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5. Selective inhibition of EZH2 by ZLD1039 blocks H3K27 methylation and leads to potent anti-tumor activity in breast cancer. Song X; Gao T; Wang N; Feng Q; You X; Ye T; Lei Q; Zhu Y; Xiong M; Xia Y; Yang F; Shi Y; Wei Y; Zhang L; Yu L Sci Rep; 2016 Feb; 6():20864. PubMed ID: 26868841 [TBL] [Abstract][Full Text] [Related]
6. Malignant rhabdoid tumors express stem cell factors, which relate to the expression of EZH2 and Id proteins. Venneti S; Le P; Martinez D; Xie SX; Sullivan LM; Rorke-Adams LB; Pawel B; Judkins AR Am J Surg Pathol; 2011 Oct; 35(10):1463-72. PubMed ID: 21921784 [TBL] [Abstract][Full Text] [Related]
7. Selective inhibition of Ezh2 by a small molecule inhibitor blocks tumor cells proliferation. Qi W; Chan H; Teng L; Li L; Chuai S; Zhang R; Zeng J; Li M; Fan H; Lin Y; Gu J; Ardayfio O; Zhang JH; Yan X; Fang J; Mi Y; Zhang M; Zhou T; Feng G; Chen Z; Li G; Yang T; Zhao K; Liu X; Yu Z; Lu CX; Atadja P; Li E Proc Natl Acad Sci U S A; 2012 Dec; 109(52):21360-5. PubMed ID: 23236167 [TBL] [Abstract][Full Text] [Related]
8. Analysis of the antiproliferative effects of 3-deazaneoplanocin A in combination with standard anticancer agents in rhabdoid tumor cell lines. Unland R; Borchardt C; Clemens D; Kool M; Dirksen U; Frühwald MC Anticancer Drugs; 2015 Mar; 26(3):301-11. PubMed ID: 25415657 [TBL] [Abstract][Full Text] [Related]
9. A selective inhibitor of EZH2 blocks H3K27 methylation and kills mutant lymphoma cells. Knutson SK; Wigle TJ; Warholic NM; Sneeringer CJ; Allain CJ; Klaus CR; Sacks JD; Raimondi A; Majer CR; Song J; Scott MP; Jin L; Smith JJ; Olhava EJ; Chesworth R; Moyer MP; Richon VM; Copeland RA; Keilhack H; Pollock RM; Kuntz KW Nat Chem Biol; 2012 Nov; 8(11):890-6. PubMed ID: 23023262 [TBL] [Abstract][Full Text] [Related]
10. EZH2: a novel target for cancer treatment. Duan R; Du W; Guo W J Hematol Oncol; 2020 Jul; 13(1):104. PubMed ID: 32723346 [TBL] [Abstract][Full Text] [Related]
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12. EZH2 inhibition as a therapeutic strategy for lymphoma with EZH2-activating mutations. McCabe MT; Ott HM; Ganji G; Korenchuk S; Thompson C; Van Aller GS; Liu Y; Graves AP; Della Pietra A; Diaz E; LaFrance LV; Mellinger M; Duquenne C; Tian X; Kruger RG; McHugh CF; Brandt M; Miller WH; Dhanak D; Verma SK; Tummino PJ; Creasy CL Nature; 2012 Dec; 492(7427):108-12. PubMed ID: 23051747 [TBL] [Abstract][Full Text] [Related]
13. Selective Killing of SMARCA2- and SMARCA4-deficient Small Cell Carcinoma of the Ovary, Hypercalcemic Type Cells by Inhibition of EZH2: Chan-Penebre E; Armstrong K; Drew A; Grassian AR; Feldman I; Knutson SK; Kuplast-Barr K; Roche M; Campbell J; Ho P; Copeland RA; Chesworth R; Smith JJ; Keilhack H; Ribich SA Mol Cancer Ther; 2017 May; 16(5):850-860. PubMed ID: 28292935 [TBL] [Abstract][Full Text] [Related]
14. Therapeutic Targeting of EZH2 and BET BRD4 in Pediatric Rhabdoid Tumors. Ishi Y; Zhang Y; Zhang A; Sasaki T; Piunti A; Suri A; Watanabe J; Abe K; He X; Katagi H; Bhalla P; Natsumeda M; Zou L; Shilatifard A; Hashizume R Mol Cancer Ther; 2022 May; 21(5):715-726. PubMed ID: 35247919 [TBL] [Abstract][Full Text] [Related]
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16. Targeted disruption of the EZH2-EED complex inhibits EZH2-dependent cancer. Kim W; Bird GH; Neff T; Guo G; Kerenyi MA; Walensky LD; Orkin SH Nat Chem Biol; 2013 Oct; 9(10):643-50. PubMed ID: 23974116 [TBL] [Abstract][Full Text] [Related]
17. Discovery of Dual Lysine Methyltransferase G9a and EZH2 Inhibitors with In Vivo Efficacy against Malignant Rhabdoid Tumor. Shi Y; Zhang Q; Zhang M; Chen Y; Sun J; Chen L; Liu S; Liu Z; Yang J; Wu C; Zheng Z; Wang L; Chen G J Med Chem; 2023 Apr; 66(8):5685-5702. PubMed ID: 37021456 [TBL] [Abstract][Full Text] [Related]
18. Combined epigenetic therapy with the histone methyltransferase EZH2 inhibitor 3-deazaneplanocin A and the histone deacetylase inhibitor panobinostat against human AML cells. Fiskus W; Wang Y; Sreekumar A; Buckley KM; Shi H; Jillella A; Ustun C; Rao R; Fernandez P; Chen J; Balusu R; Koul S; Atadja P; Marquez VE; Bhalla KN Blood; 2009 Sep; 114(13):2733-43. PubMed ID: 19638619 [TBL] [Abstract][Full Text] [Related]
19. Identification of EZH2 and EZH1 small molecule inhibitors with selective impact on diffuse large B cell lymphoma cell growth. Garapaty-Rao S; Nasveschuk C; Gagnon A; Chan EY; Sandy P; Busby J; Balasubramanian S; Campbell R; Zhao F; Bergeron L; Audia JE; Albrecht BK; Harmange JC; Cummings R; Trojer P Chem Biol; 2013 Nov; 20(11):1329-39. PubMed ID: 24183969 [TBL] [Abstract][Full Text] [Related]
20. Identification of coexistence of DNA methylation and H3K27me3 specifically in cancer cells as a promising target for epigenetic therapy. Takeshima H; Wakabayashi M; Hattori N; Yamashita S; Ushijima T Carcinogenesis; 2015 Feb; 36(2):192-201. PubMed ID: 25477340 [TBL] [Abstract][Full Text] [Related] [Next] [New Search]