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9. Lobelane analogues containing 4-hydroxy and 4-(2-fluoroethoxy) aromatic substituents: Potent and selective inhibitors of [(3)H]dopamine uptake at the vesicular monoamine transporter-2. Joolakanti SR; Nickell JR; Janganati V; Zheng G; Dwoskin LP; Crooks PA Bioorg Med Chem Lett; 2016 May; 26(10):2422-2427. PubMed ID: 27080180 [TBL] [Abstract][Full Text] [Related]
10. GZ-793A, a lobelane analog, interacts with the vesicular monoamine transporter-2 to inhibit the effect of methamphetamine. Horton DB; Nickell JR; Zheng G; Crooks PA; Dwoskin LP J Neurochem; 2013 Oct; 127(2):177-86. PubMed ID: 23875622 [TBL] [Abstract][Full Text] [Related]
11. Lobeline analogs with enhanced affinity and selectivity for plasmalemma and vesicular monoamine transporters. Miller DK; Crooks PA; Zheng G; Grinevich VP; Norrholm SD; Dwoskin LP J Pharmacol Exp Ther; 2004 Sep; 310(3):1035-45. PubMed ID: 15121762 [TBL] [Abstract][Full Text] [Related]
12. 1,4-Diphenalkylpiperidines: A new scaffold for the design of potent inhibitors of the vesicular monoamine transporter-2. Nickell JR; Culver JP; Janganati V; Zheng G; Dwoskin LP; Crooks PA Bioorg Med Chem Lett; 2016 Jul; 26(13):2997-3000. PubMed ID: 27212067 [TBL] [Abstract][Full Text] [Related]
13. Defunctionalized lobeline analogues: structure-activity of novel ligands for the vesicular monoamine transporter. Zheng G; Dwoskin LP; Deaciuc AG; Norrholm SD; Crooks PA J Med Chem; 2005 Aug; 48(17):5551-60. PubMed ID: 16107155 [TBL] [Abstract][Full Text] [Related]
15. New Scaffold for Lead Compounds to Treat Methamphetamine Use Disorders. Lee NR; Zheng G; Crooks PA; Bardo MT; Dwoskin LP AAPS J; 2018 Feb; 20(2):29. PubMed ID: 29427069 [TBL] [Abstract][Full Text] [Related]
16. GZ-11608, a Vesicular Monoamine Transporter-2 Inhibitor, Decreases the Neurochemical and Behavioral Effects of Methamphetamine. Lee NR; Zheng G; Leggas M; Janganati V; Nickell JR; Crooks PA; Bardo MT; Dwoskin LP J Pharmacol Exp Ther; 2019 Nov; 371(2):526-543. PubMed ID: 31413138 [TBL] [Abstract][Full Text] [Related]
17. GZ-793A inhibits the neurochemical effects of methamphetamine via a selective interaction with the vesicular monoamine transporter-2. Nickell JR; Siripurapu KB; Horton DB; Zheng G; Crooks PA; Dwoskin LP Eur J Pharmacol; 2017 Jan; 795():143-149. PubMed ID: 27986625 [TBL] [Abstract][Full Text] [Related]
18. Effects of VMAT2 inhibitors lobeline and GZ-793A on methamphetamine-induced changes in dopamine release, metabolism and synthesis in vivo. Meyer AC; Neugebauer NM; Zheng G; Crooks PA; Dwoskin LP; Bardo MT J Neurochem; 2013 Oct; 127(2):187-98. PubMed ID: 23875705 [TBL] [Abstract][Full Text] [Related]
19. Lobeline displaces [3H]dihydrotetrabenazine binding and releases [3H]dopamine from rat striatal synaptic vesicles: comparison with d-amphetamine. Teng L; Crooks PA; Dwoskin LP J Neurochem; 1998 Jul; 71(1):258-65. PubMed ID: 9648873 [TBL] [Abstract][Full Text] [Related]
20. Pyrrolidine analogues of lobelane: relationship of affinity for the dihydrotetrabenazine binding site with function of the vesicular monoamine transporter 2 (VMAT2). Vartak AP; Nickell JR; Chagkutip J; Dwoskin LP; Crooks PA J Med Chem; 2009 Dec; 52(23):7878-82. PubMed ID: 19691331 [TBL] [Abstract][Full Text] [Related] [Next] [New Search]