These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.


BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

136 related articles for article (PubMed ID: 22901388)

  • 1. Inhibition of α-class cytosolic human carbonic anhydrases I, II, IX and XII, and β-class fungal enzymes by carboxylic acids and their derivatives: new isoform-I selective nanomolar inhibitors.
    Sechi M; Innocenti A; Pala N; Rogolino D; Carcelli M; Scozzafava A; Supuran CT
    Bioorg Med Chem Lett; 2012 Sep; 22(18):5801-6. PubMed ID: 22901388
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Carbonic anhydrase inhibitors. Inhibition of the β-class enzymes from the fungal pathogens Candida albicans and Cryptococcus neoformans with branched aliphatic/aromatic carboxylates and their derivatives.
    Carta F; Innocenti A; Hall RA; Mühlschlegel FA; Scozzafava A; Supuran CT
    Bioorg Med Chem Lett; 2011 Apr; 21(8):2521-6. PubMed ID: 21402476
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Synthesis of rhodamine B-benzenesulfonamide conjugates and their inhibitory activity against human α- and bacterial/fungal β-carbonic anhydrases.
    Rami M; Innocenti A; Montero JL; Scozzafava A; Winum JY; Supuran CT
    Bioorg Med Chem Lett; 2011 Sep; 21(18):5210-3. PubMed ID: 21821413
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Sulfonamides incorporating 1,3,5-triazine moieties selectively and potently inhibit carbonic anhydrase transmembrane isoforms IX, XII and XIV over cytosolic isoforms I and II: Solution and X-ray crystallographic studies.
    Carta F; Garaj V; Maresca A; Wagner J; Avvaru BS; Robbins AH; Scozzafava A; McKenna R; Supuran CT
    Bioorg Med Chem; 2011 May; 19(10):3105-19. PubMed ID: 21515057
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Carbonic anhydrase inhibitors: inhibition of human cytosolic isozymes I and II and tumor-associated isozymes IX and XII with S-substituted 4-chloro-2-mercapto-5-methyl-benzenesulfonamides.
    Saczewski F; Innocenti A; Sławiński J; Kornicka A; Brzozowski Z; Pomarnacka E; Scozzafava A; Temperini C; Supuran CT
    Bioorg Med Chem; 2008 Apr; 16(7):3933-40. PubMed ID: 18242998
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Carbonic anhydrase inhibitory activity of sulfonamides and carboxylic acids incorporating cyclic imide scaffolds.
    Abdel-Aziz AA; El-Azab AS; Ceruso M; Supuran CT
    Bioorg Med Chem Lett; 2014 Nov; 24(22):5185-9. PubMed ID: 25442309
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Inhibition of the β-class carbonic anhydrases from Mycobacterium tuberculosis with carboxylic acids.
    Maresca A; Vullo D; Scozzafava A; Manole G; Supuran CT
    J Enzyme Inhib Med Chem; 2013 Apr; 28(2):392-6. PubMed ID: 22299588
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Carbonic anhydrase inhibitors. Inhibition of the beta-class enzymes from the fungal pathogens Candida albicans and Cryptococcus neoformans with aliphatic and aromatic carboxylates.
    Innocenti A; Hall RA; Schlicker C; Mühlschlegel FA; Supuran CT
    Bioorg Med Chem; 2009 Apr; 17(7):2654-7. PubMed ID: 19297172
    [TBL] [Abstract][Full Text] [Related]  

  • 9. New chemotypes acting as isozyme-selective carbonic anhydrase inhibitors with low affinity for the offtarget cytosolic isoform II.
    Carta F; Vullo D; Maresca A; Scozzafava A; Supuran CT
    Bioorg Med Chem Lett; 2012 Mar; 22(6):2182-5. PubMed ID: 22365761
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Design, synthesis and evaluation of N-substituted saccharin derivatives as selective inhibitors of tumor-associated carbonic anhydrase XII.
    D'Ascenzio M; Carradori S; De Monte C; Secci D; Ceruso M; Supuran CT
    Bioorg Med Chem; 2014 Mar; 22(6):1821-31. PubMed ID: 24560739
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Carbonic anhydrase inhibitors. Inhibition of the fungal beta-carbonic anhydrases from Candida albicans and Cryptococcus neoformans with boronic acids.
    Innocenti A; Winum JY; Hall RA; Mühlschlegel FA; Scozzafava A; Supuran CT
    Bioorg Med Chem Lett; 2009 May; 19(10):2642-5. PubMed ID: 19375309
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Carbonic anhydrase inhibitors: inhibition of mammalian isoforms I-XIV with a series of substituted phenols including paracetamol and salicylic acid.
    Innocenti A; Vullo D; Scozzafava A; Supuran CT
    Bioorg Med Chem; 2008 Aug; 16(15):7424-8. PubMed ID: 18579385
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Attachment of carbohydrates to methoxyaryl moieties leads to highly selective inhibitors of the cancer associated carbonic anhydrase isoforms IX and XII.
    Riafrecha LE; Rodríguez OM; Vullo D; Supuran CT; Colinas PA
    Bioorg Med Chem; 2014 Oct; 22(19):5308-14. PubMed ID: 25156300
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Cyclic tertiary sulfamates: selective inhibition of the tumor-associated carbonic anhydrases IX and XII by N- and O-substituted acesulfame derivatives.
    De Monte C; Carradori S; Secci D; D'Ascenzio M; Vullo D; Ceruso M; Supuran CT
    Eur J Med Chem; 2014 Sep; 84():240-6. PubMed ID: 25019479
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Carbonic anhydrase inhibitors. Inhibition of human cytosolic isoforms I and II with (reduced) Schiff's bases incorporating sulfonamide, carboxylate and carboxymethyl moieties.
    Nasr G; Cristian A; Barboiu M; Vullo D; Winum JY; Supuran CT
    Bioorg Med Chem; 2014 May; 22(10):2867-74. PubMed ID: 24746465
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Dithiocarbamates are strong inhibitors of the beta-class fungal carbonic anhydrases from Cryptococcus neoformans, Candida albicans and Candida glabrata.
    Monti SM; Maresca A; Viparelli F; Carta F; De Simone G; Mühlschlegel FA; Scozzafava A; Supuran CT
    Bioorg Med Chem Lett; 2012 Jan; 22(2):859-62. PubMed ID: 22209456
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Carbonic anhydrase inhibitors. Identification of selective inhibitors of the human mitochondrial isozymes VA and VB over the cytosolic isozymes I and II from a natural product-based phenolic library.
    Davis RA; Innocenti A; Poulsen SA; Supuran CT
    Bioorg Med Chem; 2010 Jan; 18(1):14-8. PubMed ID: 19962903
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Synthesis of aminocyanopyrazoles via a multi-component reaction and anti-carbonic anhydrase inhibitory activity of their sulfamide derivatives against cytosolic and transmembrane isoforms.
    Allouche F; Chabchoub F; Carta F; Supuran CT
    J Enzyme Inhib Med Chem; 2013 Apr; 28(2):343-9. PubMed ID: 23013533
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Kinetic and in silico analysis of thiazolidin-based inhibitors of α-carbonic anhydrase isoenzymes.
    Ekinci D; Fidan İ; Durdagi S; Kaban Ş; Supuran CT
    J Enzyme Inhib Med Chem; 2013 Apr; 28(2):370-4. PubMed ID: 23173744
    [TBL] [Abstract][Full Text] [Related]  

  • 20. C-glycosides incorporating the 6-methoxy-2-naphthyl moiety are selective inhibitors of fungal and bacterial carbonic anhydrases.
    Riafrecha LE; Vullo D; Supuran CT; Colinas PA
    J Enzyme Inhib Med Chem; 2015; 30(5):857-61. PubMed ID: 25291009
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 7.