BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

176 related articles for article (PubMed ID: 23938052)

  • 1. Synthesis, enzyme kinetics and computational evaluation of N-(β-D-glucopyranosyl) oxadiazolecarboxamides as glycogen phosphorylase inhibitors.
    Polyák M; Varga G; Szilágyi B; Juhász L; Docsa T; Gergely P; Begum J; Hayes JM; Somsák L
    Bioorg Med Chem; 2013 Sep; 21(18):5738-47. PubMed ID: 23938052
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Synthesis of heterocyclic N-(β-D-glucopyranosyl)carboxamides for inhibition of glycogen phosphorylase.
    Kónya B; Docsa T; Gergely P; Somsák L
    Carbohydr Res; 2012 Apr; 351():56-63. PubMed ID: 22365837
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Synthesis of 2-(β-D-glucopyranosylamino)-5-substituted-1,3,4-oxadiazoles for inhibition of glycogen phosphorylase.
    Tóth M; Szőcs B; Kaszás T; Docsa T; Gergely P; Somsák L
    Carbohydr Res; 2013 Nov; 381():196-204. PubMed ID: 23673237
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Synthesis of variously coupled conjugates of D-glucose, 1,3,4-oxadiazole, and 1,2,3-triazole for inhibition of glycogen phosphorylase.
    Kun S; Nagy GZ; Tóth M; Czecze L; Van Nhien AN; Docsa T; Gergely P; Charavgi MD; Skourti PV; Chrysina ED; Patonay T; Somsák L
    Carbohydr Res; 2011 Sep; 346(12):1427-38. PubMed ID: 21470596
    [TBL] [Abstract][Full Text] [Related]  

  • 5. New synthesis of 3-(β-D-glucopyranosyl)-5-substituted-1,2,4-triazoles, nanomolar inhibitors of glycogen phosphorylase.
    Kun S; Bokor É; Varga G; Szőcs B; Páhi A; Czifrák K; Tóth M; Juhász L; Docsa T; Gergely P; Somsák L
    Eur J Med Chem; 2014 Apr; 76():567-79. PubMed ID: 24608000
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Synthesis of 2-(β-D-glucopyranosyl)-5-(substituted-amino)-1,3,4-oxa- and -thiadiazoles for the inhibition of glycogen phosphorylase.
    Szőcs B; Tóth M; Docsa T; Gergely P; Somsák L
    Carbohydr Res; 2013 Nov; 381():187-95. PubMed ID: 23582340
    [TBL] [Abstract][Full Text] [Related]  

  • 7. C-Glucopyranosyl-1,2,4-triazol-5-ones: synthesis and inhibition of glycogen phosphorylase.
    Bokor É; Széles Z; Docsa T; Gergely P; Somsák L
    Carbohydr Res; 2016 Jun; 429():128-34. PubMed ID: 26818133
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Synthesis of N-(beta-D-glucopyranosyl) monoamides of dicarboxylic acids as potential inhibitors of glycogen phosphorylase.
    Czifrák K; Hadady Z; Docsa T; Gergely P; Schmidt J; Wessjohann L; Somsák L
    Carbohydr Res; 2006 Jun; 341(8):947-56. PubMed ID: 16564511
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Synthesis of New C- and N-β-d-Glucopyranosyl Derivatives of Imidazole, 1,2,3-Triazole and Tetrazole, and Their Evaluation as Inhibitors of Glycogen Phosphorylase.
    Kun S; Bokor É; Sipos Á; Docsa T; Somsák L
    Molecules; 2018 Mar; 23(3):. PubMed ID: 29543771
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Synthesis of new glycosyl biuret and urea derivatives as potential glycoenzyme inhibitors.
    Felföldi N; Tóth M; Chrysina ED; Charavgi MD; Alexacou KM; Somsák L
    Carbohydr Res; 2010 Jan; 345(2):208-13. PubMed ID: 20004366
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Synthesis of N-(beta-D-glucopyranosyl)- and N-(2-acetamido-2-deoxy-beta-D-glucopyranosyl) amides as inhibitors of glycogen phosphorylase.
    Györgydeák Z; Hadady Z; Felföldi N; Krakomperger A; Nagy V; Tóth M; Brunyánszki A; Docsa T; Gergely P; Somsák L
    Bioorg Med Chem; 2004 Sep; 12(18):4861-70. PubMed ID: 15336265
    [TBL] [Abstract][Full Text] [Related]  

  • 12. C-(2-Deoxy-d-arabino-hex-1-enopyranosyl)-oxadiazoles: synthesis of possible isomers and their evaluation as glycogen phosphorylase inhibitors.
    Bokor É; Szennyes E; Csupász T; Tóth N; Docsa T; Gergely P; Somsák L
    Carbohydr Res; 2015 Aug; 412():71-9. PubMed ID: 26082971
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Synthesis of substituted 2-(β-D-glucopyranosyl)-benzimidazoles and their evaluation as inhibitors of glycogen phosphorylase.
    Bokor É; Szilágyi E; Docsa T; Gergely P; Somsák L
    Carbohydr Res; 2013 Nov; 381():179-86. PubMed ID: 23419607
    [TBL] [Abstract][Full Text] [Related]  

  • 14. A multidisciplinary study of 3-(β-d-glucopyranosyl)-5-substituted-1,2,4-triazole derivatives as glycogen phosphorylase inhibitors: Computation, synthesis, crystallography and kinetics reveal new potent inhibitors.
    Kun S; Begum J; Kyriakis E; Stamati ECV; Barkas TA; Szennyes E; Bokor É; Szabó KE; Stravodimos GA; Sipos Á; Docsa T; Gergely P; Moffatt C; Patraskaki MS; Kokolaki MC; Gkerdi A; Skamnaki VT; Leonidas DD; Somsák L; Hayes JM
    Eur J Med Chem; 2018 Mar; 147():266-278. PubMed ID: 29453094
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Synthesis and structure-activity relationships of C-glycosylated oxadiazoles as inhibitors of glycogen phosphorylase.
    Tóth M; Kun S; Bokor E; Benltifa M; Tallec G; Vidal S; Docsa T; Gergely P; Somsák L; Praly JP
    Bioorg Med Chem; 2009 Jul; 17(13):4773-85. PubMed ID: 19450985
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Synthesis, In Silico and Kinetics Evaluation of
    Homolya L; Mathomes RT; Varga L; Docsa T; Juhász L; Hayes JM; Somsák L
    Int J Mol Sci; 2024 Apr; 25(9):. PubMed ID: 38731811
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Synthetic, enzyme kinetic, and protein crystallographic studies of C-β-d-glucopyranosyl pyrroles and imidazoles reveal and explain low nanomolar inhibition of human liver glycogen phosphorylase.
    Kantsadi AL; Bokor É; Kun S; Stravodimos GA; Chatzileontiadou DSM; Leonidas DD; Juhász-Tóth É; Szakács A; Batta G; Docsa T; Gergely P; Somsák L
    Eur J Med Chem; 2016 Nov; 123():737-745. PubMed ID: 27522507
    [TBL] [Abstract][Full Text] [Related]  

  • 18. N-(4-Substituted-benzoyl)-N'-(β-d-glucopyranosyl)ureas as inhibitors of glycogen phosphorylase: Synthesis and evaluation by kinetic, crystallographic, and molecular modelling methods.
    Nagy V; Felföldi N; Kónya B; Praly JP; Docsa T; Gergely P; Chrysina ED; Tiraidis C; Kosmopoulou MN; Alexacou KM; Konstantakaki M; Leonidas DD; Zographos SE; Oikonomakos NG; Kozmon S; Tvaroška I; Somsák L
    Bioorg Med Chem; 2012 Mar; 20(5):1801-16. PubMed ID: 22325154
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Glucopyranosylidene-spiro-iminothiazolidinone, a new bicyclic ring system: synthesis, derivatization, and evaluation for inhibition of glycogen phosphorylase by enzyme kinetic and crystallographic methods.
    Czifrák K; Páhi A; Deák S; Kiss-Szikszai A; Kövér KE; Docsa T; Gergely P; Alexacou KM; Papakonstantinou M; Leonidas DD; Zographos SE; Chrysina ED; Somsák L
    Bioorg Med Chem; 2014 Aug; 22(15):4028-41. PubMed ID: 25009003
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Crystallographic and computational studies on 4-phenyl-N-(beta-D-glucopyranosyl)-1H-1,2,3-triazole-1-acetamide, an inhibitor of glycogen phosphorylase: comparison with alpha-D-glucose, N-acetyl-beta-D-glucopyranosylamine and N-benzoyl-N'-beta-D-glucopyranosyl urea binding.
    Alexacou KM; Hayes JM; Tiraidis C; Zographos SE; Leonidas DD; Chrysina ED; Archontis G; Oikonomakos NG; Paul JV; Varghese B; Loganathan D
    Proteins; 2008 May; 71(3):1307-23. PubMed ID: 18041758
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 9.