These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.


BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

110 related articles for article (PubMed ID: 23286196)

  • 1. Discovery of 5-benzyl-3-phenyl-4,5-dihydroisoxazoles and 5-benzyl-3-phenyl-1,4,2-dioxazoles as potent firefly luciferase inhibitors.
    Poutiainen PK; Palvimo JJ; Hinkkanen AE; Valkonen A; Väisänen TK; Laatikainen R; Pulkkinen JT
    J Med Chem; 2013 Feb; 56(3):1064-73. PubMed ID: 23286196
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Reporter enzyme inhibitor study to aid assembly of orthogonal reporter gene assays.
    Ho PI; Yue K; Pandey P; Breault L; Harbinski F; McBride AJ; Webb B; Narahari J; Karassina N; Wood KV; Hill A; Auld DS
    ACS Chem Biol; 2013 May; 8(5):1009-17. PubMed ID: 23485150
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Characterization of chemical libraries for luciferase inhibitory activity.
    Auld DS; Southall NT; Jadhav A; Johnson RL; Diller DJ; Simeonov A; Austin CP; Inglese J
    J Med Chem; 2008 Apr; 51(8):2372-86. PubMed ID: 18363348
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Identification and synthesis of substituted pyrrolo[2,3-d]pyrimidines as novel firefly luciferase inhibitors.
    Liu Y; Fang J; Cai H; Xiao F; Ding K; Hu Y
    Bioorg Med Chem; 2012 Sep; 20(18):5473-82. PubMed ID: 22898255
    [TBL] [Abstract][Full Text] [Related]  

  • 5. False positives in a reporter gene assay: identification and synthesis of substituted N-pyridin-2-ylbenzamides as competitive inhibitors of firefly luciferase.
    Heitman LH; van Veldhoven JP; Zweemer AM; Ye K; Brussee J; IJzerman AP
    J Med Chem; 2008 Aug; 51(15):4724-9. PubMed ID: 18646744
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Pyrrolo[2,3-b]quinoxalines as inhibitors of firefly luciferase: their Cu-mediated synthesis and evaluation as false positives in a reporter gene assay.
    Nakhi A; Rahman MS; Kishore R; Meda CL; Deora GS; Parsa KV; Pal M
    Bioorg Med Chem Lett; 2012 Oct; 22(20):6433-41. PubMed ID: 22981335
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Mechanism of PTC124 activity in cell-based luciferase assays of nonsense codon suppression.
    Auld DS; Thorne N; Maguire WF; Inglese J
    Proc Natl Acad Sci U S A; 2009 Mar; 106(9):3585-90. PubMed ID: 19208811
    [TBL] [Abstract][Full Text] [Related]  

  • 8. The nuclear factor κB inhibitor (E)-2-fluoro-4'-methoxystilbene inhibits firefly luciferase.
    Braeuning A; Vetter S
    Biosci Rep; 2012 Dec; 32(6):531-7. PubMed ID: 22789175
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Inhibiting Firefly Bioluminescence by Chalcones.
    Zhang H; Su J; Lin Y; Bai H; Liu J; Chen H; Du L; Gu L; Li M
    Anal Chem; 2017 Jun; 89(11):6099-6105. PubMed ID: 28492074
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Characterisation of utrophin modulator SMT C1100 as a non-competitive inhibitor of firefly luciferase.
    Wilkinson IVL; Reynolds JK; Galan SRG; Vuorinen A; Sills AJ; Pires E; Wynne GM; Wilson FX; Russell AJ
    Bioorg Chem; 2020 Jan; 94():103395. PubMed ID: 31733898
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Kinetics of inhibition of firefly luciferase by oxyluciferin and dehydroluciferyl-adenylate.
    Ribeiro C; Esteves da Silva JC
    Photochem Photobiol Sci; 2008 Sep; 7(9):1085-90. PubMed ID: 18754056
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Design, synthesis and biological evaluation of heterocyclic azoles derivatives containing pyrazine moiety as potential telomerase inhibitors.
    Zhang YB; Wang XL; Liu W; Yang YS; Tang JF; Zhu HL
    Bioorg Med Chem; 2012 Nov; 20(21):6356-65. PubMed ID: 23018096
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Firefly luciferase in chemical biology: a compendium of inhibitors, mechanistic evaluation of chemotypes, and suggested use as a reporter.
    Thorne N; Shen M; Lea WA; Simeonov A; Lovell S; Auld DS; Inglese J
    Chem Biol; 2012 Aug; 19(8):1060-72. PubMed ID: 22921073
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Firefly luciferase inhibition.
    Leitão JM; Esteves da Silva JC
    J Photochem Photobiol B; 2010 Oct; 101(1):1-8. PubMed ID: 20655239
    [TBL] [Abstract][Full Text] [Related]  

  • 15. A basis for reduced chemical library inhibition of firefly luciferase obtained from directed evolution.
    Auld DS; Zhang YQ; Southall NT; Rai G; Landsman M; MacLure J; Langevin D; Thomas CJ; Austin CP; Inglese J
    J Med Chem; 2009 Mar; 52(5):1450-8. PubMed ID: 19215089
    [TBL] [Abstract][Full Text] [Related]  

  • 16. A real-time bioluminescent HTS method for measuring protein kinase activity influenced neither by ATP concentration nor by luciferase inhibition.
    Lundin A; Eriksson J
    Assay Drug Dev Technol; 2008 Aug; 6(4):531-41. PubMed ID: 18532902
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Novel, potent, selective, and metabolically stable stearoyl-CoA desaturase (SCD) inhibitors.
    Koltun DO; Parkhill EQ; Vasilevich NI; Glushkov AI; Zilbershtein TM; Ivanov AV; Cole AG; Henderson I; Zautke NA; Brunn SA; Mollova N; Leung K; Chisholm JW; Zablocki J
    Bioorg Med Chem Lett; 2009 Apr; 19(7):2048-52. PubMed ID: 19249203
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Inhibitory effect of lipoic acid on firefly luciferase bioluminescence.
    Niwa K; Ohmiya Y
    Biochem Biophys Res Commun; 2004 Oct; 323(2):625-9. PubMed ID: 15369796
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Structure-based virtual screening approach to the discovery of phosphoinositide 3-kinase alpha inhibitors.
    Park H; Choi H; Hong S; Kim D; Oh DS; Hong S
    Bioorg Med Chem Lett; 2011 Apr; 21(7):2021-4. PubMed ID: 21354792
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Discovery of (1S,2R,3R)-2,3-dimethyl-2-phenyl-1-sulfamidocyclopropanecarboxylates: novel and highly selective aggrecanase inhibitors.
    Shiozaki M; Maeda K; Miura T; Kotoku M; Yamasaki T; Matsuda I; Aoki K; Yasue K; Imai H; Ubukata M; Suma A; Yokota M; Hotta T; Tanaka M; Hase Y; Haas J; Fryer AM; Laird ER; Littmann NM; Andrews SW; Josey JA; Mimura T; Shinozaki Y; Yoshiuchi H; Inaba T
    J Med Chem; 2011 Apr; 54(8):2839-63. PubMed ID: 21417219
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 6.