149 related articles for article (PubMed ID: 22890306)
1. A two-directional strategy for the diversity-oriented synthesis of macrocyclic scaffolds.
O'Connell KM; Beckmann HS; Laraia L; Horsley HT; Bender A; Venkitaraman AR; Spring DR
Org Biomol Chem; 2012 Oct; 10(37):7545-51. PubMed ID: 22890306
[TBL] [Abstract][Full Text] [Related]
2. Diversity-oriented synthesis and cytotoxic activity evaluation of biaryl-containing macrocycles.
Pérez-Labrada K; Cruz-Mendoza MA; Chávez-Riveros A; Hernández-Vázquez E; Torroba T; Miranda LD
Org Biomol Chem; 2017 Mar; 15(11):2450-2458. PubMed ID: 28255584
[TBL] [Abstract][Full Text] [Related]
3. Design and synthesis of 14 and 15-membered macrocyclic scaffolds exhibiting inhibitory activities of hypoxia-inducible factor 1α.
Shimizu T; Takahashi N; Huber VJ; Asawa Y; Ueda H; Yoshimori A; Muramatsu Y; Seimiya H; Kouji H; Nakamura H; Oguri H
Bioorg Med Chem; 2021 Jan; 30():115949. PubMed ID: 33360196
[TBL] [Abstract][Full Text] [Related]
4. Macrocyclic pyrrolobenzodiazepine dimers as antibody-drug conjugate payloads.
Donnell AF; Zhang Y; Stang EM; Wei DD; Tebben AJ; Perez HL; Schroeder GM; Pan C; Rao C; Borzilleri RM; Vite GD; Gangwar S
Bioorg Med Chem Lett; 2017 Dec; 27(23):5267-5271. PubMed ID: 29102228
[TBL] [Abstract][Full Text] [Related]
5. Novel C2-C3' N-peptide linked macrocyclic taxoids. Part 2: synthesis and biological activities of docetaxel analogues with a peptide side chain at C2 and their macrocyclic derivatives.
Larroque AL; Dubois J; Thoret S; Aubert G; Chiaroni A; Guéritte F; Guénard D
Bioorg Med Chem; 2007 Jan; 15(1):563-74. PubMed ID: 17064914
[TBL] [Abstract][Full Text] [Related]
6. Synthesis and biological evaluation of nannocystin analogues toward understanding the binding role of the (2R,3S)-Epoxide in nannocystin A.
Tian Y; Xu X; Ding Y; Hao X; Bai Y; Tang Y; Zhang X; Li Q; Yang Z; Zhang W; Chen Y
Eur J Med Chem; 2018 Apr; 150():626-632. PubMed ID: 29554614
[TBL] [Abstract][Full Text] [Related]
7. Structure-based design, synthesis, and biological evaluation of potent and selective macrocyclic checkpoint kinase 1 inhibitors.
Tao ZF; Wang L; Stewart KD; Chen Z; Gu W; Bui MH; Merta P; Zhang H; Kovar P; Johnson E; Park C; Judge R; Rosenberg S; Sowin T; Lin NH
J Med Chem; 2007 Apr; 50(7):1514-27. PubMed ID: 17352464
[TBL] [Abstract][Full Text] [Related]
8. Diversity-oriented synthesis of macrocyclic peptidomimetics.
Isidro-Llobet A; Murillo T; Bello P; Cilibrizzi A; Hodgkinson JT; Galloway WR; Bender A; Welch M; Spring DR
Proc Natl Acad Sci U S A; 2011 Apr; 108(17):6793-8. PubMed ID: 21383137
[TBL] [Abstract][Full Text] [Related]
9. Synthesis and antiproliferative activity of new tonantzitlolone-derived diterpene derivatives.
Busch T; Dräger G; Kunst E; Benson H; Sasse F; Siems K; Kirschning A
Org Biomol Chem; 2016 Oct; 14(38):9040-5. PubMed ID: 27604289
[TBL] [Abstract][Full Text] [Related]
10. Exploring the physicochemical and antiproliferative properties of biaryl-linked [13]-macrodilactones.
Chen C; Bosko C; McGeough CP; McLean R; Zaino AM; Kyle Hadden M; Peczuh MW
Bioorg Med Chem; 2020 Oct; 28(20):115671. PubMed ID: 33069068
[TBL] [Abstract][Full Text] [Related]
11. A diversity-oriented synthesis strategy enabling the combinatorial-type variation of macrocyclic peptidomimetic scaffolds.
Isidro-Llobet A; Hadje Georgiou K; Galloway WR; Giacomini E; Hansen MR; Méndez-Abt G; Tan YS; Carro L; Sore HF; Spring DR
Org Biomol Chem; 2015 Apr; 13(15):4570-80. PubMed ID: 25778821
[TBL] [Abstract][Full Text] [Related]
12. Design, synthesis and biological evaluation of nitrogen-containing macrocyclic bisbibenzyl derivatives as potent anticancer agents by targeting the lysosome.
Sun B; Liu J; Gao Y; Zheng HB; Li L; Hu QW; Yuan HQ; Lou HX
Eur J Med Chem; 2017 Aug; 136():603-618. PubMed ID: 28570977
[TBL] [Abstract][Full Text] [Related]
13. Design, synthesis and biological evaluation of macrocyclic derivatives as TRK inhibitors.
Li P; Cai S; Zhao T; Xu L; Guan D; Li J; Zhou J; Zhang H
Bioorg Med Chem Lett; 2021 Dec; 53():128409. PubMed ID: 34628036
[TBL] [Abstract][Full Text] [Related]
14. Design and synthesis of novel macrocyclic 2-amino-6-arylpyrimidine Hsp90 inhibitors.
Suda A; Koyano H; Hayase T; Hada K; Kawasaki K; Komiyama S; Hasegawa K; Fukami TA; Sato S; Miura T; Ono N; Yamazaki T; Saitoh R; Shimma N; Shiratori Y; Tsukuda T
Bioorg Med Chem Lett; 2012 Jan; 22(2):1136-41. PubMed ID: 22192591
[TBL] [Abstract][Full Text] [Related]
15. Evaluation of alternative approaches for the synthesis of macrocyclic bisindolylmaleimides.
Bartlett S; Nelson A
Org Biomol Chem; 2004 Oct; 2(19):2874-83. PubMed ID: 15455163
[TBL] [Abstract][Full Text] [Related]
16. Novel nannocystin A analogues as anticancer therapeutics: Synthesis, biological evaluations and structure-activity relationship studies.
Liu Q; Yang X; Ji J; Zhang SL; He Y
Eur J Med Chem; 2019 May; 170():99-111. PubMed ID: 30878835
[TBL] [Abstract][Full Text] [Related]
17. Synthesis of macrocyclic bisbibenzyl derivatives and their anticancer effects as anti-tubulin agents.
Jiang J; Sun B; Wang YY; Cui M; Zhang L; Cui CZ; Wang YF; Liu XG; Lou HX
Bioorg Med Chem; 2012 Apr; 20(7):2382-91. PubMed ID: 22365913
[TBL] [Abstract][Full Text] [Related]
18. Cytotoxic Activity and Structure-Activity Relationship of Triazole-Containing Bis(Aryl Ether) Macrocycles.
Hernández-Vázquez E; Chávez-Riveros A; Romo-Pérez A; Ramírez-Apán MT; Chávez-Blanco AD; Morales-Bárcenas R; Dueñas-González A; Miranda LD
ChemMedChem; 2018 Jun; 13(12):1193-1209. PubMed ID: 29771004
[TBL] [Abstract][Full Text] [Related]
19. Macrocyclic architecture: tuning cavity size and shape through maleimide photochemistry.
Cubbage KL; Corrie T; Evans N; Haddow MF; Booker-Milburn KI
Chemistry; 2012 Sep; 18(36):11180-3. PubMed ID: 22836672
[No Abstract] [Full Text] [Related]
20. Exploring the Ring-Closing Metathesis for the Construction of the Solomonamide Macrocyclic Core: Identification of Bioactive Precursors.
Cheng-Sánchez I; Carrillo P; Sánchez-Ruiz A; Martínez-Poveda B; Quesada AR; Medina MA; López-Romero JM; Sarabia F
J Org Chem; 2018 May; 83(10):5365-5383. PubMed ID: 29676156
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]
