131 related articles for article (PubMed ID: 23884134)
1. Mechanistic studies on regioselective dephosphorylation of phosphate prodrugs during a facile synthesis of antitumor phosphorylated 2-phenyl-6,7-methylenedioxy-1H-quinolin-4-one.
Cheng YY; Liu CY; Huang LJ; Huang CH; Lee KH; Lin CT; Kuo SC
Molecules; 2013 Jul; 18(7):8028-45. PubMed ID: 23884134
[TBL] [Abstract][Full Text] [Related]
2. Water soluble prodrugs of the antitumor agent 3-[(3-amino-4-methoxy)phenyl]-2-(3,4,5-trimethoxyphenyl)cyclopent-2-ene-1-one.
Nam NH; Kim Y; You YJ; Hong DH; Kim HM; Ahn BZ
Bioorg Med Chem; 2003 Mar; 11(6):1021-9. PubMed ID: 12614888
[TBL] [Abstract][Full Text] [Related]
3. Antineoplastic agents. 578. Synthesis of stilstatins 1 and 2 and their water-soluble prodrugs.
Pettit GR; Thornhill A; Melody N; Knight JC
J Nat Prod; 2009 Mar; 72(3):380-8. PubMed ID: 19228038
[TBL] [Abstract][Full Text] [Related]
4. Synthesis and evaluation of anticancer activity of BOC26P, an ortho-aryl chalcone sodium phosphate as water-soluble prodrugs in vitro and in vivo.
Zhu C; Wang R; Zheng W; Chen D; Yue X; Cao Y; Qin W; Sun H; Wang Y; Liu Z; Li B; Du J; Bu X; Zhou B
Biomed Pharmacother; 2017 Dec; 96():551-562. PubMed ID: 29032339
[TBL] [Abstract][Full Text] [Related]
5. Synthesis and biological evaluation of hypoxia-activated prodrugs of SN-38.
Jin C; Zhang Q; Lu W
Eur J Med Chem; 2017 May; 132():135-141. PubMed ID: 28350997
[TBL] [Abstract][Full Text] [Related]
6. Synthesis of pochoxime prodrugs as potent HSP90 inhibitors.
Wang C; Barluenga S; Koripelly GK; Fontaine JG; Chen R; Yu JC; Shen X; Chabala JC; Heck JV; Rubenstein A; Winssinger N
Bioorg Med Chem Lett; 2009 Jul; 19(14):3836-40. PubMed ID: 19410458
[TBL] [Abstract][Full Text] [Related]
7. Synthesis and in vivo antitumor evaluation of 2-methoxyestradiol 3-phosphate, 17-phosphate, and 3,17-diphosphate.
Edsall AB; Agoston GE; Treston AM; Plum SM; McClanahan RH; Lu TS; Song W; Cushman M
J Med Chem; 2007 Dec; 50(26):6700-5. PubMed ID: 18052315
[TBL] [Abstract][Full Text] [Related]
8. Synthesis and evaluation of water-soluble paclitaxel prodrugs.
Feng X; Yuan YJ; Wu JC
Bioorg Med Chem Lett; 2002 Nov; 12(22):3301-3. PubMed ID: 12392737
[TBL] [Abstract][Full Text] [Related]
9. Synthesis and Evaluation of Millepachine Amino Acid Prodrugs With Enhanced Solubility as Antitumor Agents.
Wu Y; Cao D; Wang F; Ma L; Gao G; Chen L
Chem Biol Drug Des; 2015 Oct; 86(4):559-67. PubMed ID: 25643726
[TBL] [Abstract][Full Text] [Related]
10. Design, synthesis, and evaluation of water-soluble morpholino-decorated paclitaxel prodrugs with remarkably decreased toxicity.
Feng S; Chen K; Wang C; Jiang X; Dong H; Gong Z; Liu K
Bioorg Med Chem Lett; 2016 Aug; 26(15):3598-602. PubMed ID: 27311893
[TBL] [Abstract][Full Text] [Related]
11. Synthesis and biological activities of a pH-dependently activated water-soluble prodrug of a novel hexacyclic camptothecin analog.
Ohwada J; Ozawa S; Kohchi M; Fukuda H; Murasaki C; Suda H; Murata T; Niizuma S; Tsukazaki M; Ori K; Yoshinari K; Itezono Y; Endo M; Ura M; Tanimura H; Miyazaki Y; Kawashima A; Nagao S; Namba E; Ogawa K; Kobayashi K; Okabe H; Umeda I; Shimma N
Bioorg Med Chem Lett; 2009 May; 19(10):2772-6. PubMed ID: 19362835
[TBL] [Abstract][Full Text] [Related]
12. Discovery of a potent tubulin polymerization inhibitor: synthesis and evaluation of water-soluble prodrugs of benzophenone analog.
Lee J; Bae S; Lee SH; Choi H; Kim YH; Kim SJ; Park GT; Moon SK; Kim DH; Lee S; Ahn SK; Choi NS; Lee KJ
Bioorg Med Chem Lett; 2010 Nov; 20(21):6327-30. PubMed ID: 20850313
[TBL] [Abstract][Full Text] [Related]
13. Design, Synthesis, and Biological Evaluation of a Novel Water-soluble Prodrug of Docetaxel with Amino Acid as a Linker.
Ma H; Chen G; Wang T; Li Q; Liu Y
Chem Biol Drug Des; 2016 Sep; 88(3):363-9. PubMed ID: 27061863
[TBL] [Abstract][Full Text] [Related]
14. Investigation of amino acid conjugates of (S)-1-[1-(4-aminobenzoyl)-2,3-dihydro-1H-indol-6-sulfonyl]-4-phenyl-imidazolidin-2-one (DW2282) as water soluble anticancer prodrugs.
Lee KC; Venkateswararao E; Sharma VK; Jung SH
Eur J Med Chem; 2014 Jun; 80():439-46. PubMed ID: 24796884
[TBL] [Abstract][Full Text] [Related]
15. Synthesis and antitumor activities of amino acid prodrugs of amino-combretastatins.
Ohsumi K; Hatanaka T; Nakagawa R; Fukuda Y; Morinaga Y; Suga Y; Nihei Y; Ohishi K; Akiyama Y; Tsuji T
Anticancer Drug Des; 1999 Dec; 14(6):539-48. PubMed ID: 10834274
[TBL] [Abstract][Full Text] [Related]
16. Design and Characterization of a Pyridone-Containing EZH2 Inhibitor Phosphate Prodrug.
Kung PP; Fan C; Gukasyan HJ; Huang B; Kephart S; Kraus M; Lee JH; Sutton SC; Yamazaki S; Zehnder L
J Med Chem; 2021 Feb; 64(3):1725-1732. PubMed ID: 33529029
[TBL] [Abstract][Full Text] [Related]
17. Design, synthesis, and anticancer activity of phosphonic acid diphosphate derivative of adenine-containing butenolide and its water-soluble derivatives of paclitaxel with high antitumor activity.
Moosavi-Movahedi AA; Hakimelahi S; Chamani J; Khodarahmi GA; Hassanzadeh F; Luo FT; Ly TW; Shia KS; Yen CF; Jain ML; Kulatheeswaran R; Xue C; Pasdar M; Hakimelahi GH
Bioorg Med Chem; 2003 Oct; 11(20):4303-13. PubMed ID: 13129566
[TBL] [Abstract][Full Text] [Related]
18. Rational design of carbamate-based dual binding site and central AChE inhibitors by a "biooxidisable" prodrug approach: Synthesis, in vitro evaluation and docking studies.
Ţînţaş ML; Gembus V; Alix F; Barré A; Coadou G; Truong L; Sebban M; Papamicaël C; Oulyadi H; Levacher V
Eur J Med Chem; 2018 Jul; 155():171-182. PubMed ID: 29886321
[TBL] [Abstract][Full Text] [Related]
19. Heparin-paclitaxel conjugates as drug delivery system: synthesis, self-assembly property, drug release, and antitumor activity.
Wang Y; Xin D; Liu K; Zhu M; Xiang J
Bioconjug Chem; 2009 Dec; 20(12):2214-21. PubMed ID: 19950889
[TBL] [Abstract][Full Text] [Related]
20. Synthesis and antitumor activities of water-soluble benzoylphenylureas.
Okada H; Kato M; Koyanagi T; Mizuno K
Chem Pharm Bull (Tokyo); 1999 Mar; 47(3):430-3. PubMed ID: 10212393
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]
