194 related articles for article (PubMed ID: 23008217)
1. Sulfonyl fluoride analogues as activity-based probes for serine proteases.
Shannon DA; Gu C; McLaughlin CJ; Kaiser M; van der Hoorn RA; Weerapana E
Chembiochem; 2012 Nov; 13(16):2327-30. PubMed ID: 23008217
[TBL] [Abstract][Full Text] [Related]
2. Synthesis and biological evaluation of novel irreversible serine protease inhibitors using amino acid based sulfonyl fluorides as an electrophilic trap.
Brouwer AJ; Ceylan T; Jonker AM; van der Linden T; Liskamp RM
Bioorg Med Chem; 2011 Apr; 19(7):2397-406. PubMed ID: 21421320
[TBL] [Abstract][Full Text] [Related]
3. Tuning activity-based probe selectivity for serine proteases by on-resin 'click' construction of peptide diphenyl phosphonates.
Serim S; Mayer SV; Verhelst SH
Org Biomol Chem; 2013 Sep; 11(34):5714-21. PubMed ID: 23884325
[TBL] [Abstract][Full Text] [Related]
4. Rational targeting of active-site tyrosine residues using sulfonyl fluoride probes.
Hett EC; Xu H; Geoghegan KF; Gopalsamy A; Kyne RE; Menard CA; Narayanan A; Parikh MD; Liu S; Roberts L; Robinson RP; Tones MA; Jones LH
ACS Chem Biol; 2015 Apr; 10(4):1094-8. PubMed ID: 25571984
[TBL] [Abstract][Full Text] [Related]
5. Chemoselective Preparation of Clickable Aryl Sulfonyl Fluoride Monomers: A Toolbox of Highly Functionalized Intermediates for Chemical Biology Probe Synthesis.
Fadeyi O; Parikh MD; Chen MZ; Kyne RE; Taylor AP; O'Doherty I; Kaiser SE; Barbas S; Niessen S; Shi M; Weinrich SL; Kath JC; Jones LH; Robinson RP
Chembiochem; 2016 Oct; 17(20):1925-1930. PubMed ID: 27504718
[TBL] [Abstract][Full Text] [Related]
6. Alkyne derivatives of isocoumarins as clickable activity-based probes for serine proteases.
Haedke U; Götz M; Baer P; Verhelst SH
Bioorg Med Chem; 2012 Jan; 20(2):633-40. PubMed ID: 21454080
[TBL] [Abstract][Full Text] [Related]
7. Synthesis of novel phosphonic-type activity-based probes for neutrophil serine proteases and their application in spleen lysates of different organisms.
Grzywa R; Burchacka E; Łęcka M; Winiarski Ł; Walczak M; Łupicka-Słowik A; Wysocka M; Burster T; Bobrek K; Csencsits-Smith K; Lesner A; Sieńczyk M
Chembiochem; 2014 Nov; 15(17):2605-12. PubMed ID: 25236966
[TBL] [Abstract][Full Text] [Related]
8. SuFEx-enabled, agnostic discovery of covalent inhibitors of human neutrophil elastase.
Zheng Q; Woehl JL; Kitamura S; Santos-Martins D; Smedley CJ; Li G; Forli S; Moses JE; Wolan DW; Sharpless KB
Proc Natl Acad Sci U S A; 2019 Sep; 116(38):18808-18814. PubMed ID: 31484779
[TBL] [Abstract][Full Text] [Related]
9. Europium-labeled activity-based probe through click chemistry: absolute serine protease quantification using (153)Eu isotope dilution ICP/MS.
Yan X; Luo Y; Zhang Z; Li Z; Luo Q; Yang L; Zhang B; Chen H; Bai P; Wang Q
Angew Chem Int Ed Engl; 2012 Apr; 51(14):3358-63. PubMed ID: 22344943
[TBL] [Abstract][Full Text] [Related]
10. Tailored Ahp-cyclodepsipeptides as Potent Non-covalent Serine Protease Inhibitors.
Köcher S; Rey J; Bongard J; Tiaden AN; Meltzer M; Richards PJ; Ehrmann M; Kaiser M
Angew Chem Int Ed Engl; 2017 Jul; 56(29):8555-8558. PubMed ID: 28514117
[TBL] [Abstract][Full Text] [Related]
11. Fatty Acyl Sulfonyl Fluoride as an Activity-Based Probe for Profiling Fatty Acid-Associated Proteins in Living Cells.
Zhang D; Lu M; Chen C; Xu Y; Peng T
Chembiochem; 2022 Feb; 23(4):e202100628. PubMed ID: 34918441
[TBL] [Abstract][Full Text] [Related]
12. Ahp cyclodepsipeptides: the impact of the Ahp residue on the "canonical inhibition" of S1 serine proteases.
Stolze SC; Meltzer M; Ehrmann M; Kaiser M
Chembiochem; 2013 Jul; 14(11):1301-8. PubMed ID: 23794257
[TBL] [Abstract][Full Text] [Related]
13. Potential peptidic proteasome inhibitors by incorporation of an electrophilic trap based on amino acid derived α-substituted sulfonyl fluorides.
Herrero Alvarez N; van de Langemheen H; Brouwer AJ; Liskamp RMJ
Bioorg Med Chem; 2017 Oct; 25(19):5055-5063. PubMed ID: 28734665
[TBL] [Abstract][Full Text] [Related]
14. Broad-Spectrum Kinase Profiling in Live Cells with Lysine-Targeted Sulfonyl Fluoride Probes.
Zhao Q; Ouyang X; Wan X; Gajiwala KS; Kath JC; Jones LH; Burlingame AL; Taunton J
J Am Chem Soc; 2017 Jan; 139(2):680-685. PubMed ID: 28051857
[TBL] [Abstract][Full Text] [Related]
15. α-Amino-α'-halomethylketones: synthetic methodologies and pharmaceutical applications as serine and cysteine protease inhibitors.
Pace V; Castoldi L; Pregnolato M
Mini Rev Med Chem; 2013 Jun; 13(7):988-96. PubMed ID: 22931530
[TBL] [Abstract][Full Text] [Related]
16. Production, partial purification and characterization of protease from a phytopathogenic fungi Alternaria solani (Ell. and Mart.) Sorauer.
Chandrasekaran M; Sathiyabama M
J Basic Microbiol; 2014 Aug; 54(8):763-74. PubMed ID: 23712744
[TBL] [Abstract][Full Text] [Related]
17. Phosphoramidates as novel activity-based probes for serine proteases.
Haedke UR; Frommel SC; Hansen F; Hahne H; Kuster B; Bogyo M; Verhelst SH
Chembiochem; 2014 May; 15(8):1106-10. PubMed ID: 24817682
[TBL] [Abstract][Full Text] [Related]
18. Beta-sultams-mechanism of reactions and use as inhibitors of serine proteases.
Page MI
Acc Chem Res; 2004 May; 37(5):297-303. PubMed ID: 15147170
[TBL] [Abstract][Full Text] [Related]
19. Chemical proteomics with sulfonyl fluoride probes reveals selective labeling of functional tyrosines in glutathione transferases.
Gu C; Shannon DA; Colby T; Wang Z; Shabab M; Kumari S; Villamor JG; McLaughlin CJ; Weerapana E; Kaiser M; Cravatt BF; van der Hoorn RA
Chem Biol; 2013 Apr; 20(4):541-8. PubMed ID: 23601643
[TBL] [Abstract][Full Text] [Related]
20. Synthesis and biochemical evaluation of triazole/tetrazole-containing sulfonamides against thrombin and related serine proteases.
Siles R; Kawasaki Y; Ross P; Freire E
Bioorg Med Chem Lett; 2011 Sep; 21(18):5305-9. PubMed ID: 21807511
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]