BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

99 related articles for article (PubMed ID: 23320429)

  • 1. Structure-activity relationship studies of argiotoxins: selective and potent inhibitors of ionotropic glutamate receptors.
    Poulsen MH; Lucas S; Bach TB; Barslund AF; Wenzler C; Jensen CB; Kristensen AS; Strømgaard K
    J Med Chem; 2013 Feb; 56(3):1171-81. PubMed ID: 23320429
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Development of potent fluorescent polyamine toxins and application in labeling of ionotropic glutamate receptors in hippocampal neurons.
    Nørager NG; Jensen CB; Rathje M; Andersen J; Madsen KL; Kristensen AS; Strømgaard K
    ACS Chem Biol; 2013 Sep; 8(9):2033-41. PubMed ID: 23838571
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Structure-activity relationship study of spider polyamine toxins as inhibitors of ionotropic glutamate receptors.
    Xiong XF; Poulsen MH; Hussein RA; Nørager NG; Strømgaard K
    ChemMedChem; 2014 Dec; 9(12):2661-70. PubMed ID: 25267300
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Structure-activity relationship studies of N-methylated and N-hydroxylated spider polyamine toxins as inhibitors of ionotropic glutamate receptors.
    Nørager NG; Poulsen MH; Jensen AG; Jeppesen NS; Kristensen AS; Strømgaard K
    J Med Chem; 2014 Jun; 57(11):4940-9. PubMed ID: 24824658
    [TBL] [Abstract][Full Text] [Related]  

  • 5. General synthesis of β-alanine-containing spider polyamine toxins and discovery of nephila polyamine toxins 1 and 8 as highly potent inhibitors of ionotropic glutamate receptors.
    Lucas S; Poulsen MH; Nørager NG; Barslund AF; Bach TB; Kristensen AS; Strømgaard K
    J Med Chem; 2012 Nov; 55(22):10297-301. PubMed ID: 23092360
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Solid-phase synthesis and biological evaluation of Joro spider toxin-4 from Nephila clavata.
    Barslund AF; Poulsen MH; Bach TB; Lucas S; Kristensen AS; Strømgaard K
    J Nat Prod; 2011 Mar; 74(3):483-6. PubMed ID: 21188966
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Synthesis and biological activity of argiotoxin 636 and analogues: selective antagonists for ionotropic glutamate receptors.
    Nelson JK; Frølund SU; Tikhonov DB; Kristensen AS; Strømgaard K
    Angew Chem Int Ed Engl; 2009; 48(17):3087-91. PubMed ID: 19152392
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Design and synthesis of labeled analogs of PhTX-56, a potent and selective AMPA receptor antagonist.
    Andersen TF; Vogensen SB; Jensen LS; Knapp KM; Strømgaard K
    Bioorg Med Chem; 2005 Sep; 13(17):5104-12. PubMed ID: 15990320
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Binding of ArgTX-636 in the NMDA receptor ion channel.
    Poulsen MH; Andersen J; Christensen R; Hansen KB; Traynelis SF; Strømgaard K; Kristensen AS
    J Mol Biol; 2015 Jan; 427(1):176-89. PubMed ID: 24862283
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Polyamine toxins: development of selective ligands for ionotropic receptors.
    Strømgaard K; Jensen LS; Vogensen SB
    Toxicon; 2005 Mar; 45(3):249-54. PubMed ID: 15683862
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Selective antagonism of native and cloned kainate and NMDA receptors by polyamine-containing toxins.
    Brackley PT; Bell DR; Choi SK; Nakanishi K; Usherwood PN
    J Pharmacol Exp Ther; 1993 Sep; 266(3):1573-80. PubMed ID: 7690404
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Design, synthesis, and pharmacological characterization of polyamine toxin derivatives: potent ligands for the pore-forming region of AMPA receptors.
    Jensen LS; Bølcho U; Egebjerg J; Strømgaard K
    ChemMedChem; 2006 Apr; 1(4):419-28. PubMed ID: 16892377
    [TBL] [Abstract][Full Text] [Related]  

  • 13. ArgTX-636, a polyamine isolated from spider venom: A novel class of melanogenesis inhibitors.
    Verdoni M; Roudaut H; De Pomyers H; Gigmes D; Bertin D; Luis J; Bengeloune AH; Mabrouk K
    Bioorg Med Chem; 2016 Nov; 24(22):5685-5692. PubMed ID: 27647371
    [TBL] [Abstract][Full Text] [Related]  

  • 14. AMPA receptor ligands: synthetic and pharmacological studies of polyamines and polyamine toxins.
    Strømgaard K; Mellor I
    Med Res Rev; 2004 Sep; 24(5):589-620. PubMed ID: 15224382
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Assessment of structurally diverse philanthotoxin analogues for inhibitory activity on ionotropic glutamate receptor subtypes: discovery of nanomolar, nonselective, and use-dependent antagonists.
    Frølund S; Bella A; Kristensen AS; Ziegler HL; Witt M; Olsen CA; Strømgaard K; Franzyk H; Jaroszewski JW
    J Med Chem; 2010 Oct; 53(20):7441-51. PubMed ID: 20873775
    [TBL] [Abstract][Full Text] [Related]  

  • 16. [Glutamate receptor antagonists from the spider Argiope lobata venom].
    Grishin EV; Volkova TM; Arsen'ev AS
    Bioorg Khim; 1988 Jul; 14(7):883-92. PubMed ID: 2847758
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Pharmacological characterization of (4R)-alkyl glutamate analogues at the ionotropic glutamate receptors--focus on subtypes iGlu(5-7).
    Bunch L; Gefflaut T; Alaux S; Sagot E; Nielsen B; Pickering DS
    Eur J Pharmacol; 2009 May; 609(1-3):1-4. PubMed ID: 19285062
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Rational design, synthesis and pharmacological evaluation of the (2R)- and (2S)-stereoisomers of 3-(2-carboxypyrrolidinyl)-2-methyl acetic acid as ligands for the ionotropic glutamate receptors.
    Rasmussen JL; Storgaard M; Pickering DS; Bunch L
    ChemMedChem; 2011 Mar; 6(3):498-504. PubMed ID: 21268287
    [TBL] [Abstract][Full Text] [Related]  

  • 19. 5-(N-oxyaza)-7-substituted-1,4-dihydroquinoxaline-2,3-diones: novel, systemically active and broad spectrum antagonists for NMDA/glycine, AMPA, and kainate receptors.
    Cai SX; Huang JC; Espitia SA; Tran M; Ilyin VI; Hawkinson JE; Woodward RM; Weber E; Keana JF
    J Med Chem; 1997 Oct; 40(22):3679-86. PubMed ID: 9357535
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Synthesis of new isoxazoline-based acidic amino acids and investigation of their affinity and selectivity profile at ionotropic glutamate receptors.
    Pinto A; Conti P; Grazioso G; Tamborini L; Madsen U; Nielsen B; De Micheli C
    Eur J Med Chem; 2011 Feb; 46(2):787-93. PubMed ID: 21220180
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 5.