138 related articles for article (PubMed ID: 22731815)
1. Virtual screening identifies novel sulfonamide inhibitors of ecto-5'-nucleotidase.
Ripphausen P; Freundlieb M; Brunschweiger A; Zimmermann H; Müller CE; Bajorath J
J Med Chem; 2012 Jul; 55(14):6576-81. PubMed ID: 22731815
[TBL] [Abstract][Full Text] [Related]
2. Virtual Screening Approach for the Identification of Hydroxamic Acids as Novel Human Ecto-5'-Nucleotidase Inhibitors.
Viviani LG; Piccirillo E; Ulrich H; Amaral AT
J Chem Inf Model; 2020 Feb; 60(2):621-630. PubMed ID: 31714079
[TBL] [Abstract][Full Text] [Related]
3. Evaluation of molecular model-based discovery of ecto-5'-nucleotidase inhibitors on the basis of X-ray structures.
Furtmann N; Bajorath J
Bioorg Med Chem; 2013 Nov; 21(21):6616-22. PubMed ID: 24012379
[TBL] [Abstract][Full Text] [Related]
4. Development of potent and selective inhibitors of ecto-5'-nucleotidase based on an anthraquinone scaffold.
Baqi Y; Lee SY; Iqbal J; Ripphausen P; Lehr A; Scheiff AB; Zimmermann H; Bajorath J; Müller CE
J Med Chem; 2010 Mar; 53(5):2076-86. PubMed ID: 20146483
[TBL] [Abstract][Full Text] [Related]
5. Identification of sulfonic acids as efficient ecto-5'-nucleotidase inhibitors.
Iqbal J; Saeed A; Raza R; Matin A; Hameed A; Furtmann N; Lecka J; Sévigny J; Bajorath J
Eur J Med Chem; 2013; 70():685-91. PubMed ID: 24215819
[TBL] [Abstract][Full Text] [Related]
6. Identification and characterization of inhibitors of cytoplasmic 5'-nucleotidase cN-II issued from virtual screening.
Jordheim LP; Marton Z; Rhimi M; Cros-Perrial E; Lionne C; Peyrottes S; Dumontet C; Aghajari N; Chaloin L
Biochem Pharmacol; 2013 Feb; 85(4):497-506. PubMed ID: 23220537
[TBL] [Abstract][Full Text] [Related]
7. 2-Substituted α,β-Methylene-ADP Derivatives: Potent Competitive Ecto-5'-nucleotidase (CD73) Inhibitors with Variable Binding Modes.
Bhattarai S; Pippel J; Scaletti E; Idris R; Freundlieb M; Rolshoven G; Renn C; Lee SY; Abdelrahman A; Zimmermann H; El-Tayeb A; Müller CE; Sträter N
J Med Chem; 2020 Mar; 63(6):2941-2957. PubMed ID: 32045236
[TBL] [Abstract][Full Text] [Related]
8. Pursuing aldose reductase inhibitors through in situ cross-docking and similarity-based virtual screening.
Cosconati S; Marinelli L; La Motta C; Sartini S; Da Settimo F; Olson AJ; Novellino E
J Med Chem; 2009 Sep; 52(18):5578-81. PubMed ID: 19719141
[TBL] [Abstract][Full Text] [Related]
9. Therapeutic potentials of ecto-nucleoside triphosphate diphosphohydrolase, ecto-nucleotide pyrophosphatase/phosphodiesterase, ecto-5'-nucleotidase, and alkaline phosphatase inhibitors.
al-Rashida M; Iqbal J
Med Res Rev; 2014 Jul; 34(4):703-43. PubMed ID: 24115166
[TBL] [Abstract][Full Text] [Related]
10. 4-Aminopyridine based amide derivatives as dual inhibitors of tissue non-specific alkaline phosphatase and ecto-5'-nucleotidase with potential anticancer activity.
Hassan S; Ejaz SA; Saeed A; Shehzad M; Ullah Khan S; Lecka J; Sévigny J; Shabir G; Iqbal J
Bioorg Chem; 2018 Feb; 76():237-248. PubMed ID: 29197225
[TBL] [Abstract][Full Text] [Related]
11. In vitro effects of selected flavonoids on the 5'-nucleotidase activity.
Kavutcu M; Melzig MF
Pharmazie; 1999 Jun; 54(6):457-9. PubMed ID: 10399192
[TBL] [Abstract][Full Text] [Related]
12. Structure-based virtual screening approach to identify novel classes of PTP1B inhibitors.
Park H; Bhattarai BR; Ham SW; Cho H
Eur J Med Chem; 2009 Aug; 44(8):3280-4. PubMed ID: 19269068
[TBL] [Abstract][Full Text] [Related]
13. Isonicotinohydrazones as inhibitors of alkaline phosphatase and ecto-5'-nucleotidase.
Channar PA; Shah SJ; Hassan S; Nisa ZU; Lecka J; Sévigny J; Bajorath J; Saeed A; Iqbal J
Chem Biol Drug Des; 2017 Mar; 89(3):365-370. PubMed ID: 27589035
[TBL] [Abstract][Full Text] [Related]
14. Be Aware of Aggregators in the Search for Potential Human
Viviani LG; Piccirillo E; Cheffer A; de Rezende L; Ulrich H; Carmona-Ribeiro AM; Amaral AT
Molecules; 2018 Jul; 23(8):. PubMed ID: 30060466
[TBL] [Abstract][Full Text] [Related]
15. Synthesis, characterization and biological evaluation of novel chalcone sulfonamide hybrids as potent intestinal alkaline phosphatase inhibitors.
Ejaz SA; Saeed A; Siddique MN; Nisa ZU; Khan S; Lecka J; Sévigny J; Iqbal J
Bioorg Chem; 2017 Feb; 70():229-236. PubMed ID: 28110961
[TBL] [Abstract][Full Text] [Related]
16. α,β-Methylene-ADP (AOPCP) Derivatives and Analogues: Development of Potent and Selective ecto-5'-Nucleotidase (CD73) Inhibitors.
Bhattarai S; Freundlieb M; Pippel J; Meyer A; Abdelrahman A; Fiene A; Lee SY; Zimmermann H; Yegutkin GG; Sträter N; El-Tayeb A; Müller CE
J Med Chem; 2015 Aug; 58(15):6248-63. PubMed ID: 26147331
[TBL] [Abstract][Full Text] [Related]
17. Characterization of an ecto-5'-nucleotidase (EC 3.1.3.5) activity in intact trophozoites of Trichomonas gallinae.
Borges FP; Gottardi B; Stuepp C; Larré AB; Tasca T; De Carli GA; Bonan CD
Vet Parasitol; 2007 Jan; 143(2):106-11. PubMed ID: 16962709
[TBL] [Abstract][Full Text] [Related]
18. Identification of novel chromone based sulfonamides as highly potent and selective inhibitors of alkaline phosphatases.
al-Rashida M; Raza R; Abbas G; Shah MS; Kostakis GE; Lecka J; Sévigny J; Muddassar M; Papatriantafyllopoulou C; Iqbal J
Eur J Med Chem; 2013 Aug; 66():438-49. PubMed ID: 23831808
[TBL] [Abstract][Full Text] [Related]
19. Identification of small molecule sulfonic acids as ecto-5'-Nucleotidase inhibitors.
Raza R; Saeed A; Lecka J; Sévigny J; Iqbal J
Med Chem; 2012 Nov; 8(6):1133-9. PubMed ID: 22741787
[TBL] [Abstract][Full Text] [Related]
20. The effect of glibenclamide on the production of interstitial adenosine by inhibiting ecto-5'-nucleotidase in rat hearts.
Sato T; Obata T; Yamanaka Y; Arita M
Br J Pharmacol; 1997 Oct; 122(4):611-8. PubMed ID: 9375955
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]
