BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

87 related articles for article (PubMed ID: 23551102)

  • 1. Phosphoinositide 3-kinase gamma in T cell biology and disease therapy.
    Fung-Leung WP
    Ann N Y Acad Sci; 2013 Mar; 1280():40-3. PubMed ID: 23551102
    [TBL] [Abstract][Full Text] [Related]  

  • 2. PI3Kδ and PI3Kγ as targets for autoimmune and inflammatory diseases.
    Cushing TD; Metz DP; Whittington DA; McGee LR
    J Med Chem; 2012 Oct; 55(20):8559-81. PubMed ID: 22924688
    [No Abstract]   [Full Text] [Related]  

  • 3. PI3Kδ and PI3Kγ isoforms have distinct functions in regulating pro-tumoural signalling in the multiple myeloma microenvironment.
    Piddock RE; Loughran N; Marlein CR; Robinson SD; Edwards DR; Yu S; Pillinger GE; Zhou Z; Zaitseva L; Auger MJ; Rushworth SA; Bowles KM
    Blood Cancer J; 2017 Mar; 7(3):e539. PubMed ID: 28282033
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Inhibition of phosphoinositide 3-kinase γ attenuates inflammation, obesity, and cardiovascular risk factors.
    Wymann MP; Solinas G
    Ann N Y Acad Sci; 2013 Mar; 1280():44-7. PubMed ID: 23551103
    [TBL] [Abstract][Full Text] [Related]  

  • 5. The absence of functional PI3Kgamma prevents leukocyte recruitment and ameliorates DSS-induced colitis in mice.
    van Dop WA; Marengo S; te Velde AA; Ciraolo E; Franco I; ten Kate FJ; Boeckxstaens GE; Hardwick JC; Hommes DW; Hirsch E; van den Brink GR
    Immunol Lett; 2010 Jun; 131(1):33-9. PubMed ID: 20347874
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Phosphoinositide 3-kinase γ mediates microglial phagocytosis via lipid kinase-independent control of cAMP.
    Schmidt C; Schneble N; Müller JP; Bauer R; Perino A; Marone R; Rybalkin SD; Wymann MP; Hirsch E; Wetzker R
    Neuroscience; 2013 Mar; 233():44-53. PubMed ID: 23276671
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Phosphoinositide 3-kinase gamma controls inflammation-induced myocardial depression via sequential cAMP and iNOS signalling.
    Ndongson-Dongmo B; Heller R; Hoyer D; Brodhun M; Bauer M; Winning J; Hirsch E; Wetzker R; Schlattmann P; Bauer R
    Cardiovasc Res; 2015 Nov; 108(2):243-53. PubMed ID: 26334033
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Phosphoinositide 3-kinase γ plays a critical role in bleomycin-induced pulmonary inflammation and fibrosis in mice.
    Russo RC; Garcia CC; Barcelos LS; Rachid MA; Guabiraba R; Roffê E; Souza AL; Sousa LP; Mirolo M; Doni A; Cassali GD; Pinho V; Locati M; Teixeira MM
    J Leukoc Biol; 2011 Feb; 89(2):269-82. PubMed ID: 21048214
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Loss of PI3Kγ enhances cAMP-dependent MMP remodeling of the myocardial N-cadherin adhesion complexes and extracellular matrix in response to early biomechanical stress.
    Guo D; Kassiri Z; Basu R; Chow FL; Kandalam V; Damilano F; Liang W; Izumo S; Hirsch E; Penninger JM; Backx PH; Oudit GY
    Circ Res; 2010 Nov; 107(10):1275-89. PubMed ID: 20847309
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Phosphoinositide-3 kinase gamma activity contributes to sepsis and organ damage by altering neutrophil recruitment.
    Martin EL; Souza DG; Fagundes CT; Amaral FA; Assenzio B; Puntorieri V; Del Sorbo L; Fanelli V; Bosco M; Delsedime L; Pinho JF; Lemos VS; Souto FO; Alves-Filho JC; Cunha FQ; Slutsky AS; Ruckle T; Hirsch E; Teixeira MM; Ranieri VM
    Am J Respir Crit Care Med; 2010 Sep; 182(6):762-73. PubMed ID: 20508212
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Phosphoinositide 3-kinase gamma (PI3Kgamma) inhibitors for the treatment of inflammation and autoimmune disease.
    Venable JD; Ameriks MK; Blevitt JM; Thurmond RL; Fung-Leung WP
    Recent Pat Inflamm Allergy Drug Discov; 2010 Jan; 4(1):1-15. PubMed ID: 20017720
    [TBL] [Abstract][Full Text] [Related]  

  • 12. PI3Kγ kinase activity is required for optimal T-cell activation and differentiation.
    Ladygina N; Gottipati S; Ngo K; Castro G; Ma JY; Banie H; Rao TS; Fung-Leung WP
    Eur J Immunol; 2013 Dec; 43(12):3183-96. PubMed ID: 24030559
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Evolution of PI3Kγ and δ Inhibitors for Inflammatory and Autoimmune Diseases.
    Perry MWD; Abdulai R; Mogemark M; Petersen J; Thomas MJ; Valastro B; Westin Eriksson A
    J Med Chem; 2019 May; 62(10):4783-4814. PubMed ID: 30582813
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Loss of phosphoinositide 3-kinase gamma decreases migration and activation of phagocytes but not T cell activation in antigen-induced arthritis.
    Gruen M; Rose C; König C; Gajda M; Wetzker R; Bräuer R
    BMC Musculoskelet Disord; 2010 Apr; 11():63. PubMed ID: 20374644
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Importance of phosphoinositide 3-kinase gamma in the host defense against pneumococcal infection.
    Maus UA; Backi M; Winter C; Srivastava M; Schwarz MK; Rückle T; Paton JC; Briles D; Mack M; Welte T; Maus R; Bohle RM; Seeger W; Rommel C; Hirsch E; Lohmeyer J; Preissner KT
    Am J Respir Crit Care Med; 2007 May; 175(9):958-66. PubMed ID: 17322108
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Discovery of N-{5-[3-(3-hydroxypiperidin-1-yl)-1,2,4-oxadiazol-5-yl]-4-methyl-1,3-thiazol-2-yl}acetamide (TASP0415914) as an orally potent phosphoinositide 3-kinase γ inhibitor for the treatment of inflammatory diseases.
    Oka Y; Yabuuchi T; Oi T; Kuroda S; Fujii Y; Ohtake H; Inoue T; Wakahara S; Kimura K; Fujita K; Endo M; Taguchi K; Sekiguchi Y
    Bioorg Med Chem; 2013 Dec; 21(24):7578-83. PubMed ID: 24262886
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Ex vivo blockade of PI3K gamma or delta signaling enhances the antitumor potency of adoptively transferred CD8
    Dwyer CJ; Arhontoulis DC; Rangel Rivera GO; Knochelmann HM; Smith AS; Wyatt MM; Rubinstein MP; Atkinson C; Thaxton JE; Neskey DM; Paulos CM
    Eur J Immunol; 2020 Sep; 50(9):1386-1399. PubMed ID: 32383488
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Targeting phosphatidylinositol 3-kinase gamma (PI3Kγ): Discovery and development of its selective inhibitors.
    Zhu J; Li K; Yu L; Chen Y; Cai Y; Jin J; Hou T
    Med Res Rev; 2021 May; 41(3):1599-1621. PubMed ID: 33300614
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Discovery and optimization of a series of 2-aminothiazole-oxazoles as potent phosphoinositide 3-kinase γ inhibitors.
    Oka Y; Yabuuchi T; Fujii Y; Ohtake H; Wakahara S; Matsumoto K; Endo M; Tamura Y; Sekiguchi Y
    Bioorg Med Chem Lett; 2012 Dec; 22(24):7534-8. PubMed ID: 23122859
    [TBL] [Abstract][Full Text] [Related]  

  • 20. SAR studies around a series of triazolopyridines as potent and selective PI3Kγ inhibitors.
    Bell K; Sunose M; Ellard K; Cansfield A; Taylor J; Miller W; Ramsden N; Bergamini G; Neubauer G
    Bioorg Med Chem Lett; 2012 Aug; 22(16):5257-63. PubMed ID: 22819766
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 5.