162 related articles for article (PubMed ID: 24476926)
1. Molecular determinants responsible for sedative and non-sedative properties of histamine H₁-receptor antagonists.
Uesawa Y; Hishinuma S; Shoji M
J Pharmacol Sci; 2014; 124(2):160-8. PubMed ID: 24476926
[TBL] [Abstract][Full Text] [Related]
2. Intact cell binding for in vitro prediction of sedative and non-sedative histamine H1-receptor antagonists based on receptor internalization.
Hishinuma S; Sato Y; Kobayashi Y; Komazaki H; Saito M
J Pharmacol Sci; 2008 May; 107(1):66-79. PubMed ID: 18446005
[TBL] [Abstract][Full Text] [Related]
3. Why are second-generation H1-antihistamines minimally sedating?
Hu Y; Sieck DE; Hsu WH
Eur J Pharmacol; 2015 Oct; 765():100-6. PubMed ID: 26291661
[TBL] [Abstract][Full Text] [Related]
4. Factors involved in the absence of sedative effects by the second-generation antihistamines.
Timmerman H
Allergy; 2000; 55 Suppl 60():5-10. PubMed ID: 10887969
[No Abstract] [Full Text] [Related]
5. The clinical pharmacology of non-sedating antihistamines.
Yanai K; Yoshikawa T; Yanai A; Nakamura T; Iida T; Leurs R; Tashiro M
Pharmacol Ther; 2017 Oct; 178():148-156. PubMed ID: 28457804
[TBL] [Abstract][Full Text] [Related]
6. Affinity for the P-glycoprotein efflux pump at the blood-brain barrier may explain the lack of CNS side-effects of modern antihistamines.
Chishty M; Reichel A; Siva J; Abbott NJ; Begley DJ
J Drug Target; 2001 Jun; 9(3):223-8. PubMed ID: 11697207
[TBL] [Abstract][Full Text] [Related]
7. Positron emission tomography evaluation of sedative properties of antihistamines.
Yanai K; Zhang D; Tashiro M; Yoshikawa T; Naganuma F; Harada R; Nakamura T; Shibuya K; Okamura N
Expert Opin Drug Saf; 2011 Jul; 10(4):613-22. PubMed ID: 21521134
[TBL] [Abstract][Full Text] [Related]
8. P-glycoprotein limits the brain penetration of nonsedating but not sedating H1-antagonists.
Chen C; Hanson E; Watson JW; Lee JS
Drug Metab Dispos; 2003 Mar; 31(3):312-8. PubMed ID: 12584158
[TBL] [Abstract][Full Text] [Related]
9. Effects of first- and second-generation histamine-H1-receptor antagonists on the pentobarbital-induced loss of the righting reflex in streptozotocin-induced diabetic mice.
Kamei J; Hirano S; Miyata S; Saitoh A; Onodera K
J Pharmacol Sci; 2005 Feb; 97(2):266-72. PubMed ID: 15699576
[TBL] [Abstract][Full Text] [Related]
10. Relationship between occupation of cerebral H1-receptors and sedative properties of antihistamines. Assessment in the case of terfenadine.
Rose C; Quach TT; Llorens C; Schwartz JC
Arzneimittelforschung; 1982; 32(9a):1171-3. PubMed ID: 6129863
[TBL] [Abstract][Full Text] [Related]
11. Quantitative prediction of histamine H1 receptor occupancy by the sedative and non-sedative antagonists in the human central nervous system based on systemic exposure and preclinical data.
Kanamitsu K; Nozaki Y; Nagaya Y; Sugiyama Y; Kusuhara H
Drug Metab Pharmacokinet; 2017 Apr; 32(2):135-144. PubMed ID: 28190755
[TBL] [Abstract][Full Text] [Related]
12. Central effects of fexofenadine and cetirizine: measurement of psychomotor performance, subjective sleepiness, and brain histamine H1-receptor occupancy using 11C-doxepin positron emission tomography.
Tashiro M; Sakurada Y; Iwabuchi K; Mochizuki H; Kato M; Aoki M; Funaki Y; Itoh M; Iwata R; Wong DF; Yanai K
J Clin Pharmacol; 2004 Aug; 44(8):890-900. PubMed ID: 15286093
[TBL] [Abstract][Full Text] [Related]
13. Are antihistamines sedative via a blockade of brain H1 receptors?
Uzan A; Le Fur G; Malgouris C
J Pharm Pharmacol; 1979 Oct; 31(10):701-2. PubMed ID: 41044
[No Abstract] [Full Text] [Related]
14. New antihistamines: a critical view.
Camelo-Nunes IC
J Pediatr (Rio J); 2006 Nov; 82(5 Suppl):S173-80. PubMed ID: 17136293
[TBL] [Abstract][Full Text] [Related]
15. Variations among non-sedating antihistamines: are there real differences?
Mattila MJ; Paakkari I
Eur J Clin Pharmacol; 1999 Apr; 55(2):85-93. PubMed ID: 10335901
[TBL] [Abstract][Full Text] [Related]
16. [Molecular imaging of histamine receptors in the human brain].
Tashiro M; Yanai K
Brain Nerve; 2007 Mar; 59(3):221-31. PubMed ID: 17370648
[TBL] [Abstract][Full Text] [Related]
17. Computational Analysis of Structure-Based Interactions for Novel H₁-Antihistamines.
Yang Y; Li Y; Pan Y; Wang J; Lin F; Wang C; Zhang S; Yang L
Int J Mol Sci; 2016 Jan; 17(1):. PubMed ID: 26797608
[TBL] [Abstract][Full Text] [Related]
18. [Oral second generation antihistamines in allergic rhinitis].
Riechelmann H
Laryngorhinootologie; 2005 Jan; 84(1):30-41. PubMed ID: 15647976
[TBL] [Abstract][Full Text] [Related]
19. Roles of Lys191 and Lys179 in regulating thermodynamic binding forces of ligands to determine their binding affinity for human histamine H
Kobayashi C; Tanaka A; Yasuda T; Hishinuma S
Biochem Pharmacol; 2020 Oct; 180():114185. PubMed ID: 32738199
[TBL] [Abstract][Full Text] [Related]
20. Antihistamines for Allergic Rhinitis Treatment from the Viewpoint of Nonsedative Properties.
Kawauchi H; Yanai K; Wang DY; Itahashi K; Okubo K
Int J Mol Sci; 2019 Jan; 20(1):. PubMed ID: 30626077
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]