These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.


BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

138 related articles for article (PubMed ID: 22958368)

  • 1. Synthesis and anti-HIV properties of new carbamate prodrugs of AZT.
    Solyev PN; Shipitsin AV; Karpenko IL; Nosik DN; Kalnina LB; Kochetkov SN; Kukhanova MK; Jasko MV
    Chem Biol Drug Des; 2012 Dec; 80(6):947-52. PubMed ID: 22958368
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Synthesis, in vitro and in vivo release kinetics, and anti-HIV activity of a sustained-release prodrug (mPEG-AZT) of 3'-azido-3'-deoxythymidine (AZT, Zidovudine).
    Li W; Chang Y; Zhan P; Zhang N; Liu X; Pannecouque C; De Clercq E
    ChemMedChem; 2010 Nov; 5(11):1893-8. PubMed ID: 20936623
    [TBL] [Abstract][Full Text] [Related]  

  • 3. New 3'-azido-3'-deoxythymidin-5'-yl O-(omega-hydroxyalkyl) carbonate prodrugs: synthesis and anti-HIV evaluation.
    Vlieghe P; Bihel F; Clerc T; Pannecouque C; Witvrouw M; De Clercq E; Salles JP; Chermann JC; Kraus JL
    J Med Chem; 2001 Mar; 44(5):777-86. PubMed ID: 11262088
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Poly(HEMA-Zidovudine) conjugate: a macromolecular pro-drug for improvement in the biopharmaceutical properties of the drug.
    Neeraj A; Chandrasekar MJ; Sara UV; Rohini A
    Drug Deliv; 2011 May; 18(4):272-80. PubMed ID: 21110710
    [TBL] [Abstract][Full Text] [Related]  

  • 5. In vitro and in vivo pharmacokinetic characterization of two novel prodrugs of zidovudine.
    Quevedo MA; Briñón MC
    Antiviral Res; 2009 Aug; 83(2):103-11. PubMed ID: 19549583
    [TBL] [Abstract][Full Text] [Related]  

  • 6. 5'-aminocarbonyl phosphonates as new zidovudine depot forms: antiviral properties, intracellular transformations, and pharmacokinetic parameters.
    Khandazhinskaya AL; Yanvarev DV; Jasko MV; Shipitsin AV; Khalizev VA; Shram SI; Skoblov YS; Shirokova EA; Kukhanova MK
    Drug Metab Dispos; 2009 Mar; 37(3):494-501. PubMed ID: 19106116
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Dipeptide derivatives of AZT: synthesis, chemical stability, activation in human plasma, hPEPT1 affinity, and antiviral activity.
    Santos C; Morais J; Gouveia L; de Clercq E; Pannecouque C; Nielsen CU; Steffansen B; Moreira R; Gomes P
    ChemMedChem; 2008 Jun; 3(6):970-8. PubMed ID: 18389514
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Synthesis and preliminary evaluation of anti-HIV agent AZT prodrug.
    Cui QB; Zhang GX; Yu P; Wang YQ
    Yao Xue Xue Bao; 2011 Aug; 46(8):1015-8. PubMed ID: 22007530
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Novel approaches for designing 5'-O-ester prodrugs of 3'-azido-2', 3'-dideoxythymidine (AZT).
    Parang K; Wiebe LI; Knaus EE
    Curr Med Chem; 2000 Oct; 7(10):995-1039. PubMed ID: 10911016
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Synthesis and antiviral activity of amino acid carbamate derivatives of AZT.
    Chang SL; Griesgraber G; Abraham TW; Garg T; Song H; Zimmerman CL; Wagner CR
    Nucleosides Nucleotides Nucleic Acids; 2000; 19(1-2):87-100. PubMed ID: 10772704
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Combination anti-HIV therapy with the self-assemblies of an asymmetric bolaamphiphilic zidovudine/didanosine prodrug.
    Jin Y; Xin R; Tong L; Du L; Li M
    Mol Pharm; 2011 Jun; 8(3):867-76. PubMed ID: 21553876
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Synthesis, in vitro anti-human immunodeficiency virus structure-activity relationships and biological stability of 5'-O-myristoyl analogue derivatives of 3'-azido-2',3'-dideoxythymidine (AZT) as potential prodrugs.
    Parang K; Wiebe LI; Knaus EE
    Antivir Chem Chemother; 1998 Jul; 9(4):311-23. PubMed ID: 9875410
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Synthesis of methoxypoly(ethylene glycol) carbonate prodrugs of zidovudine and penetration through human skin in vitro.
    N'da DD; Breytenbach JC
    J Pharm Pharmacol; 2009 Jun; 61(6):721-31. PubMed ID: 19505362
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Self-assembled drug delivery systems. Part 4. In vitro/in vivo studies of the self-assemblies of cholesteryl-phosphonyl zidovudine.
    Jin Y; Xing L; Tian Y; Li M; Gao C; Du L; Dong J; Chen H
    Int J Pharm; 2009 Oct; 381(1):40-8. PubMed ID: 19646518
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Synthesis and anti-HIV activity of steroidal prodrugs of 3'-azido-3'-deoxythymidine (AZT).
    Balagopala MI; Ollapally AP; Lee HJ
    Cell Mol Biol (Noisy-le-grand); 1995; 41 Suppl 1():S1-7. PubMed ID: 8574137
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Pharmacokinetics of bis(t-butyl-SATE)-AZTMP, a bispivaloylthioethyl prodrug for intracellular delivery of zidovudine monophosphate, in mice.
    Tan X; Boudinot FD; Chu CK; Egron D; Perigaud C; Gosselin G; Imbach JL
    Antivir Chem Chemother; 2000 May; 11(3):203-11. PubMed ID: 10901291
    [TBL] [Abstract][Full Text] [Related]  

  • 17. In vivo biodistribution, pharmacokinetic parameters, and brain uptake of 5-halo-y-methoxy(or ethoxy)-5,6-dihydro-3'-azido-3'-deoxythymidine diastereomers as potential prodrugs of 3'-azido-3'-deoxythymidine.
    Wang L; Morin KW; Kumar R; Cheraghali M; Todd KG; Baker GB; Knaus EE; Wiebe LI
    J Med Chem; 1996 Feb; 39(4):826-33. PubMed ID: 8632406
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Synthesis, anti-HIV, and cytotoxic activity of new AZT conjugates of steroid acids.
    You Z; Mian AM; Agarwal RP; Lee HJ
    Nucleosides Nucleotides Nucleic Acids; 2003 Nov; 22(11):2049-60. PubMed ID: 14680027
    [TBL] [Abstract][Full Text] [Related]  

  • 19. New dinucleoside phosphonate derivatives as prodrugs of 3'-azido-3'-deoxythymidine and β-L-2',3'-dideoxy-3'-thiacytidine: synthesis and anti-HIV properties.
    Solyev PN; Jasko MV; Karpenko IL; Sharkin YA; Shipitsyn AV; Kukhanova MK
    Nucleosides Nucleotides Nucleic Acids; 2014; 33(2):64-79. PubMed ID: 24660881
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Uncharged AZT and D4T derivatives of phosphonoformic and phosphonoacetic acids as anti-HIV pronucleosides.
    Shirokova EA; Jasko MV; Khandazhinskaya AL; Ivanov AV; Yanvarev DV; Skoblov YS; Mitkevich VA; Bocharov EV; Pronyaeva TR; Fedyuk NV; Kukhanova MK; Pokrovsky AG
    J Med Chem; 2004 Jul; 47(14):3606-14. PubMed ID: 15214788
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 7.