These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.


BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

133 related articles for article (PubMed ID: 22542502)

  • 1. Synthesis of 2-[11C]methoxy-3,17β-O,O-bis(sulfamoyl)estradiol as a new potential PET agent for imaging of steroid sulfatase (STS) in cancers.
    Wang M; Xu L; Gao M; Miller KD; Sledge GW; Zheng QH
    Steroids; 2012 Jul; 77(8-9):864-70. PubMed ID: 22542502
    [TBL] [Abstract][Full Text] [Related]  

  • 2. 2-substituted estradiol bis-sulfamates, multitargeted antitumor agents: synthesis, in vitro SAR, protein crystallography, and in vivo activity.
    Leese MP; Leblond B; Smith A; Newman SP; Di Fiore A; De Simone G; Supuran CT; Purohit A; Reed MJ; Potter BV
    J Med Chem; 2006 Dec; 49(26):7683-96. PubMed ID: 17181151
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Design and synthesis of carbon-11-labeled dual aromatase-steroid sulfatase inhibitors as new potential PET agents for imaging of aromatase and steroid sulfatase expression in breast cancer.
    Wang M; Mickens J; Gao M; Miller KD; Sledge GW; Hutchins GD; Zheng QH
    Steroids; 2009 Nov; 74(12):896-905. PubMed ID: 19559719
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Simple synthesis of carbon-11-labeled chromen-4-one derivatives as new potential PET agents for imaging of DNA-dependent protein kinase (DNA-PK) in cancer.
    Gao M; Wang M; Miller KD; Zheng QH
    Appl Radiat Isot; 2012 Aug; 70(8):1558-63. PubMed ID: 22732390
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Solid-phase parallel synthesis of 17alpha-substituted estradiol sulfamate and phenol libraries using the multidetachable sulfamate linker.
    Ciobanu LC; Poirier D
    J Comb Chem; 2003; 5(4):429-40. PubMed ID: 12857111
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Steroidal and nonsteroidal sulfamates as potent inhibitors of steroid sulfatase.
    Woo LW; Howarth NM; Purohit A; Hejaz HA; Reed MJ; Potter BV
    J Med Chem; 1998 Mar; 41(7):1068-83. PubMed ID: 9544207
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Synthesis of new carbon-11 labeled naphthalene-sulfonamides for PET imaging of human CCR8.
    Wang M; Cooley B; Gao M; Miller KD; Sledge GW; Hutchins GD; Zheng QH
    Appl Radiat Isot; 2008 Oct; 66(10):1406-13. PubMed ID: 18455923
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Facile synthesis of carbon-11-labeled cholesterol-based cationic lipids as new potential PET probes for imaging of gene delivery in cancer.
    Gao M; Wang M; Miller KD; Sledge GW; Hutchins GD; Zheng QH
    Steroids; 2010 Oct; 75(10):715-20. PubMed ID: 20451540
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Simple synthesis of carbon-11 labeled styryl dyes as new potential PET RNA-specific, living cell imaging probes.
    Wang M; Gao M; Miller KD; Sledge GW; Hutchins GD; Zheng QH
    Eur J Med Chem; 2009 May; 44(5):2300-6. PubMed ID: 18396357
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Highly potent first examples of dual aromatase-steroid sulfatase inhibitors based on a biphenyl template.
    Woo LW; Jackson T; Putey A; Cozier G; Leonard P; Acharya KR; Chander SK; Purohit A; Reed MJ; Potter BV
    J Med Chem; 2010 Mar; 53(5):2155-70. PubMed ID: 20148564
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Synthesis of 2,6-difluoro-N-(3-[11C]methoxy-1H-pyrazolo[3,4-b]pyridine-5-yl)-3-(propylsulfonamidio)benzamide as a new potential PET agent for imaging of B-Raf(V600E) in cancers.
    Wang M; Gao M; Miller KD; Zheng QH
    Bioorg Med Chem Lett; 2013 Feb; 23(4):1017-21. PubMed ID: 23294704
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Synthesis of new carbon-11 labeled benzoxazole derivatives for PET imaging of 5-HT(3) receptor.
    Gao M; Wang M; Hutchins GD; Zheng QH
    Eur J Med Chem; 2008 Jul; 43(7):1570-4. PubMed ID: 18045745
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Synthesis of [¹¹C]PBR06 and [¹⁸F]PBR06 as agents for positron emission tomographic (PET) imaging of the translocator protein (TSPO).
    Wang M; Gao M; Miller KD; Zheng QH
    Steroids; 2011 Nov; 76(12):1331-40. PubMed ID: 21756927
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Inhibition of estrone sulfate-induced uterine growth by potent nonestrogenic steroidal inhibitors of steroid sulfatase.
    Ciobanu LC; Luu-The V; Martel C; Labrie F; Poirier D
    Cancer Res; 2003 Oct; 63(19):6442-6. PubMed ID: 14559834
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Facile and high-yield synthesis of N-(4-diethylamino)benzyl-4-[¹¹C]methoxy-N-(p-tolyl)benzenesulfonamide as a new potential PET selective CB2 radioligand.
    Gao M; Xu J; Wang M; Zheng QH
    Appl Radiat Isot; 2014 Aug; 90():181-6. PubMed ID: 24768996
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Inhibition of steroid sulfatase with 4-substituted estrone and estradiol derivatives.
    Phan CM; Liu Y; Kim BM; Mostafa Y; Taylor SD
    Bioorg Med Chem; 2011 Oct; 19(20):5999-6005. PubMed ID: 21925885
    [TBL] [Abstract][Full Text] [Related]  

  • 17. 3,17-disubstituted 2-alkylestra-1,3,5(10)-trien-3-ol derivatives: synthesis, in vitro and in vivo anticancer activity.
    Bubert C; Leese MP; Mahon MF; Ferrandis E; Regis-Lydi S; Kasprzyk PG; Newman SP; Ho YT; Purohit A; Reed MJ; Potter BV
    J Med Chem; 2007 Sep; 50(18):4431-43. PubMed ID: 17696419
    [TBL] [Abstract][Full Text] [Related]  

  • 18. The first synthesis of [11C]J147, a new potential PET agent for imaging of Alzheimer's disease.
    Wang M; Gao M; Zheng QH
    Bioorg Med Chem Lett; 2013 Jan; 23(2):524-7. PubMed ID: 23237833
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Synthesis of aromatase inhibitors and dual aromatase steroid sulfatase inhibitors by linking an arylsulfamate motif to 4-(4H-1,2,4-triazol-4-ylamino)benzonitrile: SAR, crystal structures, in vitro and in vivo activities.
    Bubert C; Woo LW; Sutcliffe OB; Mahon MF; Chander SK; Purohit A; Reed MJ; Potter BV
    ChemMedChem; 2008 Nov; 3(11):1708-30. PubMed ID: 18816537
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Synthesis and biological activity of the superestrogen (E)-17-oximino-3-O-sulfamoyl-1,3,5(10)-estratriene: x-ray crystal structure of (E)-17-oximino-3-hydroxy-1,3,5(10)-estratriene.
    Hejaz HA; Purohit A; Mahon MF; Reed MJ; Potter BV
    J Med Chem; 1999 Aug; 42(16):3188-92. PubMed ID: 10447965
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 7.