142 related articles for article (PubMed ID: 22901388)
1. Inhibition of α-class cytosolic human carbonic anhydrases I, II, IX and XII, and β-class fungal enzymes by carboxylic acids and their derivatives: new isoform-I selective nanomolar inhibitors.
Sechi M; Innocenti A; Pala N; Rogolino D; Carcelli M; Scozzafava A; Supuran CT
Bioorg Med Chem Lett; 2012 Sep; 22(18):5801-6. PubMed ID: 22901388
[TBL] [Abstract][Full Text] [Related]
2. Carbonic anhydrase inhibitors. Inhibition of the β-class enzymes from the fungal pathogens Candida albicans and Cryptococcus neoformans with branched aliphatic/aromatic carboxylates and their derivatives.
Carta F; Innocenti A; Hall RA; Mühlschlegel FA; Scozzafava A; Supuran CT
Bioorg Med Chem Lett; 2011 Apr; 21(8):2521-6. PubMed ID: 21402476
[TBL] [Abstract][Full Text] [Related]
3. Synthesis of rhodamine B-benzenesulfonamide conjugates and their inhibitory activity against human α- and bacterial/fungal β-carbonic anhydrases.
Rami M; Innocenti A; Montero JL; Scozzafava A; Winum JY; Supuran CT
Bioorg Med Chem Lett; 2011 Sep; 21(18):5210-3. PubMed ID: 21821413
[TBL] [Abstract][Full Text] [Related]
4. Sulfonamides incorporating 1,3,5-triazine moieties selectively and potently inhibit carbonic anhydrase transmembrane isoforms IX, XII and XIV over cytosolic isoforms I and II: Solution and X-ray crystallographic studies.
Carta F; Garaj V; Maresca A; Wagner J; Avvaru BS; Robbins AH; Scozzafava A; McKenna R; Supuran CT
Bioorg Med Chem; 2011 May; 19(10):3105-19. PubMed ID: 21515057
[TBL] [Abstract][Full Text] [Related]
5. Carbonic anhydrase inhibitors: inhibition of human cytosolic isozymes I and II and tumor-associated isozymes IX and XII with S-substituted 4-chloro-2-mercapto-5-methyl-benzenesulfonamides.
Saczewski F; Innocenti A; Sławiński J; Kornicka A; Brzozowski Z; Pomarnacka E; Scozzafava A; Temperini C; Supuran CT
Bioorg Med Chem; 2008 Apr; 16(7):3933-40. PubMed ID: 18242998
[TBL] [Abstract][Full Text] [Related]
6. Carbonic anhydrase inhibitory activity of sulfonamides and carboxylic acids incorporating cyclic imide scaffolds.
Abdel-Aziz AA; El-Azab AS; Ceruso M; Supuran CT
Bioorg Med Chem Lett; 2014 Nov; 24(22):5185-9. PubMed ID: 25442309
[TBL] [Abstract][Full Text] [Related]
7. Inhibition of the β-class carbonic anhydrases from Mycobacterium tuberculosis with carboxylic acids.
Maresca A; Vullo D; Scozzafava A; Manole G; Supuran CT
J Enzyme Inhib Med Chem; 2013 Apr; 28(2):392-6. PubMed ID: 22299588
[TBL] [Abstract][Full Text] [Related]
8. Carbonic anhydrase inhibitors. Inhibition of the beta-class enzymes from the fungal pathogens Candida albicans and Cryptococcus neoformans with aliphatic and aromatic carboxylates.
Innocenti A; Hall RA; Schlicker C; Mühlschlegel FA; Supuran CT
Bioorg Med Chem; 2009 Apr; 17(7):2654-7. PubMed ID: 19297172
[TBL] [Abstract][Full Text] [Related]
9. New chemotypes acting as isozyme-selective carbonic anhydrase inhibitors with low affinity for the offtarget cytosolic isoform II.
Carta F; Vullo D; Maresca A; Scozzafava A; Supuran CT
Bioorg Med Chem Lett; 2012 Mar; 22(6):2182-5. PubMed ID: 22365761
[TBL] [Abstract][Full Text] [Related]
10. Design, synthesis and evaluation of N-substituted saccharin derivatives as selective inhibitors of tumor-associated carbonic anhydrase XII.
D'Ascenzio M; Carradori S; De Monte C; Secci D; Ceruso M; Supuran CT
Bioorg Med Chem; 2014 Mar; 22(6):1821-31. PubMed ID: 24560739
[TBL] [Abstract][Full Text] [Related]
11. Carbonic anhydrase inhibitors. Inhibition of the fungal beta-carbonic anhydrases from Candida albicans and Cryptococcus neoformans with boronic acids.
Innocenti A; Winum JY; Hall RA; Mühlschlegel FA; Scozzafava A; Supuran CT
Bioorg Med Chem Lett; 2009 May; 19(10):2642-5. PubMed ID: 19375309
[TBL] [Abstract][Full Text] [Related]
12. Carbonic anhydrase inhibitors: inhibition of mammalian isoforms I-XIV with a series of substituted phenols including paracetamol and salicylic acid.
Innocenti A; Vullo D; Scozzafava A; Supuran CT
Bioorg Med Chem; 2008 Aug; 16(15):7424-8. PubMed ID: 18579385
[TBL] [Abstract][Full Text] [Related]
13. Attachment of carbohydrates to methoxyaryl moieties leads to highly selective inhibitors of the cancer associated carbonic anhydrase isoforms IX and XII.
Riafrecha LE; Rodríguez OM; Vullo D; Supuran CT; Colinas PA
Bioorg Med Chem; 2014 Oct; 22(19):5308-14. PubMed ID: 25156300
[TBL] [Abstract][Full Text] [Related]
14. Cyclic tertiary sulfamates: selective inhibition of the tumor-associated carbonic anhydrases IX and XII by N- and O-substituted acesulfame derivatives.
De Monte C; Carradori S; Secci D; D'Ascenzio M; Vullo D; Ceruso M; Supuran CT
Eur J Med Chem; 2014 Sep; 84():240-6. PubMed ID: 25019479
[TBL] [Abstract][Full Text] [Related]
15. Carbonic anhydrase inhibitors. Inhibition of human cytosolic isoforms I and II with (reduced) Schiff's bases incorporating sulfonamide, carboxylate and carboxymethyl moieties.
Nasr G; Cristian A; Barboiu M; Vullo D; Winum JY; Supuran CT
Bioorg Med Chem; 2014 May; 22(10):2867-74. PubMed ID: 24746465
[TBL] [Abstract][Full Text] [Related]
16. Dithiocarbamates are strong inhibitors of the beta-class fungal carbonic anhydrases from Cryptococcus neoformans, Candida albicans and Candida glabrata.
Monti SM; Maresca A; Viparelli F; Carta F; De Simone G; Mühlschlegel FA; Scozzafava A; Supuran CT
Bioorg Med Chem Lett; 2012 Jan; 22(2):859-62. PubMed ID: 22209456
[TBL] [Abstract][Full Text] [Related]
17. Carbonic anhydrase inhibitors. Identification of selective inhibitors of the human mitochondrial isozymes VA and VB over the cytosolic isozymes I and II from a natural product-based phenolic library.
Davis RA; Innocenti A; Poulsen SA; Supuran CT
Bioorg Med Chem; 2010 Jan; 18(1):14-8. PubMed ID: 19962903
[TBL] [Abstract][Full Text] [Related]
18. Synthesis of aminocyanopyrazoles via a multi-component reaction and anti-carbonic anhydrase inhibitory activity of their sulfamide derivatives against cytosolic and transmembrane isoforms.
Allouche F; Chabchoub F; Carta F; Supuran CT
J Enzyme Inhib Med Chem; 2013 Apr; 28(2):343-9. PubMed ID: 23013533
[TBL] [Abstract][Full Text] [Related]
19. Kinetic and in silico analysis of thiazolidin-based inhibitors of α-carbonic anhydrase isoenzymes.
Ekinci D; Fidan İ; Durdagi S; Kaban Ş; Supuran CT
J Enzyme Inhib Med Chem; 2013 Apr; 28(2):370-4. PubMed ID: 23173744
[TBL] [Abstract][Full Text] [Related]
20. C-glycosides incorporating the 6-methoxy-2-naphthyl moiety are selective inhibitors of fungal and bacterial carbonic anhydrases.
Riafrecha LE; Vullo D; Supuran CT; Colinas PA
J Enzyme Inhib Med Chem; 2015; 30(5):857-61. PubMed ID: 25291009
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]
