138 related articles for article (PubMed ID: 22731815)
21. Giardia duodenalis: biochemical characterization of an ecto-5'-nucleotidase activity.
Russo-Abrahão T; Cosentino-Gomes D; Daflon-Yunes N; Meyer-Fernandes JR
Exp Parasitol; 2011 Jan; 127(1):66-71. PubMed ID: 20599434
[TBL] [Abstract][Full Text] [Related]
22. Structure-based virtual screening of novel inhibitors of the uridyltransferase activity of Xanthomonas oryzae pv. oryzae GlmU.
Min J; Lin D; Zhang Q; Zhang J; Yu Z
Eur J Med Chem; 2012 Jul; 53():150-8. PubMed ID: 22521370
[TBL] [Abstract][Full Text] [Related]
23. Structural and Modeling Studies on ecto-5'-nucleotidase Aiding in Inhibitor Design.
Furtmann N; Bajorath J
Mini Rev Med Chem; 2015; 15(1):34-40. PubMed ID: 25694084
[TBL] [Abstract][Full Text] [Related]
24. Structure-based virtual screening approach to the discovery of novel inhibitors of factor-inhibiting HIF-1: identification of new chelating groups for the active-site ferrous ion.
Ko S; Lee MK; Shin D; Park H
Bioorg Med Chem; 2009 Nov; 17(22):7769-74. PubMed ID: 19822432
[TBL] [Abstract][Full Text] [Related]
25. CD73 inhibition by purine cytotoxic nucleoside analogue-based diphosphonates.
Dumontet C; Peyrottes S; Rabeson C; Cros-Perrial E; Géant PY; Chaloin L; Jordheim LP
Eur J Med Chem; 2018 Sep; 157():1051-1055. PubMed ID: 30176535
[TBL] [Abstract][Full Text] [Related]
26. Identification of allosteric inhibitors of the ecto-5'-nucleotidase (CD73) targeting the dimer interface.
Rahimova R; Fontanel S; Lionne C; Jordheim LP; Peyrottes S; Chaloin L
PLoS Comput Biol; 2018 Jan; 14(1):e1005943. PubMed ID: 29377887
[TBL] [Abstract][Full Text] [Related]
27. Crystal structure of the human ecto-5'-nucleotidase (CD73): insights into the regulation of purinergic signaling.
Knapp K; Zebisch M; Pippel J; El-Tayeb A; Müller CE; Sträter N
Structure; 2012 Dec; 20(12):2161-73. PubMed ID: 23142347
[TBL] [Abstract][Full Text] [Related]
28. A new, sensitive ecto-5'-nucleotidase assay for compound screening.
Freundlieb M; Zimmermann H; Müller CE
Anal Biochem; 2014 Feb; 446():53-8. PubMed ID: 24144488
[TBL] [Abstract][Full Text] [Related]
29. A domino reaction of 3-chlorochromones with aminoheterocycles. Synthesis of pyrazolopyridines and benzofuropyridines and their optical and ecto-5'-nucleotidase inhibitory effects.
Miliutina M; Janke J; Hassan S; Zaib S; Iqbal J; Lecka J; Sévigny J; Villinger A; Friedrich A; Lochbrunner S; Langer P
Org Biomol Chem; 2018 Jan; 16(5):717-732. PubMed ID: 29303198
[TBL] [Abstract][Full Text] [Related]
30. Characterization of an ecto-5'-nucleotidase (EC 3.1.3.5) activity in intact cells of Trichomonas vaginalis.
Tasca T; Bonan CD; Carli GA; Battastini AM; Sarkis JJ
Exp Parasitol; 2003 Oct; 105(2):167-73. PubMed ID: 14969694
[TBL] [Abstract][Full Text] [Related]
31. E-NTPDases and ecto-5'-nucleotidase expression profile in rat heart left ventricle and the extracellular nucleotide hydrolysis by their nerve terminal endings.
Rücker B; Almeida ME; Libermann TA; Zerbini LF; Wink MR; Sarkis JJ
Life Sci; 2008 Feb; 82(9-10):477-86. PubMed ID: 18201730
[TBL] [Abstract][Full Text] [Related]
32. Inhibition of CD73 AMP hydrolysis by a therapeutic antibody with a dual, non-competitive mechanism of action.
Geoghegan JC; Diedrich G; Lu X; Rosenthal K; Sachsenmeier KF; Wu H; Dall'Acqua WF; Damschroder MM
MAbs; 2016; 8(3):454-67. PubMed ID: 26854859
[TBL] [Abstract][Full Text] [Related]
33. Structure-based virtual screening approach to the discovery of phosphoinositide 3-kinase alpha inhibitors.
Park H; Choi H; Hong S; Kim D; Oh DS; Hong S
Bioorg Med Chem Lett; 2011 Apr; 21(7):2021-4. PubMed ID: 21354792
[TBL] [Abstract][Full Text] [Related]
34. Progresses in the pursuit of aldose reductase inhibitors: the structure-based lead optimization step.
Ramunno A; Cosconati S; Sartini S; Maglio V; Angiuoli S; La Pietra V; Di Maro S; Giustiniano M; La Motta C; Da Settimo F; Marinelli L; Novellino E
Eur J Med Chem; 2012 May; 51():216-26. PubMed ID: 22436396
[TBL] [Abstract][Full Text] [Related]
35. Vanillin analog--vanillyl mandelic acid, a novel specific inhibitor of snake venom 5'-nucleotidase.
Arun R; Arafat AS; D'Souza CJ; Sivaramakrishnan V; Dhananjaya BL
Arch Pharm (Weinheim); 2014 Sep; 347(9):616-23. PubMed ID: 25042467
[TBL] [Abstract][Full Text] [Related]
36. Structure-Activity Relationship of Purine and Pyrimidine Nucleotides as Ecto-5'-Nucleotidase (CD73) Inhibitors.
Junker A; Renn C; Dobelmann C; Namasivayam V; Jain S; Losenkova K; Irjala H; Duca S; Balasubramanian R; Chakraborty S; Börgel F; Zimmermann H; Yegutkin GG; Müller CE; Jacobson KA
J Med Chem; 2019 Apr; 62(7):3677-3695. PubMed ID: 30895781
[TBL] [Abstract][Full Text] [Related]
37. Design, synthesis and structure-activity relationship of novel [3.3.1] bicyclic sulfonamide-pyrazoles as potent γ-secretase inhibitors.
Aubele DL; Truong AP; Dressen DB; Probst GD; Bowers S; Mattson MN; Semko CM; Sun M; Garofalo AW; Konradi AW; Sham HL; Zmolek W; Wong K; Goldbach E; Quinn KP; Sauer JM; Brigham EF; Wallace W; Nguyen L; Bova MP; Hemphill SS; Basi G
Bioorg Med Chem Lett; 2011 Oct; 21(19):5791-4. PubMed ID: 21885276
[TBL] [Abstract][Full Text] [Related]
38. Some sulfonamide drugs inhibit ATPase activity of heat shock protein 90: investigation by docking simulation and experimental validation.
Sheikha GA; Al-Sha'er MA; Taha MO
J Enzyme Inhib Med Chem; 2011 Oct; 26(5):603-9. PubMed ID: 21190426
[TBL] [Abstract][Full Text] [Related]
39. Small-molecule CD73 inhibitors for the immunotherapy of cancer: a patent and literature review (2017-present).
Nocentini A; Capasso C; Supuran CT
Expert Opin Ther Pat; 2021 Oct; 31(10):867-876. PubMed ID: 33909515
[TBL] [Abstract][Full Text] [Related]
40. 3-hydroxymethyl-7-(N-substituted aminosulfonyl)-1,2,3,4-tetrahydroisoquinoline inhibitors of phenylethanolamine N-methyltransferase that display remarkable potency and selectivity.
Grunewald GL; Romero FA; Criscione KR
J Med Chem; 2005 Jan; 48(1):134-40. PubMed ID: 15634007
[TBL] [Abstract][Full Text] [Related]
[Previous] [Next] [New Search]
