179 related articles for article (PubMed ID: 23953686)
1. Design and synthesis of (4E)-4-(4-substitutedbenzylideneamino)-3-substituted-2,3-dihydro-2-thioxothiazole-5-carbonitrile as novel A2A receptor antagonists.
Mishra CB; Sharma D; Prakash A; Kumari N; Kumar N; Luthra PM
Bioorg Med Chem; 2013 Oct; 21(19):6077-83. PubMed ID: 23953686
[TBL] [Abstract][Full Text] [Related]
2. 8-(Furan-2-yl)-3-phenethylthiazolo[5,4-e][1,2,4]triazolo[1,5-c]pyrimidine-2(3H)-thione as novel, selective and potent adenosine A(2A) receptor antagonist.
Kumari N; Mishra CB; Prakash A; Kumar N; Mongre R; Luthra PM
Neurosci Lett; 2014 Jan; 558():203-7. PubMed ID: 24161891
[TBL] [Abstract][Full Text] [Related]
3. Novel 8-(furan-2-yl)-3-substituted thiazolo [5,4-e][1,2,4] triazolo[1,5-c] pyrimidine-2(3H)-thione derivatives as potential adenosine A(2A) receptor antagonists.
Mishra CB; Barodia SK; Prakash A; Senthil Kumar JB; Luthra PM
Bioorg Med Chem; 2010 Apr; 18(7):2491-500. PubMed ID: 20303771
[TBL] [Abstract][Full Text] [Related]
4. Novel 8-(furan-2-yl)-3-benzyl thiazolo [5,4-e][1,2,4] triazolo [1,5-c] pyrimidine-2(3H)-thione as selective adenosine A(2A) receptor antagonist.
Barodia SK; Mishra CB; Prakash A; Senthil Kumar JB; Kumari N; Luthra PM
Neurosci Lett; 2011 Jan; 488(1):1-5. PubMed ID: 20708066
[TBL] [Abstract][Full Text] [Related]
5. Synthesis of novel 7-imino-2-thioxo-3,7-dihydro-2H-thiazolo [4,5-d] pyrimidine derivatives as adenosine A2A receptor antagonists.
Luthra PM; Mishra CB; Jha PK; Barodia SK
Bioorg Med Chem Lett; 2010 Feb; 20(3):1214-8. PubMed ID: 20018509
[TBL] [Abstract][Full Text] [Related]
6. Novel adenosine A(2A) receptor ligands: a synthetic, functional and computational investigation of selected literature adenosine A(2A) receptor antagonists for extending into extracellular space.
Jörg M; Shonberg J; Mak FS; Miller ND; Yuriev E; Scammells PJ; Capuano B
Bioorg Med Chem Lett; 2013 Jun; 23(11):3427-33. PubMed ID: 23602401
[TBL] [Abstract][Full Text] [Related]
7. 2-Aminopyrimidines as dual adenosine A1/A2A antagonists.
Robinson SJ; Petzer JP; Terre'Blanche G; Petzer A; van der Walt MM; Bergh JJ; Lourens AC
Eur J Med Chem; 2015 Nov; 104():177-88. PubMed ID: 26462195
[TBL] [Abstract][Full Text] [Related]
8. Design, synthesis and biological evaluation of Tozadenant analogues as adenosine A
Renk DR; Skraban M; Bier D; Schulze A; Wabbals E; Wedekind F; Neumaier F; Neumaier B; Holschbach M
Eur J Med Chem; 2021 Mar; 214():113214. PubMed ID: 33548636
[TBL] [Abstract][Full Text] [Related]
9. Replacement of amide with bioisosteres led to a new series of potent adenosine A2A receptor antagonists.
Yang Z; Li X; Ma H; Zheng J; Zhen X; Zhang X
Bioorg Med Chem Lett; 2014 Jan; 24(1):152-5. PubMed ID: 24332624
[TBL] [Abstract][Full Text] [Related]
10. Novel approaches for targeting the adenosine A2A receptor.
Yuan G; Gedeon NG; Jankins TC; Jones GB
Expert Opin Drug Discov; 2015 Jan; 10(1):63-80. PubMed ID: 25311639
[TBL] [Abstract][Full Text] [Related]
11. New insight into adenosine receptors selectivity derived from a novel series of [5-substituted-4-phenyl-1,3-thiazol-2-yl] benzamides and furamides.
Inamdar GS; Pandya AN; Thakar HM; Sudarsanam V; Kachler S; Sabbadin D; Moro S; Klotz KN; Vasu KK
Eur J Med Chem; 2013 May; 63():924-34. PubMed ID: 23685887
[TBL] [Abstract][Full Text] [Related]
12. Revisiting a receptor-based pharmacophore hypothesis for human A(2A) adenosine receptor antagonists.
Bacilieri M; Ciancetta A; Paoletta S; Federico S; Cosconati S; Cacciari B; Taliani S; Da Settimo F; Novellino E; Klotz KN; Spalluto G; Moro S
J Chem Inf Model; 2013 Jul; 53(7):1620-37. PubMed ID: 23705857
[TBL] [Abstract][Full Text] [Related]
13. Synthesis and SAR studies of analogues of 4-(3,3-dimethyl-butyrylamino)-3,5-difluoro-N-thiazol-2-yl-benzamide (Lu AA41063) as adenosine A2A receptor ligands with improved aqueous solubility.
Mikkelsen GK; Langgård M; Schrøder TJ; Kreilgaard M; Jørgensen EB; Brandt G; Griffon Y; Boffey R; Bang-Andersen B
Bioorg Med Chem Lett; 2015 Mar; 25(6):1212-6. PubMed ID: 25701253
[TBL] [Abstract][Full Text] [Related]
14. In silico study of naphtha [1, 2-d] thiazol-2-amine with adenosine A 2A receptor and its role in antagonism of haloperidol-induced motor impairments in mice.
Luthra PM; Prakash A; Barodia SK; Kumari R; Mishra CB; Kumar JB
Neurosci Lett; 2009 Oct; 463(3):215-8. PubMed ID: 19654038
[TBL] [Abstract][Full Text] [Related]
15. Binding kinetics of ZM241385 derivatives at the human adenosine A2A receptor.
Guo D; Xia L; van Veldhoven JP; Hazeu M; Mocking T; Brussee J; Ijzerman AP; Heitman LH
ChemMedChem; 2014 Apr; 9(4):752-61. PubMed ID: 24591302
[TBL] [Abstract][Full Text] [Related]
16. Substituted thieno[2,3-d]pyrimidines as adenosine A2A receptor antagonists.
Shook BC; Chakravarty D; Barbay JK; Wang A; Leonard K; Alford V; Powell MT; Rassnick S; Scannevin RH; Carroll K; Wallace N; Crooke J; Ault M; Lampron L; Westover L; Rhodes K; Jackson PF
Bioorg Med Chem Lett; 2013 May; 23(9):2688-91. PubMed ID: 23522563
[TBL] [Abstract][Full Text] [Related]
17. Allosteric interactions between agonists and antagonists within the adenosine A2A receptor-dopamine D2 receptor heterotetramer.
Bonaventura J; Navarro G; Casadó-Anguera V; Azdad K; Rea W; Moreno E; Brugarolas M; Mallol J; Canela EI; Lluís C; Cortés A; Volkow ND; Schiffmann SN; Ferré S; Casadó V
Proc Natl Acad Sci U S A; 2015 Jul; 112(27):E3609-18. PubMed ID: 26100888
[TBL] [Abstract][Full Text] [Related]
18. Design, synthesis and biological evaluation of novel scaffold benzo[4,5]imidazo [1,2-a]pyrazin-1-amine: Towards adenosine A
Reddy GL; Sarma R; Liu S; Huang W; Lei J; Fu J; Hu W
Eur J Med Chem; 2021 Jan; 210():113040. PubMed ID: 33316692
[TBL] [Abstract][Full Text] [Related]
19. Crystal structure of the adenosine A
Sun B; Bachhawat P; Chu ML; Wood M; Ceska T; Sands ZA; Mercier J; Lebon F; Kobilka TS; Kobilka BK
Proc Natl Acad Sci U S A; 2017 Feb; 114(8):2066-2071. PubMed ID: 28167788
[TBL] [Abstract][Full Text] [Related]
20. The adenosine A(2A) antagonistic properties of selected C8-substituted xanthines.
Van der Walt MM; Terre'Blanche G; Petzer A; Lourens AC; Petzer JP
Bioorg Chem; 2013 Aug; 49():49-58. PubMed ID: 23892098
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]