These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.


BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

199 related articles for article (PubMed ID: 22883051)

  • 1. Insights into the structure and pharmacology of the human trace amine-associated receptor 1 (hTAAR1): homology modelling and docking studies.
    Cichero E; Espinoza S; Gainetdinov RR; Brasili L; Fossa P
    Chem Biol Drug Des; 2013 Apr; 81(4):509-16. PubMed ID: 22883051
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Further insights into the pharmacology of the human trace amine-associated receptors: discovery of novel ligands for TAAR1 by a virtual screening approach.
    Cichero E; Espinoza S; Franchini S; Guariento S; Brasili L; Gainetdinov RR; Fossa P
    Chem Biol Drug Des; 2014 Dec; 84(6):712-20. PubMed ID: 24894156
    [TBL] [Abstract][Full Text] [Related]  

  • 3. New insights into the structure of the trace amine-associated receptor 2: Homology modelling studies exploring the binding mode of 3-iodothyronamine.
    Cichero E; Tonelli M
    Chem Biol Drug Des; 2017 May; 89(5):790-796. PubMed ID: 27863038
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Differential modulation of Beta-adrenergic receptor signaling by trace amine-associated receptor 1 agonists.
    Kleinau G; Pratzka J; Nürnberg D; Grüters A; Führer-Sakel D; Krude H; Köhrle J; Schöneberg T; Biebermann H
    PLoS One; 2011; 6(10):e27073. PubMed ID: 22073124
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Targeting species-specific trace amine-associated receptor 1 ligands: to date perspective of the rational drug design process.
    Cichero E; Tonelli M
    Future Med Chem; 2017 Sep; 9(13):1507-1527. PubMed ID: 28791911
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Discovery of a Novel Chemo-Type for TAAR1 Agonism via Molecular Modeling.
    Grossi G; Scarano N; Musumeci F; Tonelli M; Kanov E; Carbone A; Fossa P; Gainetdinov RR; Cichero E; Schenone S
    Molecules; 2024 Apr; 29(8):. PubMed ID: 38675561
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Pharmacologic characterization of the cloned human trace amine-associated receptor1 (TAAR1) and evidence for species differences with the rat TAAR1.
    Wainscott DB; Little SP; Yin T; Tu Y; Rocco VP; He JX; Nelson DL
    J Pharmacol Exp Ther; 2007 Jan; 320(1):475-85. PubMed ID: 17038507
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Tyramine and β-phenylethylamine, from fermented food products, as agonists for the human trace amine-associated receptor 1 (hTAAR1) in the stomach.
    Ohta H; Takebe Y; Murakami Y; Takahama Y; Morimura S
    Biosci Biotechnol Biochem; 2017 May; 81(5):1002-1006. PubMed ID: 28084165
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Design, Synthesis, and Evaluation of Thyronamine Analogues as Novel Potent Mouse Trace Amine Associated Receptor 1 (mTAAR1) Agonists.
    Chiellini G; Nesi G; Digiacomo M; Malvasi R; Espinoza S; Sabatini M; Frascarelli S; Laurino A; Cichero E; Macchia M; Gainetdinov RR; Fossa P; Raimondi L; Zucchi R; Rapposelli S
    J Med Chem; 2015 Jun; 58(12):5096-107. PubMed ID: 26010728
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Recognition of methamphetamine and other amines by trace amine receptor TAAR1.
    Liu H; Zheng Y; Wang Y; Wang Y; He X; Xu P; Huang S; Yuan Q; Zhang X; Wang L; Jiang K; Chen H; Li Z; Liu W; Wang S; Xu HE; Xu F
    Nature; 2023 Dec; 624(7992):663-671. PubMed ID: 37935377
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Is there a role for biogenic amine receptors in mediating β-phenylethylamine and RO5256390-induced vascular contraction?
    Voisey AC; Broadley HD; Broadley KJ; Ford WR
    Eur J Pharmacol; 2024 Oct; 981():176895. PubMed ID: 39153650
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Trace amine-associated receptor 1: a multimodal therapeutic target for neuropsychiatric diseases.
    Schwartz MD; Canales JJ; Zucchi R; Espinoza S; Sukhanov I; Gainetdinov RR
    Expert Opin Ther Targets; 2018 Jun; 22(6):513-526. PubMed ID: 29798691
    [TBL] [Abstract][Full Text] [Related]  

  • 13. The molecular basis of species-specific ligand activation of trace amine-associated receptor 1 (TAAR(1)).
    Tan ES; Naylor JC; Groban ES; Bunzow JR; Jacobson MP; Grandy DK; Scanlan TS
    ACS Chem Biol; 2009 Mar; 4(3):209-20. PubMed ID: 19256523
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Interaction analyses of hTAAR1 and mTAAR1 with antagonist EPPTB.
    Liao S; Pino MJ; Deleon C; Lindner-Jackson M; Wu C
    Life Sci; 2022 Jul; 300():120553. PubMed ID: 35452636
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Search for Structural Basis of Interactions of Biogenic Amines with Human TAAR1 and TAAR6 Receptors.
    Glyakina AV; Pavlov CD; Sopova JV; Gainetdinov RR; Leonova EI; Galzitskaya OV
    Int J Mol Sci; 2021 Dec; 23(1):. PubMed ID: 35008636
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Toward deciphering the code to aminergic G protein-coupled receptor drug design.
    Tan ES; Groban ES; Jacobson MP; Scanlan TS
    Chem Biol; 2008 Apr; 15(4):343-53. PubMed ID: 18420141
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Identification of a Potent Human Trace Amine-Associated Receptor 1 Antagonist.
    Decker AM; Brackeen MF; Mohammadkhani A; Kormos CM; Hesk D; Borgland SL; Blough BE
    ACS Chem Neurosci; 2022 Apr; 13(7):1082-1095. PubMed ID: 35325532
    [TBL] [Abstract][Full Text] [Related]  

  • 18. TAAR1 activation modulates monoaminergic neurotransmission, preventing hyperdopaminergic and hypoglutamatergic activity.
    Revel FG; Moreau JL; Gainetdinov RR; Bradaia A; Sotnikova TD; Mory R; Durkin S; Zbinden KG; Norcross R; Meyer CA; Metzler V; Chaboz S; Ozmen L; Trube G; Pouzet B; Bettler B; Caron MG; Wettstein JG; Hoener MC
    Proc Natl Acad Sci U S A; 2011 May; 108(20):8485-90. PubMed ID: 21525407
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Novel biguanide-based derivatives scouted as TAAR1 agonists: Synthesis, biological evaluation, ADME prediction and molecular docking studies.
    Tonelli M; Espinoza S; Gainetdinov RR; Cichero E
    Eur J Med Chem; 2017 Feb; 127():781-792. PubMed ID: 27823885
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Potential of Ligands for Trace Amine-Associated Receptor 1 (TAAR1) in the Management of Substance Use Disorders.
    Wu R; Li JX
    CNS Drugs; 2021 Dec; 35(12):1239-1248. PubMed ID: 34766253
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 10.