraborty K; Francis P
Bioorg Chem; 2020 Oct; 103():104140. PubMed ID: 32763520
[TBL] [Abstract][Full Text] [Related]
11. Thiazole derivatives as inhibitors of cyclooxygenases in vitro and in vivo.
El-Achkar GA; Jouni M; Mrad MF; Hirz T; El Hachem N; Khalaf A; Hammoud S; Fayyad-Kazan H; Eid AA; Badran B; Merhi RA; Hachem A; Hamade E; Habib A
Eur J Pharmacol; 2015 Mar; 750():66-73. PubMed ID: 25617797
[TBL] [Abstract][Full Text] [Related]
12. Design of balanced COX inhibitors based on anti-inflammatory and/or COX-2 inhibitory ascidian metabolites.
Ju Z; Su M; Hong J; La Kim E; Moon HR; Chung HY; Kim S; Jung JH
Eur J Med Chem; 2019 Oct; 180():86-98. PubMed ID: 31301566
[TBL] [Abstract][Full Text] [Related]
13. Synthesis and discovery of pyrazolo-pyridine analogs as inflammation medications through pro- and anti-inflammatory cytokine and COX-2 inhibition assessments.
Dennis Bilavendran J; Manikandan A; Thangarasu P; Sivakumar K
Bioorg Chem; 2020 Jan; 94():103484. PubMed ID: 31796215
[TBL] [Abstract][Full Text] [Related]
14. Design, synthesis, and SAR study of novel 4,5-dihydropyrazole-Thiazole derivatives with anti-inflammatory activities for the treatment of sepsis.
Zhang Z; Cao P; Fang M; Zou T; Han J; Duan Y; Xu H; Yang X; Li QS
Eur J Med Chem; 2021 Dec; 225():113743. PubMed ID: 34403978
[TBL] [Abstract][Full Text] [Related]
15. Design, synthesis and bioactivity study of N-salicyloyl tryptamine derivatives as multifunctional agents for the treatment of neuroinflammation.
Fan X; Li J; Deng X; Lu Y; Feng Y; Ma S; Wen H; Zhao Q; Tan W; Shi T; Wang Z
Eur J Med Chem; 2020 May; 193():112217. PubMed ID: 32182488
[TBL] [Abstract][Full Text] [Related]
16. Discovery of a novel COX-2 inhibitor as an orally potent anti-pyretic and anti-inflammatory drug: design, synthesis, and structure-activity relationship.
Hayashi S; Sumi Y; Ueno N; Murase A; Takada J
Biochem Pharmacol; 2011 Oct; 82(7):755-68. PubMed ID: 21741371
[TBL] [Abstract][Full Text] [Related]
17. Anti-inflammatory activity of compounds from the rhizome of Cnidium officinale.
Tran HNK; Cao TQ; Kim JA; Youn UJ; Kim S; Woo MH; Min BS
Arch Pharm Res; 2018 Oct; 41(10):977-985. PubMed ID: 29961195
[TBL] [Abstract][Full Text] [Related]
18. Protective effect of pine (Pinus morrisonicola Hay.) needle on LDL oxidation and its anti-inflammatory action by modulation of iNOS and COX-2 expression in LPS-stimulated RAW 264.7 macrophages.
Yen GC; Duh PD; Huang DW; Hsu CL; Fu TY
Food Chem Toxicol; 2008 Jan; 46(1):175-85. PubMed ID: 17804140
[TBL] [Abstract][Full Text] [Related]
19. Design, synthesis and analgesic/anti-inflammatory evaluation of novel diarylthiazole and diarylimidazole derivatives towards selective COX-1 inhibitors with better gastric profile.
Abdelazeem AH; El-Saadi MT; Safi El-Din AG; Omar HA; El-Moghazy SM
Bioorg Med Chem; 2017 Jan; 25(2):665-676. PubMed ID: 27916468
[TBL] [Abstract][Full Text] [Related]
20. Synthesis of unsymmetrical monocarbonyl curcumin analogues with potent inhibition on prostaglandin E2 production in LPS-induced murine and human macrophages cell lines.
Mohd Aluwi MFF; Rullah K; Yamin BM; Leong SW; Abdul Bahari MN; Lim SJ; Mohd Faudzi SM; Jalil J; Abas F; Mohd Fauzi N; Ismail NH; Jantan I; Lam KW
Bioorg Med Chem Lett; 2016 May; 26(10):2531-2538. PubMed ID: 27040659
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]