126 related articles for article (PubMed ID: 2353556)
1. Selective aromatase inhibition by pyridoglutethimide, an analogue of aminoglutethimide.
Kitawaki J; Yamamoto T; Urabe M; Tamura T; Inoue S; Honjo H; Okada H
Acta Endocrinol (Copenh); 1990 May; 122(5):592-8. PubMed ID: 2353556
[TBL] [Abstract][Full Text] [Related]
2. Effect of aromatase inhibitors on estrogen 2-hydroxylase in rat liver.
Purba HS; King EJ; Richert P; Bhatnagar AS
J Steroid Biochem Mol Biol; 1994 Feb; 48(2-3):215-9. PubMed ID: 8142297
[TBL] [Abstract][Full Text] [Related]
3. Pyridoglutethimide [3-ethyl-3-(4-pyridyl)-piperidine-2,6-dione], an analogue of aminoglutethimide. Metabolism and pharmacokinetics.
Seago A; Goss PE; Griggs LJ; Jarman M
Biochem Pharmacol; 1986 Sep; 35(17):2911-6. PubMed ID: 3741481
[TBL] [Abstract][Full Text] [Related]
4. Analogues of aminoglutethimide based on 1-phenyl-3-azabicyclo[3.1.0]hexane-2,4-dione: selective inhibition of aromatase activity.
Rowlands MG; Bunnett MA; Foster AB; Jarman M; Stanek J; Schweizer E
J Med Chem; 1988 May; 31(5):971-6. PubMed ID: 3361583
[TBL] [Abstract][Full Text] [Related]
5. Analogues of aminoglutethimide: selective inhibition of aromatase.
Foster AB; Jarman M; Leung CS; Rowlands MG; Taylor GN; Plevey RG; Sampson P
J Med Chem; 1985 Feb; 28(2):200-4. PubMed ID: 3968684
[TBL] [Abstract][Full Text] [Related]
6. The effect of the aromatase inhibitor, rogletimide (pyridoglutethimide), on guinea pig adrenal cell steroidogenesis and placental microsomal aromatase activity: comparison with aminoglutethimide and CGS 16949A.
Newton CJ; Mehta A; Dowsett M
J Steroid Biochem Mol Biol; 1991 Nov; 39(5A):723-7. PubMed ID: 1659868
[TBL] [Abstract][Full Text] [Related]
7. Analogues of 3-ethyl-3-(4-pyridyl)piperidine-2,6-dione as selective inhibitors of aromatase: derivatives with variable 1-alkyl and 3-alkyl substituents.
Leung CS; Rowlands MG; Jarman M; Foster AB; Griggs LJ; Wilman DE
J Med Chem; 1987 Sep; 30(9):1550-4. PubMed ID: 3625703
[TBL] [Abstract][Full Text] [Related]
8. Metabolism and pharmacokinetics of the N- and C-n-octyl analogues of pyridoglutethimide [3-ethyl-3-(4-pyridyl)piperidine-2,6-dione]: novel inhibitors of aromatase.
Seago A; Baker MH; Houghton J; Leung CS; Jarman M
Biochem Pharmacol; 1987 Feb; 36(4):573-7. PubMed ID: 3827945
[No Abstract] [Full Text] [Related]
9. Inhibition of estrogen synthetase (aromatase) by 4-cyclohexylaniline.
Kellis JT; Vickery LE
Endocrinology; 1984 Jun; 114(6):2128-37. PubMed ID: 6723577
[TBL] [Abstract][Full Text] [Related]
10. Synthesis and biochemical evaluation of analogues of aminoglutethimide based on phenylpyrrolidine-2,5-dione.
Daly MJ; Jones GW; Nicholls PJ; Smith HJ; Rowlands MG; Bunnett MA
J Med Chem; 1986 Apr; 29(4):520-3. PubMed ID: 3754286
[TBL] [Abstract][Full Text] [Related]
11. Pharmacology of aminoglutethimide: structure/activity relationships and receptor interactions.
Nicholls PJ; Daly MJ; Smith HJ
Breast Cancer Res Treat; 1986; 7 Suppl():S55-67. PubMed ID: 3755630
[TBL] [Abstract][Full Text] [Related]
12. Analogues of aminoglutethimide: selective inhibition of cholesterol side-chain cleavage.
Foster AB; Jarman M; Leung CS; Rowlands MG; Taylor GN
J Med Chem; 1983 Jan; 26(1):50-4. PubMed ID: 6827528
[TBL] [Abstract][Full Text] [Related]
13. Evaluation of the racemate and the enantiomers of a new highly active and selective aromatase inhibitor of the aminoglutethimide type.
Hartmann RW; GrĂ¼n G; Bartz U; Palzer M
J Steroid Biochem Mol Biol; 1992 Dec; 43(7):641-8. PubMed ID: 1472456
[TBL] [Abstract][Full Text] [Related]
14. 1-Alkyl analogues of aminoglutethimide. Comparative inhibition of cholesterol side chain cleavage and aromatase and metabolism of the 1-propyl derivative, a highly selective inhibitor of aromatase.
Seago A; Baker MH; Houghton J; Jarman M; Leung CS; Rowlands MG
Biochem Pharmacol; 1988 Jun; 37(11):2167-72. PubMed ID: 3377817
[TBL] [Abstract][Full Text] [Related]
15. Selective inhibition of cholesterol side-chain cleavage by potential pro-drug forms of aminoglutethimide.
Jarman M; Barrie SE; Leung CS; Rowlands MG
Anticancer Drug Des; 1988 Dec; 3(3):185-90. PubMed ID: 3264700
[TBL] [Abstract][Full Text] [Related]
16. Synthesis and aromatase inhibition of 3-cycloalkyl-substituted 3-(4-aminophenyl)piperidine-2,6-diones.
Hartmann RW; Batzl C; Pongratz TM; Mannschreck A
J Med Chem; 1992 Jun; 35(12):2210-4. PubMed ID: 1613747
[TBL] [Abstract][Full Text] [Related]
17. [The inhibitory effect of miconazole on aromatase activity for androstenedione in human placental and ovarian preparations].
Yamamoto T; Urabe M; Okada H
Nihon Naibunpi Gakkai Zasshi; 1987 Nov; 63(11):1379-85. PubMed ID: 3443212
[TBL] [Abstract][Full Text] [Related]
18. Antitumor effect of pyridoglutethimide, an aromatase inhibitor, on 7,12-dimethylbenz(a)anthracene-induced mammary tumors of rat.
Yamamoto T; Urabe M; Tamura T; Kitawaki J; Honjo H; Okada H
Anticancer Res; 1991; 11(6):1999-2002. PubMed ID: 1776832
[TBL] [Abstract][Full Text] [Related]
19. Aromatase inhibitors--mechanisms for non-steroidal inhibitors.
Vanden Bossche HV; Moereels H; Koymans LM
Breast Cancer Res Treat; 1994; 30(1):43-55. PubMed ID: 7949204
[TBL] [Abstract][Full Text] [Related]
20. Endocrine, pharmacokinetic and clinical studies of the aromatase inhibitor 3-ethyl-3-(4-pyridyl)piperidine-2,6-dione ('pyridoglutethimide') in postmenopausal breast cancer patients.
Dowsett M; MacNeill F; Mehta A; Newton C; Haynes B; Jones A; Jarman M; Lonning P; Powles TJ; Coombes RC
Br J Cancer; 1991 Nov; 64(5):887-94. PubMed ID: 1931611
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]