156 related articles for article (PubMed ID: 23020658)
1. Biochemical characterization of selective inhibitors of human group IIA secreted phospholipase A(2) and hyaluronic acid-linked inhibitor conjugates.
Oslund RC; Gelb MH
Biochemistry; 2012 Oct; 51(43):8617-26. PubMed ID: 23020658
[TBL] [Abstract][Full Text] [Related]
2. Inhibition of the complete set of mammalian secreted phospholipases A(2) by indole analogues: a structure-guided study.
Smart BP; Pan YH; Weeks AK; Bollinger JG; Bahnson BJ; Gelb MH
Bioorg Med Chem; 2004 Apr; 12(7):1737-49. PubMed ID: 15028265
[TBL] [Abstract][Full Text] [Related]
3. Design of new secreted phospholipase A2 inhibitors based on docking calculations by modifying the pharmacophore segments of the FPL67047XX inhibitor.
Mouchlis VD; Mavromoustakos TM; Kokotos G
J Comput Aided Mol Des; 2010 Feb; 24(2):107-15. PubMed ID: 20130961
[TBL] [Abstract][Full Text] [Related]
4. Secreted phospholipase A2 inhibitors are also potent blockers of binding to the M-type receptor.
Boilard E; Rouault M; Surrel F; Le Calvez C; Bezzine S; Singer A; Gelb MH; Lambeau G
Biochemistry; 2006 Nov; 45(44):13203-18. PubMed ID: 17073442
[TBL] [Abstract][Full Text] [Related]
5. Molecular docking and 3D-QSAR CoMFA studies on indole inhibitors of GIIA secreted phospholipase A(2).
Mouchlis VD; Mavromoustakos TM; Kokotos G
J Chem Inf Model; 2010 Sep; 50(9):1589-601. PubMed ID: 20795712
[TBL] [Abstract][Full Text] [Related]
6. A novel approach to the design of inhibitors of human secreted phospholipase A2 based on native peptide inhibition.
Church WB; Inglis AS; Tseng A; Duell R; Lei PW; Bryant KJ; Scott KF
J Biol Chem; 2001 Aug; 276(35):33156-64. PubMed ID: 11427527
[TBL] [Abstract][Full Text] [Related]
7. Inhibition of secreted phospholipases A₂ by 2-oxoamides based on α-amino acids: Synthesis, in vitro evaluation and molecular docking calculations.
Mouchlis VD; Magrioti V; Barbayianni E; Cermak N; Oslund RC; Mavromoustakos TM; Gelb MH; Kokotos G
Bioorg Med Chem; 2011 Jan; 19(2):735-43. PubMed ID: 21216150
[TBL] [Abstract][Full Text] [Related]
8. Phospholipase A2 superfamily members play divergent roles after spinal cord injury.
López-Vales R; Ghasemlou N; Redensek A; Kerr BJ; Barbayianni E; Antonopoulou G; Baskakis C; Rathore KI; Constantinou-Kokotou V; Stephens D; Shimizu T; Dennis EA; Kokotos G; David S
FASEB J; 2011 Dec; 25(12):4240-52. PubMed ID: 21868473
[TBL] [Abstract][Full Text] [Related]
9. Reductions of phospholipase A(2) inhibition of pulmonary surfactant with hyaluronan.
Iwanicki JL; Lu KW; Taeusch HW
Exp Lung Res; 2010 Apr; 36(3):167-74. PubMed ID: 20334607
[TBL] [Abstract][Full Text] [Related]
10. Selective inhibition of human group IIA-secreted phospholipase A2 (hGIIA) signaling reveals arachidonic acid metabolism is associated with colocalization of hGIIA to vimentin in rheumatoid synoviocytes.
Lee LK; Bryant KJ; Bouveret R; Lei PW; Duff AP; Harrop SJ; Huang EP; Harvey RP; Gelb MH; Gray PP; Curmi PM; Cunningham AM; Church WB; Scott KF
J Biol Chem; 2013 May; 288(21):15269-79. PubMed ID: 23482564
[TBL] [Abstract][Full Text] [Related]
11. Molecular dynamics simulations reveal structural insights into inhibitor binding modes and functionality in human Group IIA phospholipase A
Kim RR; Malde AK; Nematollahi A; Scott KF; Church WB
Proteins; 2017 May; 85(5):827-842. PubMed ID: 28056488
[TBL] [Abstract][Full Text] [Related]
12. Blockade of human group X secreted phospholipase A2 (GX-sPLA2)-induced airway inflammation and hyperresponsiveness in a mouse asthma model by a selective GX-sPLA2 inhibitor.
Henderson WR; Oslund RC; Bollinger JG; Ye X; Tien YT; Xue J; Gelb MH
J Biol Chem; 2011 Aug; 286(32):28049-55. PubMed ID: 21652694
[TBL] [Abstract][Full Text] [Related]
13. On the binding preference of human groups IIA and X phospholipases A2 for membranes with anionic phospholipids.
Bezzine S; Bollinger JG; Singer AG; Veatch SL; Keller SL; Gelb MH
J Biol Chem; 2002 Dec; 277(50):48523-34. PubMed ID: 12244093
[TBL] [Abstract][Full Text] [Related]
14. Basic residues of human group IIA phospholipase A2 are important for binding to factor Xa and prothrombinase inhibition comparison with other mammalian secreted phospholipases A2.
Mounier CM; Luchetta P; Lecut C; Koduri RS; Faure G; Lambeau G; Valentin E; Singer A; Ghomashchi F; Béguin S; Gelb MH; Bon C
Eur J Biochem; 2000 Aug; 267(16):4960-9. PubMed ID: 10931177
[TBL] [Abstract][Full Text] [Related]
15. Group IIA secreted phospholipase A
Giresha AS; Urs D; Manjunatha JG; Sophiya P; Supreetha BH; Jayarama S; Dharmappa KK
Sci Rep; 2022 May; 12(1):7649. PubMed ID: 35538123
[TBL] [Abstract][Full Text] [Related]
16. Design of new potent and selective secretory phospholipase A2 inhibitors. Part 5: synthesis and biological activity of 1-alkyl-4-[4,5-dihydro-1,2,4-[4H]-oxadiazol-5-one-3-ylmethylbenz-4'-yl(oyl)] piperazines.
Boukli L; Touaibia M; Meddad-Belhabich N; Djimdé A; Park CH; Kim JJ; Yoon JH; Lamouri A; Heymans F
Bioorg Med Chem; 2008 Feb; 16(3):1242-53. PubMed ID: 17993277
[TBL] [Abstract][Full Text] [Related]
17. Effect of NGF on the subcellular localization of group IIA secretory phospholipase A(2) (GIIA) in PC12 cells: role in neuritogenesis.
Ferrini M; Nardicchi V; Mannucci R; Arcuri C; Nicoletti I; Donato R; Goracci G
Neurochem Res; 2010 Dec; 35(12):2168-74. PubMed ID: 21125328
[TBL] [Abstract][Full Text] [Related]
18. Structural and Functional Aspects of Targeting the Secreted Human Group IIA Phospholipase A
Kim RR; Chen Z; Mann TJ; Bastard K; F Scott K; Church WB
Molecules; 2020 Sep; 25(19):. PubMed ID: 32998383
[TBL] [Abstract][Full Text] [Related]
19. Development of a potent 2-oxoamide inhibitor of secreted phospholipase A2 guided by molecular docking calculations and molecular dynamics simulations.
Vasilakaki S; Barbayianni E; Leonis G; Papadopoulos MG; Mavromoustakos T; Gelb MH; Kokotos G
Bioorg Med Chem; 2016 Apr; 24(8):1683-95. PubMed ID: 26970660
[TBL] [Abstract][Full Text] [Related]
20. Unusual mode of binding of human group IIA secreted phospholipase A2 to anionic interfaces as studied by continuous wave and time domain electron paramagnetic resonance spectroscopy.
Canaan S; Nielsen R; Ghomashchi F; Robinson BH; Gelb MH
J Biol Chem; 2002 Aug; 277(34):30984-90. PubMed ID: 12039961
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]