These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.


BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

334 related articles for article (PubMed ID: 23122522)

  • 1. Discovery of di-indolinone as a novel scaffold for protein tyrosine phosphatase 1B inhibitors.
    Dai HL; Gao LX; Yang Y; Li JY; Cheng JG; Li J; Wen R; Peng YQ; Zheng JB
    Bioorg Med Chem Lett; 2012 Dec; 22(24):7440-3. PubMed ID: 23122522
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Discovery of Bisindole as a Novel Scaffold for Protein Tyrosine Phosphatase 1B Inhibitors.
    Jing C; Li Z; Jia K; Chen C; Liu X; Wang B; Hu W; Li J; Zhu T; Dong S
    Arch Pharm (Weinheim); 2017 Jan; 350(1):. PubMed ID: 28029177
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Synthesis and biological evaluation of 2,4,6-trihydroxychalcone derivatives as novel protein tyrosine phosphatase 1B inhibitors.
    Sun LP; Gao LX; Ma WP; Nan FJ; Li J; Piao HR
    Chem Biol Drug Des; 2012 Oct; 80(4):584-90. PubMed ID: 22805439
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Pyrrolo[2,3-c]azepine derivatives: a new class of potent protein tyrosine phosphatase 1B inhibitors.
    Xie J; Tian J; Su L; Huang M; Zhu X; Ye F; Wan Y
    Bioorg Med Chem Lett; 2011 Jul; 21(14):4306-9. PubMed ID: 21696953
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Synthesis and biological evaluation of heterocyclic ring-substituted maslinic acid derivatives as novel inhibitors of protein tyrosine phosphatase 1B.
    Qiu WW; Shen Q; Yang F; Wang B; Zou H; Li JY; Li J; Tang J
    Bioorg Med Chem Lett; 2009 Dec; 19(23):6618-22. PubMed ID: 19846303
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Synthesis and characterization of 5,7-dihydroxyflavanone derivatives as novel protein tyrosine phosphatase 1B inhibitors.
    Sun LP; Ma WP; Gao LX; Yang LL; Quan YC; Li J; Piao HR
    J Enzyme Inhib Med Chem; 2013 Dec; 28(6):1199-204. PubMed ID: 23009604
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Preparation of triazole-linked glycosylated α-ketocarboxylic acid derivatives as new PTP1B inhibitors.
    Song Z; He XP; Li C; Gao LX; Wang ZX; Tang Y; Xie J; Li J; Chen GR
    Carbohydr Res; 2011 Jan; 346(1):140-5. PubMed ID: 21111404
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Discovery of potent, selective and orally bioavailable triaryl-sulfonamide based PTP1B inhibitors.
    Patel D; Jain M; Shah SR; Bahekar R; Jadav P; Joharapurkar A; Dhanesha N; Shaikh M; Sairam KV; Kapadnis P
    Bioorg Med Chem Lett; 2012 Jan; 22(2):1111-7. PubMed ID: 22189136
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Design, synthesis and docking study of 5-(substituted benzylidene)thiazolidine-2,4-dione derivatives as inhibitors of protein tyrosine phosphatase 1B.
    Wang Z; Liu Z; Lee W; Kim SN; Yoon G; Cheon SH
    Bioorg Med Chem Lett; 2014 Aug; 24(15):3337-40. PubMed ID: 24953600
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Discovery of novel bromophenol 3,4-dibromo-5-(2-bromo-3,4-dihydroxy-6-(isobutoxymethyl)benzyl)benzene-1,2-diol as protein tyrosine phosphatase 1B inhibitor and its anti-diabetic properties in C57BL/KsJ-db/db mice.
    Jiang B; Guo S; Shi D; Guo C; Wang T
    Eur J Med Chem; 2013 Jun; 64():129-36. PubMed ID: 23644196
    [TBL] [Abstract][Full Text] [Related]  

  • 11. [Design, synthesis and evaluation of malonic acid-based PTP1B inhibitors].
    Du X; Zhang SE; Liu JZ; Nie FL; Ye F; Tian JY; Xiao ZY
    Yao Xue Xue Bao; 2012 Mar; 47(3):367-73. PubMed ID: 22645761
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Discovery of novel high potent and cellular active ADC type PTP1B inhibitors with selectivity over TC-PTP via modification interacting with C site.
    Du Y; Zhang Y; Ling H; Li Q; Shen J
    Eur J Med Chem; 2018 Jan; 144():692-700. PubMed ID: 29289892
    [TBL] [Abstract][Full Text] [Related]  

  • 13. PTP1B inhibitors: synthesis and evaluation of difluoro-methylenephosphonate bioisosteres on a sulfonamide scaffold.
    Holmes CP; Li X; Pan Y; Xu C; Bhandari A; Moody CM; Miguel JA; Ferla SW; De Francisco MN; Frederick BT; Zhou S; Macher N; Jang L; Irvine JD; Grove JR
    Bioorg Med Chem Lett; 2008 Apr; 18(8):2719-24. PubMed ID: 18372175
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Design, synthesis, and biological evaluation of bromophenol derivatives as protein tyrosine phosphatase 1B inhibitors.
    Jiang B; Shi D; Cui Y; Guo S
    Arch Pharm (Weinheim); 2012 Jun; 345(6):444-53. PubMed ID: 22307562
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Novel thiophene derivatives as PTP1B inhibitors with selectivity and cellular activity.
    Ye D; Zhang Y; Wang F; Zheng M; Zhang X; Luo X; Shen X; Jiang H; Liu H
    Bioorg Med Chem; 2010 Mar; 18(5):1773-82. PubMed ID: 20153651
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Design, synthesis, and biological evaluation of novel 2-ethyl-5-phenylthiazole-4-carboxamide derivatives as protein tyrosine phosphatase 1B inhibitors with improved cellular efficacy.
    Chen YT; Tang CL; Ma WP; Gao LX; Wei Y; Zhang W; Li JY; Li J; Nan FJ
    Eur J Med Chem; 2013 Nov; 69():399-412. PubMed ID: 24090912
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Discovery of core-structurally novel PTP1B inhibitors with specific selectivity containing oxindole-fused spirotetrahydrofurochroman by one-pot reaction.
    Dong S; Lei Y; Jia S; Gao L; Li J; Zhu T; Liu S; Hu W
    Bioorg Med Chem Lett; 2017 Feb; 27(4):1105-1108. PubMed ID: 28111140
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Synthesis and biological evaluation of novel bis-aromatic amides as novel PTP1B inhibitors.
    Wang WL; Huang C; Gao LX; Tang CL; Wang JQ; Wu MC; Sheng L; Chen HJ; Nan FJ; Li JY; Li J; Feng B
    Bioorg Med Chem Lett; 2014 Apr; 24(8):1889-94. PubMed ID: 24684845
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Synthesis and biological evaluation of 4,4-dimethyl lithocholic acid derivatives as novel inhibitors of protein tyrosine phosphatase 1B.
    He HB; Gao LX; Deng QF; Ma WP; Tang CL; Qiu WW; Tang J; Li JY; Li J; Yang F
    Bioorg Med Chem Lett; 2012 Dec; 22(23):7237-42. PubMed ID: 23067554
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Design, synthesis and molecular modelling studies of novel 3-acetamido-4-methyl benzoic acid derivatives as inhibitors of protein tyrosine phosphatase 1B.
    Rakse M; Karthikeyan C; Deora GS; Moorthy NS; Rathore V; Rawat AK; Srivastava AK; Trivedi P
    Eur J Med Chem; 2013; 70():469-76. PubMed ID: 24185377
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 17.