BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

146 related articles for article (PubMed ID: 24022991)

  • 1. Synthesis and anti-Plasmodium activity of benzimidazole analogues structurally related to astemizole.
    Roman G; Crandall IE; Szarek WA
    ChemMedChem; 2013 Nov; 8(11):1795-804. PubMed ID: 24022991
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Astemizole analogues with reduced hERG inhibition as potent antimalarial compounds.
    Tian J; Vandermosten L; Peigneur S; Moreels L; Rozenski J; Tytgat J; Herdewijn P; Van den Steen PE; De Jonghe S
    Bioorg Med Chem; 2017 Dec; 25(24):6332-6344. PubMed ID: 29042223
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Multistage Antiplasmodium Activity of Astemizole Analogues and Inhibition of Hemozoin Formation as a Contributor to Their Mode of Action.
    Kumar M; Okombo J; Mambwe D; Taylor D; Lawrence N; Reader J; van der Watt M; Fontinha D; Sanches-Vaz M; Bezuidenhout BC; Lauterbach SB; Liebenberg D; Birkholtz LM; Coetzer TL; Prudêncio M; Egan TJ; Wittlin S; Chibale K
    ACS Infect Dis; 2019 Feb; 5(2):303-315. PubMed ID: 30525439
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Synthesis and antiprotozoal activity of some 2-(trifluoromethyl)-1H-benzimidazole bioisosteres.
    Navarrete-Vázquez G; Rojano-Vilchis Mde M; Yépez-Mulia L; Meléndez V; Gerena L; Hernández-Campos A; Castillo R; Hernández-Luis F
    Eur J Med Chem; 2006 Jan; 41(1):135-41. PubMed ID: 16260067
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Bis(oxyphenylene)benzimidazoles: a novel class of anti-Plasmodium falciparum agents.
    Mayence A; Vanden Eynde JJ; Kaiser M; Brun R; Yarlett N; Huang TL
    Bioorg Med Chem; 2011 Dec; 19(24):7493-500. PubMed ID: 22061825
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Chloroquine-astemizole hybrids with potent in vitro and in vivo antiplasmodial activity.
    Musonda CC; Whitlock GA; Witty MJ; Brun R; Kaiser M
    Bioorg Med Chem Lett; 2009 Jan; 19(2):481-4. PubMed ID: 19054674
    [TBL] [Abstract][Full Text] [Related]  

  • 7. New benzimidazole derivatives as antiplasmodial agents and plasmepsin inhibitors: synthesis and analysis of structure-activity relationships.
    Saify ZS; Azim MK; Ahmad W; Nisa M; Goldberg DE; Hussain SA; Akhtar S; Akram A; Arayne A; Oksman A; Khan IA
    Bioorg Med Chem Lett; 2012 Jan; 22(2):1282-6. PubMed ID: 22204908
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Syntheses and in Vitro Antiplasmodial Activity of Aminoalkylated Chalcones and Analogues.
    Wilhelm A; Kendrekar P; Noreljaleel AE; Abay ET; Bonnet SL; Wiesner L; de Kock C; Swart KJ; van der Westhuizen JH
    J Nat Prod; 2015 Aug; 78(8):1848-58. PubMed ID: 26235033
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Synthesis and biological evaluation of 2-aminothiazole derivatives as antimycobacterial and antiplasmodial agents.
    Mjambili F; Njoroge M; Naran K; De Kock C; Smith PJ; Mizrahi V; Warner D; Chibale K
    Bioorg Med Chem Lett; 2014 Jan; 24(2):560-4. PubMed ID: 24373723
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Benzoheterocyclic amodiaquine analogues with potent antiplasmodial activity: synthesis and pharmacological evaluation.
    Ongarora DS; Gut J; Rosenthal PJ; Masimirembwa CM; Chibale K
    Bioorg Med Chem Lett; 2012 Aug; 22(15):5046-50. PubMed ID: 22749280
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Antimalarial and insecticidal activities of newly synthesized derivatives of Benzimidazole.
    Kamil A; Akhter S; Ahmed M; Rizwani GH; Hassan S; Naeem S; Jahan S; Khursheed R; Zahid H
    Pak J Pharm Sci; 2015 Nov; 28(6):2179-84. PubMed ID: 26639510
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Anti-Plasmodium activity of imidazole-dioxolane compounds.
    Vlahakis JZ; Kinobe RT; Nakatsu K; Szarek WA; Crandall IE
    Bioorg Med Chem Lett; 2006 May; 16(9):2396-406. PubMed ID: 16495054
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Borrelidin analogues with antimalarial activity: design, synthesis and biological evaluation against Plasmodium falciparum parasites.
    Sugawara A; Tanaka T; Hirose T; Ishiyama A; Iwatsuki M; Takahashi Y; Otoguro K; Ōmura S; Sunazuka T
    Bioorg Med Chem Lett; 2013 Apr; 23(8):2302-5. PubMed ID: 23499502
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Anti-Plasmodium activity of imidazolium and triazolium salts.
    Vlahakis JZ; Lazar C; Crandall IE; Szarek WA
    Bioorg Med Chem; 2010 Aug; 18(16):6184-96. PubMed ID: 20634079
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Synthesis of novel benzimidazole acrylonitriles for inhibition of Plasmodium falciparum growth by dual target inhibition.
    Sharma K; Shrivastava A; Mehra RN; Deora GS; Alam MM; Zaman MS; Akhter M
    Arch Pharm (Weinheim); 2018 Jan; 351(1):. PubMed ID: 29227011
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Pharmacomodulation on the 3-acetylursolic acid skeleton: Design, synthesis, and biological evaluation of novel N-{3-[4-(3-aminopropyl)piperazinyl]propyl}-3-O-acetylursolamide derivatives as antimalarial agents.
    Gnoatto SC; Susplugas S; Dalla Vechia L; Ferreira TB; Dassonville-Klimpt A; Zimmer KR; Demailly C; Da Nascimento S; Guillon J; Grellier P; Verli H; Gosmann G; Sonnet P
    Bioorg Med Chem; 2008 Jan; 16(2):771-82. PubMed ID: 17967541
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Synthesis, characterization and antimalarial activity of quinoline-pyrimidine hybrids.
    Pretorius SI; Breytenbach WJ; de Kock C; Smith PJ; N'Da DD
    Bioorg Med Chem; 2013 Jan; 21(1):269-77. PubMed ID: 23168082
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Mechanism-based inhibitors of the aspartyl protease plasmepsin II as potential antimalarial agents.
    Gupta D; Yedidi RS; Varghese S; Kovari LC; Woster PM
    J Med Chem; 2010 May; 53(10):4234-47. PubMed ID: 20438064
    [TBL] [Abstract][Full Text] [Related]  

  • 19. 2-Acylamino-5-chlorobenzophenones with enhanced selectivity towards malaria parasites.
    Heinrich S; Altenkämper M; Bechem B; Perruchon J; Ortmann R; Dahse HM; Wang Y; Lanzer M; Schlitzer M
    Eur J Med Chem; 2011 Apr; 46(4):1331-42. PubMed ID: 21345543
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Synthetic indole and melatonin derivatives exhibit antimalarial activity on the cell cycle of the human malaria parasite Plasmodium falciparum.
    Schuck DC; Jordão AK; Nakabashi M; Cunha AC; Ferreira VF; Garcia CR
    Eur J Med Chem; 2014 May; 78():375-82. PubMed ID: 24699367
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 8.