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4. Synthesis of peptidyl fluoromethyl ketones and peptidyl alpha-keto esters as inhibitors of porcine pancreatic elastase, human neutrophil elastase, and rat and human neutrophil cathepsin G. Peet NP; Burkhart JP; Angelastro MR; Giroux EL; Mehdi S; Bey P; Kolb M; Neises B; Schirlin D J Med Chem; 1990 Jan; 33(1):394-407. PubMed ID: 2296031 [TBL] [Abstract][Full Text] [Related]
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6. Mechanism of slow-binding inhibition of human leukocyte elastase by trifluoromethyl ketones. Stein RL; Strimpler AM; Edwards PD; Lewis JJ; Mauger RC; Schwartz JA; Stein MM; Trainor DA; Wildonger RA; Zottola MA Biochemistry; 1987 May; 26(10):2682-9. PubMed ID: 3649251 [TBL] [Abstract][Full Text] [Related]
7. Reversible, slow, tight-binding inhibition of human leukocyte elastase. Dunlap RP; Stone PJ; Abeles RH Biochem Biophys Res Commun; 1987 May; 145(1):509-13. PubMed ID: 3647764 [TBL] [Abstract][Full Text] [Related]
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10. Proline-valine pseudo peptide enol lactones. Effective and selective inhibitors of chymotrypsin and human leukocyte elastase. Reed PE; Katzenellenbogen JA J Biol Chem; 1991 Jan; 266(1):13-21. PubMed ID: 1985887 [TBL] [Abstract][Full Text] [Related]
11. The kinetic mechanism of inhibition of human leukocyte elastase by MR889, a new cyclic thiolic compound. Baici A; Pelloso R; Hörler D Biochem Pharmacol; 1990 Mar; 39(5):919-24. PubMed ID: 2310417 [TBL] [Abstract][Full Text] [Related]
12. Inhibition of the serine proteases leukocyte elastase, pancreatic elastase, cathepsin G, and chymotrypsin by peptide boronic acids. Kettner CA; Shenvi AB J Biol Chem; 1984 Dec; 259(24):15106-14. PubMed ID: 6392293 [TBL] [Abstract][Full Text] [Related]
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17. Inhibition of human leukocyte elastase by N-substituted tripeptide trifluoromethyl ketones. Skiles JW; Fuchs V; Chow G; Skoog M Res Commun Chem Pathol Pharmacol; 1990 Jun; 68(3):365-74. PubMed ID: 2385759 [TBL] [Abstract][Full Text] [Related]
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19. The inhibition of human neutrophil elastase and cathepsin G by peptidyl 1,2-dicarbonyl derivatives. Mehdi S; Angelastro MR; Burkhart JP; Koehl JR; Peet NP; Bey P Biochem Biophys Res Commun; 1990 Jan; 166(2):595-600. PubMed ID: 2302225 [TBL] [Abstract][Full Text] [Related]
20. Irreversible inhibition of serine proteases by peptidyl derivatives of alpha-aminoalkylphosphonate diphenyl esters. Oleksyszyn J; Powers JC Biochem Biophys Res Commun; 1989 May; 161(1):143-9. PubMed ID: 2730652 [TBL] [Abstract][Full Text] [Related] [Next] [New Search]