294 related articles for article (PubMed ID: 22649514)
1. Antimalarial activity and mechanisms of action of two novel 4-aminoquinolines against chloroquine-resistant parasites.
Aguiar AC; Santos Rde M; Figueiredo FJ; Cortopassi WA; Pimentel AS; França TC; Meneghetti MR; Krettli AU
PLoS One; 2012; 7(5):e37259. PubMed ID: 22649514
[TBL] [Abstract][Full Text] [Related]
2. 4-Aminoquinoline derivatives: Synthesis, in vitro and in vivo antiplasmodial activity against chloroquine-resistant parasites.
Singh S; Agarwal D; Sharma K; Sharma M; Nielsen MA; Alifrangis M; Singh AK; Gupta RD; Awasthi SK
Eur J Med Chem; 2016 Oct; 122():394-407. PubMed ID: 27394399
[TBL] [Abstract][Full Text] [Related]
3. Antiplasmodial activity of chloroquine analogs against chloroquine-resistant parasites, docking studies and mechanisms of drug action.
de Souza NB; Carmo AM; da Silva AD; França TC; Krettli AU
Malar J; 2014 Dec; 13():469. PubMed ID: 25440372
[TBL] [Abstract][Full Text] [Related]
4. Novel 4-aminoquinoline analogs highly active against the blood and sexual stages of Plasmodium in vivo and in vitro.
Sáenz FE; Mutka T; Udenze K; Oduola AM; Kyle DE
Antimicrob Agents Chemother; 2012 Sep; 56(9):4685-92. PubMed ID: 22710117
[TBL] [Abstract][Full Text] [Related]
5. Examination of the antimalarial potential of experimental aminoquinolines: poor in vitro effect does not preclude in vivo efficacy.
Srbljanović J; Štajner T; Konstantinović J; Terzić-Jovanović N; Uzelac A; Bobić B; Šolaja BA; Djurković-Djaković O
Int J Antimicrob Agents; 2017 Sep; 50(3):461-466. PubMed ID: 28668677
[TBL] [Abstract][Full Text] [Related]
6. Activity of piperaquine and other 4-aminoquinoline antiplasmodial drugs against chloroquine-sensitive and resistant blood-stages of Plasmodium falciparum. Role of beta-haematin inhibition and drug concentration in vacuolar water- and lipid-phases.
Warhurst DC; Craig JC; Adagu IS; Guy RK; Madrid PB; Fivelman QL
Biochem Pharmacol; 2007 Jun; 73(12):1910-26. PubMed ID: 17466277
[TBL] [Abstract][Full Text] [Related]
7. Antimalarial activity of potential inhibitors of Plasmodium falciparum lactate dehydrogenase enzyme selected by docking studies.
Penna-Coutinho J; Cortopassi WA; Oliveira AA; França TC; Krettli AU
PLoS One; 2011; 6(7):e21237. PubMed ID: 21779323
[TBL] [Abstract][Full Text] [Related]
8. Antiplasmodial activity of new 4-aminoquinoline derivatives against chloroquine resistant strain.
Sinha M; Dola VR; Agarwal P; Srivastava K; Haq W; Puri SK; Katti SB
Bioorg Med Chem; 2014 Jul; 22(14):3573-86. PubMed ID: 24906512
[TBL] [Abstract][Full Text] [Related]
9. Synergistic interaction of a chloroquine metabolite with chloroquine against drug-resistant malaria parasites.
Kalkanidis M; Klonis N; Tschan S; Deady LW; Tilley L
Biochem Pharmacol; 2004 Apr; 67(7):1347-53. PubMed ID: 15013850
[TBL] [Abstract][Full Text] [Related]
10. 4-Aminoquinoline quinolizidinyl- and quinolizidinylalkyl-derivatives with antimalarial activity.
Sparatore A; Basilico N; Parapini S; Romeo S; Novelli F; Sparatore F; Taramelli D
Bioorg Med Chem; 2005 Sep; 13(18):5338-45. PubMed ID: 16054368
[TBL] [Abstract][Full Text] [Related]
11. Enhanced antimalarial effects of chloroquine by aqueous Vernonia amygdalina leaf extract in mice infected with chloroquine resistant and sensitive Plasmodium berghei strains.
Iwalokun BA
Afr Health Sci; 2008 Mar; 8(1):25-35. PubMed ID: 19357729
[TBL] [Abstract][Full Text] [Related]
12. 4-Aminoquinoline Antimalarials Containing a Benzylmethylpyridylmethylamine Group Are Active against Drug Resistant Plasmodium falciparum and Exhibit Oral Activity in Mice.
Joshi MC; Okombo J; Nsumiwa S; Ndove J; Taylor D; Wiesner L; Hunter R; Chibale K; Egan TJ
J Med Chem; 2017 Dec; 60(24):10245-10256. PubMed ID: 29185748
[TBL] [Abstract][Full Text] [Related]
13. Docking, synthesis and antimalarial activity of novel 4-anilinoquinoline derivatives.
Vijayaraghavan S; Mahajan S
Bioorg Med Chem Lett; 2017 Apr; 27(8):1693-1697. PubMed ID: 28318947
[TBL] [Abstract][Full Text] [Related]
14. 3-Iodo-4-aminoquinoline derivative sensitises resistant strains of Plasmodium falciparum to chloroquine.
Edaye S; Tazoo D; Bohle DS; Georges E
Int J Antimicrob Agents; 2016 Jun; 47(6):482-5. PubMed ID: 27211211
[TBL] [Abstract][Full Text] [Related]
15. Design, Synthesis, and Evaluation of Novel Ferroquine and Phenylequine Analogues as Potential Antiplasmodial Agents.
Jacobs L; de Kock C; de Villiers KA; Smith PJ; Smith VJ; van Otterlo WA; Blackie MA
ChemMedChem; 2015 Dec; 10(12):2099-110. PubMed ID: 26447782
[TBL] [Abstract][Full Text] [Related]
16. Antimalarial activity of novel pyrrolizidinyl derivatives of 4-aminoquinoline.
Sparatore A; Basilico N; Casagrande M; Parapini S; Taramelli D; Brun R; Wittlin S; Sparatore F
Bioorg Med Chem Lett; 2008 Jul; 18(13):3737-40. PubMed ID: 18538567
[TBL] [Abstract][Full Text] [Related]
17. Antimalarial benzoheterocyclic 4-aminoquinolines: Structure-activity relationship, in vivo evaluation, mechanistic and bioactivation studies.
Ongarora DS; Strydom N; Wicht K; Njoroge M; Wiesner L; Egan TJ; Wittlin S; Jurva U; Masimirembwa CM; Chibale K
Bioorg Med Chem; 2015 Sep; 23(17):5419-32. PubMed ID: 26264839
[TBL] [Abstract][Full Text] [Related]
18. Quantitative characterization of hemozoin in Plasmodium berghei and vivax.
Pisciotta JM; Scholl PF; Shuman JL; Shualev V; Sullivan DJ
Int J Parasitol Drugs Drug Resist; 2017 Apr; 7(1):110-119. PubMed ID: 28279945
[TBL] [Abstract][Full Text] [Related]
19. Antimalarials with Benzothiophene Moieties as Aminoquinoline Partners.
Konstantinović J; Videnović M; Srbljanović J; Djurković-Djaković O; Bogojević K; Sciotti R; Šolaja B
Molecules; 2017 Feb; 22(3):. PubMed ID: 28245583
[TBL] [Abstract][Full Text] [Related]
20. In vitro synergistic interaction of potent 4-aminoquinolines in combination with dihydroartemisinin against chloroquine-resistant Plasmodium falciparum.
Agarwal D; Singh S; Gupta RD; Awasthi SK
Acta Trop; 2019 Nov; 199():105109. PubMed ID: 31351071
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]