These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.
200 related articles for article (PubMed ID: 22608920)
1. Synthesis and evaluation of 11β-(4-substituted phenyl) estradiol analogs: transition from estrogen receptor agonists to antagonists. Hanson RN; Hua E; Hendricks JA; Labaree D; Hochberg RB Bioorg Med Chem; 2012 Jun; 20(12):3768-80. PubMed ID: 22608920 [TBL] [Abstract][Full Text] [Related]
2. Synthesis and biochemical characterization of a series of 17α-perfluoroalkylated estradiols as selective ligands for estrogen receptor α. Eignerová B; Sedlák D; Dracínský M; Bartunek P; Kotora M J Med Chem; 2010 Oct; 53(19):6947-53. PubMed ID: 20812681 [TBL] [Abstract][Full Text] [Related]
3. The terminal substituents of 7α, 6-hexanyl derivatives of estradiol determine their selective estrogen receptor modulator versus agonist activities. Hoffman KL; Foster EA; Smith CL Steroids; 2012 Apr; 77(5):496-503. PubMed ID: 22326682 [TBL] [Abstract][Full Text] [Related]
4. Steroidal affinity labels of the estrogen receptor alpha. 4. Electrophilic 11beta-aryl derivatives of estradiol. Aliau S; Delettre G; Mattras H; El Garrouj D; Nique F; Teutsch G; Borgna JL J Med Chem; 2000 Feb; 43(4):613-28. PubMed ID: 10691688 [TBL] [Abstract][Full Text] [Related]
5. Cysteine 530 of the human estrogen receptor alpha is the main covalent attachment site of 11beta-(aziridinylalkoxyphenyl)estradiols. Aliau S; Mattras H; Richard E; Borgna JL Biochemistry; 1999 Nov; 38(45):14752-62. PubMed ID: 10555957 [TBL] [Abstract][Full Text] [Related]
6. Synthesis and evaluation of 17α-E-20-(heteroaryl)norpregn-1,3,5(10),20 tetraene-3,17β-diols [17α-(heteroaryl)vinyl estradiols] as ligands for the estrogen receptor-α ligand binding domain (ERα-LBD). Olmsted SL; Tongcharoensirikul P; McCaskill E; Gandiaga K; Labaree D; Hochberg RB; Hanson RN Bioorg Med Chem Lett; 2012 Jan; 22(2):977-9. PubMed ID: 22178552 [TBL] [Abstract][Full Text] [Related]
7. Nonpolar and short side chain groups at C-11beta of estradiol result in antiestrogens. Zhang JX; Labaree DC; Hochberg RB J Med Chem; 2005 Mar; 48(5):1428-47. PubMed ID: 15743187 [TBL] [Abstract][Full Text] [Related]
8. Synthesis, binding affinity, and transcriptional activity of hydroxy- and methoxy-substituted 3,4-diarylsalicylaldoximes on estrogen receptors alpha and beta. Minutolo F; Antonello M; Bertini S; Rapposelli S; Rossello A; Sheng S; Carlson KE; Katzenellenbogen JA; Macchia M Bioorg Med Chem; 2003 Apr; 11(7):1247-57. PubMed ID: 12628652 [TBL] [Abstract][Full Text] [Related]
9. Synthesis and evaluation of 17α-(dimethylphenyl)vinyl estradiols as probes of the estrogen receptor-α ligand binding domain. Hanson RN; McCaskill E; Tongcharoensirikul P; Dilis R; Labaree D; Hochberg RB Steroids; 2012 Apr; 77(5):471-6. PubMed ID: 22273809 [TBL] [Abstract][Full Text] [Related]
10. Synthesis and evaluation of 11beta-substituted 21-chloro/iodo-(17alpha,20E/Z)-19-norpregna-1,3,5(10),20-te traene-3, 17beta-diols: high-affinity ligands for the estrogen receptor. Hanson RN; Napolitano E; Fiaschi R J Med Chem; 1998 Nov; 41(24):4686-92. PubMed ID: 9822539 [TBL] [Abstract][Full Text] [Related]
14. Synthesis and evaluation of 17α-triazolyl and 9α-cyano derivatives of estradiol. Wetzel EA; Hanson AM; Troutfetter CL; Burkett DJ; Sem DS; Donaldson WA Bioorg Med Chem; 2020 Oct; 28(19):115670. PubMed ID: 32912438 [TBL] [Abstract][Full Text] [Related]
15. Synthesis of benzoylbenzamide derivatives of 17α-E-vinyl estradiol and evaluation as ligands for the estrogen receptor-α ligand binding domain. Hanson RN; McCaskill E; Hua E; Tongcharoensirikul P; Dilis R; Silver JL; Coulther TA; Ondrechen MJ; Labaree D; Hochberg RB Steroids; 2019 Apr; 144():15-20. PubMed ID: 30738075 [TBL] [Abstract][Full Text] [Related]
16. Functional characterization of estrogen receptor subtypes, ERalpha and ERbeta, mediating vitellogenin production in the liver of rainbow trout. Leaños-Castañeda O; Van Der Kraak G Toxicol Appl Pharmacol; 2007 Oct; 224(2):116-25. PubMed ID: 17662327 [TBL] [Abstract][Full Text] [Related]
17. Estrogen to antiestrogen with a single methylene group resulting in an unusual steroidal selective estrogen receptor modulator. Zhang JX; Labaree DC; Mor G; Hochberg RB J Clin Endocrinol Metab; 2004 Jul; 89(7):3527-35. PubMed ID: 15240642 [TBL] [Abstract][Full Text] [Related]
18. Synthesis and evaluation of B-, C-, and D-ring-substituted estradiol carboxylic acid esters as locally active estrogens. Labaree DC; Zhang JX; Harris HA; O'Connor C; Reynolds TY; Hochberg RB J Med Chem; 2003 May; 46(10):1886-904. PubMed ID: 12723952 [TBL] [Abstract][Full Text] [Related]
19. Differential response of estrogen receptor alpha and estrogen receptor beta to partial estrogen agonists/antagonists. Barkhem T; Carlsson B; Nilsson Y; Enmark E; Gustafsson J; Nilsson S Mol Pharmacol; 1998 Jul; 54(1):105-12. PubMed ID: 9658195 [TBL] [Abstract][Full Text] [Related]