BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

81 related articles for article (PubMed ID: 23602523)

  • 1. The discovery of colchicine-SAHA hybrids as a new class of antitumor agents.
    Zhang X; Zhang J; Tong L; Luo Y; Su M; Zang Y; Li J; Lu W; Chen Y
    Bioorg Med Chem; 2013 Jun; 21(11):3240-4. PubMed ID: 23602523
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Design, synthesis and mechanistic study of new dual targeting HDAC/tubulin inhibitors.
    El-Zoghbi MS; Bass AK; A Abuo-Rahma GE; Mohamed MF; Badr M; Al-Ghulikah HA; Abdelhafez EM
    Future Med Chem; 2024 Apr; 16(7):601-622. PubMed ID: 38436113
    [No Abstract]   [Full Text] [Related]  

  • 3. Hydroxamic Acids Immobilized on Resins (HAIRs): Synthesis of Dual-Targeting HDAC Inhibitors and HDAC Degraders (PROTACs).
    Sinatra L; Bandolik JJ; Roatsch M; Sönnichsen M; Schoeder CT; Hamacher A; Schöler A; Borkhardt A; Meiler J; Bhatia S; Kassack MU; Hansen FK
    Angew Chem Int Ed Engl; 2020 Dec; 59(50):22494-22499. PubMed ID: 32780485
    [TBL] [Abstract][Full Text] [Related]  

  • 4. First-in-Class Dual Mechanism Ferroptosis-HDAC Inhibitor Hybrids.
    Karaj E; Sindi SH; Kuganesan N; Koranne RA; Knoff JR; James AW; Fu Y; Kotsull LN; Pflum MK; Shah Z; Taylor WR; Tillekeratne LMV
    J Med Chem; 2022 Nov; 65(21):14764-14791. PubMed ID: 36306372
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Bifunctional conjugates with potent inhibitory activity towards cyclooxygenase and histone deacetylase.
    Raji I; Yadudu F; Janeira E; Fathi S; Szymczak L; Kornacki JR; Komatsu K; Li JD; Mrksich M; Oyelere AK
    Bioorg Med Chem; 2017 Feb; 25(3):1202-1218. PubMed ID: 28057407
    [TBL] [Abstract][Full Text] [Related]  

  • 6. A chimeric SERM-histone deacetylase inhibitor approach to breast cancer therapy.
    Patel HK; Siklos MI; Abdelkarim H; Mendonca EL; Vaidya A; Petukhov PA; Thatcher GR
    ChemMedChem; 2014 Mar; 9(3):602-13. PubMed ID: 23956109
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Design, synthesis and evaluation of antiproliferative activity of melanoma-targeted histone deacetylase inhibitors.
    Raji I; Ahluwalia K; Oyelere AK
    Bioorg Med Chem Lett; 2017 Feb; 27(4):744-749. PubMed ID: 28131715
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Divergent JNK Phosphorylation of HDAC3 in Triple-Negative Breast Cancer Cells Determines HDAC Inhibitor Binding and Selectivity.
    Hanigan TW; Aboukhatwa SM; Taha TY; Frasor J; Petukhov PA
    Cell Chem Biol; 2017 Nov; 24(11):1356-1367.e8. PubMed ID: 28943357
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Dual-acting histone deacetylase-topoisomerase I inhibitors.
    Guerrant W; Patil V; Canzoneri JC; Yao LP; Hood R; Oyelere AK
    Bioorg Med Chem Lett; 2013 Jun; 23(11):3283-7. PubMed ID: 23622981
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Aza-SAHA Derivatives Are Selective Histone Deacetylase 10 Chemical Probes That Inhibit Polyamine Deacetylation and Phenocopy HDAC10 Knockout.
    Steimbach RR; Herbst-Gervasoni CJ; Lechner S; Stewart TM; Klinke G; Ridinger J; Géraldy MNE; Tihanyi G; Foley JR; Uhrig U; Kuster B; Poschet G; Casero RA; Médard G; Oehme I; Christianson DW; Gunkel N; Miller AK
    J Am Chem Soc; 2022 Oct; 144(41):18861-18875. PubMed ID: 36200994
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Synthesis and HDAC inhibitory activity of isosteric thiazoline-oxazole largazole analogs.
    Guerra-Bubb JM; Bowers AA; Smith WB; Paranal R; Estiu G; Wiest O; Bradner JE; Williams RM
    Bioorg Med Chem Lett; 2013 Nov; 23(21):6025-8. PubMed ID: 24035339
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Anti-tumor activity of phenoxybenzamine and its inhibition of histone deacetylases.
    Inchiosa MA
    PLoS One; 2018; 13(6):e0198514. PubMed ID: 29897996
    [TBL] [Abstract][Full Text] [Related]  

  • 13. A "Double-Locked" and Enzyme/pH-Activated Theranostic Agent for Accurate Tumor Imaging and Therapy.
    Luo J; Guan Z; Gao W; Wang C; Xu Z; Meng C; Liu Y; Zhang Y; Guo Q; Ling Y
    Molecules; 2022 Jan; 27(2):. PubMed ID: 35056740
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Design, synthesis and biological evaluation of colchicine derivatives as novel tubulin and histone deacetylase dual inhibitors.
    Zhang X; Kong Y; Zhang J; Su M; Zhou Y; Zang Y; Li J; Chen Y; Fang Y; Zhang X; Lu W
    Eur J Med Chem; 2015 May; 95():127-35. PubMed ID: 25805446
    [TBL] [Abstract][Full Text] [Related]  

  • 15. The Development of HDAC and Tubulin Dual-Targeting Inhibitors for Cancer Therapy.
    Nie J; Wu H; Luan Y; Wu J
    Mini Rev Med Chem; 2024; 24(5):480-490. PubMed ID: 37461341
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Panobinostat Synergistically Enhances the Cytotoxicity of Microtubule Destabilizing Drugs in Ovarian Cancer Cells.
    Ovejero-Sánchez M; Asensio-Juárez G; González M; Puebla P; Vicente-Manzanares M; Pélaez R; González-Sarmiento R; Herrero AB
    Int J Mol Sci; 2022 Oct; 23(21):. PubMed ID: 36361809
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Prognostic and Predictive Biomarkers in Gliomas.
    Śledzińska P; Bebyn MG; Furtak J; Kowalewski J; Lewandowska MA
    Int J Mol Sci; 2021 Sep; 22(19):. PubMed ID: 34638714
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Bifunctional HDAC Therapeutics: One Drug to Rule Them All?
    Smalley JP; Cowley SM; Hodgkinson JT
    Molecules; 2020 Sep; 25(19):. PubMed ID: 32987782
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Discovery of a Novel Hybrid of Vorinostat and Riluzole as a Potent Antitumor Agent.
    Xu Q; Liu C; Zang J; Gao S; Chou CJ; Zhang Y
    Front Cell Dev Biol; 2020; 8():454. PubMed ID: 32760715
    [TBL] [Abstract][Full Text] [Related]  

  • 20.
    ; ; . PubMed ID:
    [No Abstract]   [Full Text] [Related]  

    [Next]    [New Search]
    of 5.